Development of Tridentate Iron Chelators: From Desferrithiocin to ICL670
Nick, Hanspeter, Acklin, Pierre, Lattmann, René, Buehlmayer, Peter, Hauffe, Suzanne, Schupp, Joachim, Alberti, Daniele
Published in Current medicinal chemistry (01.06.2003)
Published in Current medicinal chemistry (01.06.2003)
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Journal Article
An Oral Sphingosine 1‑Phosphate Receptor 1 (S1P1) Antagonist Prodrug with Efficacy in Vivo: Discovery, Synthesis, and Evaluation
Angst, Daniela, Janser, Philipp, Quancard, Jean, Buehlmayer, Peter, Berst, Frederic, Oberer, Lukas, Beerli, Christian, Streiff, Markus, Pally, Charles, Hersperger, Rene, Bruns, Christian, Bassilana, Frederic, Bollbuck, Birgit
Published in Journal of medicinal chemistry (26.11.2012)
Published in Journal of medicinal chemistry (26.11.2012)
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Journal Article
Synthesis and biological activity of some transition-state inhibitors of human renin
Buehlmayer, Peter, Caselli, Anthony, Fuhrer, Walter, Goeschke, Richard, Rasetti, Vittorio, Rueger, Heinrich, Stanton, James L, Criscione, Leoluca, Wood, Jeanette M
Published in Journal of medicinal chemistry (01.09.1988)
Published in Journal of medicinal chemistry (01.09.1988)
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Journal Article
Syk inhibitors with high potency in presence of blood
Thoma, Gebhard, Blanz, Joachim, Bühlmayer, Peter, Drückes, Peter, Kittelmann, Matthias, Smith, Alexander B., van Eis, Maurice, Vangrevelinghe, Eric, Zerwes, Hans-Günter, Che, Jianwei (John), He, Xiaohui, Jin, Yunho, Lee, Christian C., Michellys, Pierre-Yves, Uno, Tetsuo, Liu, Hong
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
Published in Bioorganic & medicinal chemistry letters (15.05.2014)
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Journal Article
Nonpeptidic angiotensin II antagonists: synthesis and in vitro activity of a series of novel naphthalene and tetrahydronaphthalene derivatives
Buehlmayer, Peter, Criscione, Leoluca, Fuhrer, Walter, Furet, Pascal, De Gasparo, Marc, Stutz, Stefan, Whitebread, Steven
Published in Journal of medicinal chemistry (01.10.1991)
Published in Journal of medicinal chemistry (01.10.1991)
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Journal Article
New pyrazolo[1,5a]pyrimidines as orally active inhibitors of Lck
Gommermann, Nina, Buehlmayer, Peter, von Matt, Anette, Breitenstein, Werner, Masuya, Keiichi, Pirard, Bernard, Furet, Pascal, Cowan-Jacob, Sandra W., Weckbecker, Gisbert
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Journal Article
Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-thia-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists
Rueeger, Heinrich, Gerspacher, Marc, Buehlmayer, Peter, Rigollier, Pascal, Yamaguchi, Yasuchika, Schmidlin, Tibur, Whitebread, Steven, Nuesslein-Hildesheim, Barbara, Nick, Hanspeter, Cricione, Leoluca
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
Published in Bioorganic & medicinal chemistry letters (17.05.2004)
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Journal Article
PYRAZOLO[1,5-A]PYRIMIDINE DERIVATIVES AND THEIR THERAPEUTIC USE
VON MATT ANETTE, PIRARD BERNARD, FURET PASCAL, ZOLLER THOMAS, BUEHLMAYER PETER, BREITENSTEIN WERNER
Year of Publication 02.07.2009
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Year of Publication 02.07.2009
Patent
Synthesis of chiral analogues of FTY720 and its phosphate
Hinterding, K, Cottens, S, Albert, R, Zecri, F, Buehlmayer, PB, Spanka, C, Brinkmann, Nussbaumer, P, Ettmayer, P, Hoegenauer, K, Gray, N, Pan, SF
Published in Synthesis (Stuttgart) (01.01.2003)
Published in Synthesis (Stuttgart) (01.01.2003)
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Journal Article
Development of tridentate iron chelators: From desferrithiocin to ICL670: Iron Chelation and Human Diseases
NICK, Hanspeter, ACKLIN, Pierre, LATTMANN, René, BUEHLMAYER, Peter, HAUFFE, Suzanne, SCHUPP, Joachim, ALBERTI, Daniele
Published in Current medicinal chemistry (2003)
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Published in Current medicinal chemistry (2003)
Journal Article
A Potent and Selective S1P1 Antagonist with Efficacy in Experimental Autoimmune Encephalomyelitis
Quancard, Jean, Bollbuck, Birgit, Janser, Philipp, Angst, Daniela, Berst, Frédéric, Buehlmayer, Peter, Streiff, Markus, Beerli, Christian, Brinkmann, Volker, Guerini, Danilo, Smith, Paul A., Seabrook, Timothy J., Traebert, Martin, Seuwen, Klaus, Hersperger, René, Bruns, Christian, Bassilana, Frédéric, Bigaud, Marc
Published in Chemistry & biology (21.09.2012)
Published in Chemistry & biology (21.09.2012)
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Journal Article
A potent and selective S1P(1) antagonist with efficacy in experimental autoimmune encephalomyelitis
Quancard, Jean, Bollbuck, Birgit, Janser, Philipp, Angst, Daniela, Berst, Frédéric, Buehlmayer, Peter, Streiff, Markus, Beerli, Christian, Brinkmann, Volker, Guerini, Danilo, Smith, Paul A, Seabrook, Timothy J, Traebert, Martin, Seuwen, Klaus, Hersperger, René, Bruns, Christian, Bassilana, Frédéric, Bigaud, Marc
Published in Chemistry & biology (21.09.2012)
Published in Chemistry & biology (21.09.2012)
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Journal Article
BICYCLIC HETEROARYL CYCLOALKYLDIAMINE DERIVATIVES AS INHIBITORS OF SPLEEN TYROSINE KINASES (SYK)
SMITH, ALEXANDER BAXTER, THOMA, GEBHARD, BUEHLMAYER, PETER, VAN EIS, MAURICE
Year of Publication 08.09.2020
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Year of Publication 08.09.2020
Patent
Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4H-3-this-1-aza-benzo[e]azulen- and 4,5-dihydro-6-oxa-3-this-1-aza-benzo[e]azulen derivatives as neuropeptide Y Y5 receptor antagonists
RUEEGER, Heinrich, GERSPACHER, Marc, BUEHLMAYER, Peter, RIGOLLIER, Pascal, YAMAGUCHI, Yasuchika, SCHMIDLIN, Tibur, WHITEBREAD, Steven, NUESSLEIN-HILDESHEIM, Barbara, NICK, Hanspeter, CRICIONE, Leoluca
Published in Bioorganic & medicinal chemistry letters (2004)
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Published in Bioorganic & medicinal chemistry letters (2004)
Journal Article
Discovery and SAR of potent, orally available and brain-penetrable 5,6-dihydro-4 H-3-thia-1-aza-benzo[ e]azulen- and 4,5-dihydro-6-oxa-3-thia-1-aza-benzo[ e]azulen derivatives as neuropeptide Y Y5 receptor antagonists
Rueeger, Heinrich, Gerspacher, Marc, Buehlmayer, Peter, Rigollier, Pascal, Yamaguchi, Yasuchika, Schmidlin, Tibur, Whitebread, Steven, Nuesslein-Hildesheim, Barbara, Nick, Hanspeter, Cricione, Leoluca
Published in Bioorganic & medicinal chemistry letters (2004)
Published in Bioorganic & medicinal chemistry letters (2004)
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Journal Article
BICYCLIC HETEROARYL CYCLOALKYLDIAMINE DERIVATIVES AS INHIBITORS OF SPLEEN TYROSINE KINASES (SYK)
Smith Alexander Baxter, Buehlmayer Peter, Thoma Gebhard, Van Eis Maurice
Year of Publication 28.07.2016
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Year of Publication 28.07.2016
Patent
BICYCLIC HETEROARYL CYCLOALKYLDIAMINE DERIVATIVES AS INHIBITORS OF SPLEEN TYROSINE KINASES (SYK)
SMITH, ALEXANDER BAXTER, THOMA, GEBHARD, BUEHLMAYER, PETER, VAN EIS, MAURICE
Year of Publication 27.04.2016
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Year of Publication 27.04.2016
Patent
Bicyclic heteroaryl cycloalkyldiamine derivatives
THOMA GEBHARD, SMITH ALEXANDER BAXTER, BUEHLMAYER PETER, VAN EIS MAURICE
Year of Publication 19.04.2016
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Year of Publication 19.04.2016
Patent