Blocking Blood Flow to Solid Tumors by Destabilizing Tubulin: An Approach to Targeting Tumor Growth
Pérez-Pérez, María-Jesús, Priego, Eva-María, Bueno, Oskía, Martins, Maria Solange, Canela, María-Dolores, Liekens, Sandra
Published in Journal of medicinal chemistry (13.10.2016)
Published in Journal of medicinal chemistry (13.10.2016)
Get full text
Journal Article
High-affinity ligands of the colchicine domain in tubulin based on a structure-guided design
Bueno, Oskía, Estévez Gallego, Juan, Martins, Solange, Prota, Andrea E, Gago, Federico, Gómez-SanJuan, Asier, Camarasa, María-José, Barasoain, Isabel, Steinmetz, Michel O, Díaz, J Fernando, Pérez-Pérez, María-Jesús, Liekens, Sandra, Priego, Eva-María
Published in Scientific reports (09.03.2018)
Published in Scientific reports (09.03.2018)
Get full text
Journal Article
Antiviral activity of [1,2,3]triazolo[4,5-d]pyrimidin-7(6H)-ones against chikungunya virus targeting the viral capping nsP1
Gigante, Alba, Gómez-SanJuan, Asier, Delang, Leen, Li, Changqing, Bueno, Oskía, Gamo, Ana-María, Priego, Eva-María, Camarasa, María-José, Jochmans, Dirk, Leyssen, Pieter, Decroly, Etienne, Coutard, Bruno, Querat, Gilles, Neyts, Johan, Pérez-Pérez, María-Jesús
Published in Antiviral research (01.08.2017)
Published in Antiviral research (01.08.2017)
Get full text
Journal Article
Conformational mimetics of the α-methyl chalcone TUB091 binding tubulin: Design, synthesis and antiproliferative activity
Bueno, Oskía, Tobajas, Gloria, Quesada, Ernesto, Estévez-Gallego, Juan, Noppen, Sam, Camarasa, María-José, Díaz, José-Fernando, Liekens, Sandra, Priego, Eva-María, Pérez-Pérez, María-Jesús
Published in European journal of medicinal chemistry (25.03.2018)
Published in European journal of medicinal chemistry (25.03.2018)
Get full text
Journal Article
Antivascular and antitumor properties of the tubulin-binding chalcone TUB091
Canela, María-Dolores, Noppen, Sam, Bueno, Oskía, Prota, Andrea E, Bargsten, Katja, Sáez-Calvo, Gonzalo, Jimeno, María-Luisa, Benkheil, Mohammed, Ribatti, Domenico, Velázquez, Sonsoles, Camarasa, María-José, Díaz, J Fernando, Steinmetz, Michel O, Priego, Eva-María, Pérez-Pérez, María-Jesús, Liekens, Sandra
Published in Oncotarget (28.02.2017)
Published in Oncotarget (28.02.2017)
Get full text
Journal Article
Targeting the colchicine site in tubulin through cyclohexanedione derivatives
Canela, María-Dolores, Bueno, Oskía, Noppen, Sam, Sáez Calvo, Gonzalo, Estévez Gallego, Juan, Díaz, J. F., Camarasa, María-José, Liekens, Sandra, Pérez-Pérez, María-Jesús, Priego, Eva-María
Published in RSC advances (01.01.2016)
Published in RSC advances (01.01.2016)
Get full text
Journal Article
Targeting the colchicine site in tubulin through cyclohexanedione derivativesElectronic supplementary information (ESI) available. See DOI: 10.1039/c5ra26807a
Canela, María-Dolores, Bueno, Oskía, Noppen, Sam, Sáez Calvo, Gonzalo, Estévez Gallego, Juan, Díaz, J. F, Camarasa, María-José, Liekens, Sandra, Pérez-Pérez, María-Jesús, Priego, Eva-María
Year of Publication 16.02.2016
Year of Publication 16.02.2016
Get full text
Journal Article
Monitoring of PIK3CA and ESR1 mutations in circulating tumor DNA as predictive and prognostic biomarkers in patients with endocrine-resistant ER+/HER2- advanced breast cancer
Fuentes Antrás, Jesús, García-Barberán, Vanesa, Gonzalo, Irene, Moreno, Fernando, López-Cade, Igor, Ramírez-Ruda, Carmen, Bueno, Oskia, Ascaso del Rio, Ana, Pascual, Alejandro, Ocana, Alberto, Caldes, Trinidad, Garcia-Saenz, Jose Angel
Published in Journal of clinical oncology (20.05.2020)
Published in Journal of clinical oncology (20.05.2020)
Get full text
Journal Article
Diphenyl ether derivatives occupy the expanded binding site of cyclohexanedione compounds at the colchicine site in tubulin by movement of the αT5 loop
Bueno, Oskia, Gargantilla, Marta, Estévez-Gallego, Juan, Martins, Solange, Díaz, J. Fernando, Camarasa, María-José, Liekens, Sandra, Pérez-Pérez, María-Jesús, Priego, Eva-María
Published in European journal of medicinal chemistry (01.06.2019)
Published in European journal of medicinal chemistry (01.06.2019)
Get full text
Journal Article