Structure-Based Design, Synthesis, and Biological Evaluation of Potent and Selective Macrocyclic Checkpoint Kinase 1 Inhibitors
Tao, Zhi-Fu, Wang, Le, Stewart, Kent D, Chen, Zehan, Gu, Wendy, Bui, Mai-Ha, Merta, Philip, Zhang, Haiying, Kovar, Peter, Johnson, Eric, Park, Chang, Judge, Russell, Rosenberg, Saul, Sowin, Thomas, Lin, Nan-Horng
Published in Journal of medicinal chemistry (05.04.2007)
Published in Journal of medicinal chemistry (05.04.2007)
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Journal Article
Design, Synthesis, and Biological Activity of 5,10-Dihydro-dibenzo[b,e][1,4]diazepin-11-one-Based Potent and Selective Chk-1 Inhibitors
Wang, Le, Sullivan, Gerard M, Hexamer, Laura A, Hasvold, Lisa A, Thalji, Reema, Przytulinska, Magdalena, Tao, Zhi-Fu, Li, Gaoquan, Chen, Zehan, Xiao, Zhan, Gu, Wen-Zhen, Xue, John, Bui, Mai-Ha, Merta, Philip, Kovar, Peter, Bouska, Jennifer J, Zhang, Haiying, Park, Chang, Stewart, Kent D, Sham, Hing L, Sowin, Thomas J, Rosenberg, Saul H, Lin, Nan-Horng
Published in Journal of medicinal chemistry (23.08.2007)
Published in Journal of medicinal chemistry (23.08.2007)
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Journal Article
Discovery of 4′-(1,4-dihydro-indeno[1,2- c]pyrazol-3-yl)-benzonitriles and 4′-(1,4-dihydro-indeno[1,2- c]pyrazol-3-yl)-pyridine-2′-carbonitriles as potent checkpoint kinase 1 (Chk1) inhibitors
Tao, Zhi-Fu, Li, Gaoquan, Tong, Yunsong, Stewart, Kent D., Chen, Zehan, Bui, Mai-Ha, Merta, Philip, Park, Chang, Kovar, Peter, Zhang, Haiying, Sham, Hing L., Rosenberg, Saul H., Sowin, Thomas J., Lin, Nan-Horng
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
Published in Bioorganic & medicinal chemistry letters (01.11.2007)
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1-Benzyl-3-cetyl-2-methylimidazolium iodide (NH125) induces phosphorylation of eukaryotic elongation factor-2 (eEF2): a cautionary note on the anticancer mechanism of an eEF2 kinase inhibitor
Chen, Zehan, Gopalakrishnan, Sujatha M, Bui, Mai-Ha, Soni, Niru B, Warrior, Usha, Johnson, Eric F, Donnelly, Jennifer B, Glaser, Keith B
Published in The Journal of biological chemistry (23.12.2011)
Published in The Journal of biological chemistry (23.12.2011)
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Journal Article
Reversing the Antibiotic Resistance "Yelp Effect" Through the Use of Emotionally Framed Responses to Negative Reviews of Providers: Questionnaire Study
Turner, Monique Mitchell, Choung, Hyesun, Bui, Quoc-Ha Hannah Mai, Beck, Paige, Ashraf, Hera
Published in JMIR formative research (22.03.2022)
Published in JMIR formative research (22.03.2022)
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PCR-Oligonucleotide Ligation Assay for Detection of Point Mutations Associated with Quinolone Resistance in Streptococcus pneumoniae
BUI, Mai-Ha, STONE, Gregory G, NILIUS, Angela M, ALMER, Laurel, FLAMM, Robert K
Published in Antimicrobial Agents and Chemotherapy (01.04.2003)
Published in Antimicrobial Agents and Chemotherapy (01.04.2003)
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Macrocyclic ureas as potent and selective Chk1 inhibitors: An improved synthesis, kinome profiling, structure–activity relationships, and preliminary pharmacokinetics
Tao, Zhi-Fu, Chen, Zehan, Bui, Mai-Ha, Kovar, Peter, Johnson, Eric, Bouska, Jennifer, Zhang, Haiying, Rosenberg, Saul, Sowin, Thomas, Lin, Nan-Horng
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
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Journal Article
Cyanopyridyl containing 1,4-dihydroindeno[1,2- c]pyrazoles as potent checkpoint kinase 1 inhibitors: Improving oral biovailability
Tong, Yunsong, Przytulinska, Magdalena, Tao, Zhi-Fu, Bouska, Jennifer, Stewart, Kent D., Park, Chang, Li, Gaoquan, Claiborne, Akiyo, Kovar, Peter, Chen, Zehan, Merta, Philip J., Bui, Mai-Ha, Olson, Amanda, Osterling, Donald, Zhang, Haiying, Sham, Hing L., Rosenberg, Saul H., Sowin, Thomas J., Lin, Nan-horng
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
Published in Bioorganic & medicinal chemistry letters (15.10.2007)
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Journal Article
Abstract 4960: First-in-class, highly BDII-selective BET family inhibitor ABBV-744 displays potent anti-tumor activity in androgen receptor positive prostate cancer models and an improved tolerability profile
Faivre, Emily J., Wilcox, Denise, Ha-Bui, Mai, Hessler, Paul, Sehgal, Vasudha, Lu, Xin, Uziel, Tamar, Mehta, Gaurav, Albert, Daniel H., McDaniel, Keith, Kati, Warren, Shen, Yu
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract 800: ABBV-744, a first-in-class and highly selective inhibitor of the second bromodomain of BET family proteins, displays robust activities in preclinical models of acute myelogenous leukemia
Lin, Xiaoyu, Huang, Xiaoli, Bellin, Richard, Faivre, Emily, Hessler, Paul, Lam, Lloyd, Bui, Mai Ha, Wilcox, Denise, Uziel, Tamar, Ferguson, Debra C., Magoc, Terrance J., Albert, Daniel H., McDaniel, Keith F., Kati, Warren, Shen, Yu
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract 931: Discovery of ABBV-744, a first-in-class highly BDII-selective BET bromodomain inhibitor
Sheppard, George S., Wang, Le, Fidanze, Steven D., Hasvold, Lisa A., Liu, Dachun, Pratt, John K., Park, Chang H., Bui, Mai-Ha, Faivre, Emily J., Huang, Xiaoli, Lin, Xiaoyu, Wilcox, Denise M., Shen, Yu, Albert, Daniel H., Magoc, Terrance J., Rajaraman, Ganesh, Kati, Warren M., McDaniel, Keith F.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Anhydrolide Macrolides. 2. Synthesis and Antibacterial Activity of 2,3-Anhydro-6-O-methyl 11,12-Carbazate Erythromycin A Analogues
Griesgraber, George, Kramer, Mark J, Elliott, Richard L, Nilius, Angela M, Ewing, Patty J, Raney, Patti M, Bui, Mai-Ha, Flamm, Robert K, Chu, Daniel T. W, Plattner, Jacob J, Or, Yat Sun
Published in Journal of medicinal chemistry (07.05.1998)
Published in Journal of medicinal chemistry (07.05.1998)
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Abstract 4706: ABBV-075 exhibits robust in vitro and in vivo activities against the ABC and GCB subtypes of DLBCL
Lin, Xiaoyu, Huang, Xiaoli, Sarthy, Aparna, Magoc, Terry, Albert, Daniel, Lam, Lloyd, Uziel, Tamar, Lu, Xin, Bui, Mai-Ha, Faivre, Emily, Wilcox, Denise, Elmore, Steven, McDaniel, Keith, Kati, Warren, Shen, Yu
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Anhydrolide Macrolides. 1. Synthesis and Antibacterial Activity of 2,3-Anhydro-6-O-methyl 11,12-Carbamate Erythromycin A Analogues
Elliott, Richard L, Pireh, Daisy, Griesgraber, George, Nilius, Angela M, Ewing, Patty J, Bui, Mai Ha, Raney, Patti M, Flamm, Robert K, Kim, Ki, Henry, Rodger F, Chu, Daniel T. W, Plattner, Jacob J, Or, Yat Sun
Published in Journal of medicinal chemistry (07.05.1998)
Published in Journal of medicinal chemistry (07.05.1998)
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1-Benzyl-3-cetyl-2-methylimidazolium iodide (NH125) Induces Phosphorylation of Eukaryotic Elongation Factor-2 (eEF2)
Chen, Zehan, Gopalakrishnan, Sujatha M., Bui, Mai-Ha, Soni, Niru B., Warrior, Usha, Johnson, Eric F., Donnelly, Jennifer B., Glaser, Keith B.
Published in The Journal of biological chemistry (23.12.2011)
Published in The Journal of biological chemistry (23.12.2011)
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Journal Article