Adenosine analogues as inhibitors of Trypanosoma brucei phosphoglycerate kinase: Elucidation of a novel binding mode for a 2-amino-N-6-substituted adenosine
Bressi, JC, Choe, J, Hough, MT, Buckner, FS, Van Voorhis, WC, Verlinde, CLMJ, Hol, WGJ, Gelb, MH
Published in Journal of medicinal chemistry (02.11.2000)
Published in Journal of medicinal chemistry (02.11.2000)
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Journal Article
Design and Synthesis of Peptidomimetic Protein Farnesyltransferase Inhibitors as Anti-Trypanosoma brucei Agents
Ohkanda, Junko, Buckner, Frederick S, Lockman, Jeffrey W, Yokoyama, Kohei, Carrico, Dora, Eastman, Richard, de Luca-Fradley, Kate, Davies, Wendy, Croft, Simon L, Van Voorhis, Wesley C, Gelb, Michael H, Sebti, Saïd M, Hamilton, Andrew D
Published in Journal of medicinal chemistry (15.01.2004)
Published in Journal of medicinal chemistry (15.01.2004)
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Journal Article
Structurally Simple Farnesyltransferase Inhibitors Arrest the Growth of Malaria Parasites
Glenn, Matthew P., Chang, Sung-Youn, Hucke, Oliver, Verlinde, Christophe L. M. J., Rivas, Kasey, Hornéy, Carrie, Yokoyama, Kohei, Buckner, Frederick S., Pendyala, Prakash R., Chakrabarti, Debopam, Gelb, Michael, Van Voorhis, Wesley C., Sebti, Saïd M., Hamilton, Andrew D.
Published in Angewandte Chemie (International ed.) (05.08.2005)
Published in Angewandte Chemie (International ed.) (05.08.2005)
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Journal Article
In vitro and in vivo antimalarial activity of peptidomimetic protein farnesyltransferase inhibitors with improved membrane permeability
Carrico, Dora, Ohkanda, Junko, Kendrick, Howard, Yokoyama, Kohei, Blaskovich, Michelle A., Bucher, Cynthia J., Buckner, Frederick S., Van Voorhis, Wesley C., Chakrabarti, Debopam, Croft, Simon L., Gelb, Michael H., Sebti, Saïd M., Hamilton, Andrew D.
Published in Bioorganic & medicinal chemistry (15.12.2004)
Published in Bioorganic & medicinal chemistry (15.12.2004)
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Journal Article
Oxidosqualene Cyclase Inhibitors as Antimicrobial Agents
Hinshaw, Jerald C, Suh, Dae-Yeon, Garnier, Philippe, Buckner, Frederick S, Eastman, Richard T, Matsuda, Seiichi P. T, Joubert, Bridget M, Coppens, Isabelle, Joiner, Keith A, Merali, Salim, Nash, Theodore E, Prestwich, Glenn D
Published in Journal of medicinal chemistry (25.09.2003)
Published in Journal of medicinal chemistry (25.09.2003)
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Journal Article
TcRho1, a Farnesylated Rho Family Homologue from Trypanosoma cruzi
José L. Nepomuceno-Silva, Kohei Yokoyama, Luiz D. B. de Mello, Sérgio M. Mendonça, Júlio C. Paixão, Rudi Baron, Jean-Charles Faye, Frederick S. Buckner, Wesley C. Van Voorhis, Michael H. Gelb, Ulisses G. Lopes
Published in The Journal of biological chemistry (10.08.2001)
Published in The Journal of biological chemistry (10.08.2001)
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Journal Article
Isothiazole dioxides: synthesis and inhibition of Trypanosoma brucei protein farnesyltransferase
Clerici, Francesca, Gelmi, Maria Luisa, Yokoyama, Kohei, Pocar, Donato, Van Voorhis, Wesley C., Buckner, Frederick S., Gelb, Michael H.
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
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Journal Article
The First Impeachment: The Constitution's Framers and the Case of Senator William Blount
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Book Review
Journal Article
Structure of ribose 5-phosphate isomerase from Plasmodium falciparum
Boni, Erica, Luft, Joseph, Holmes, Margaret A., Buckner, Frederick S., Van Voorhis, Wesley C., Verlinde, Christophe L. M. J., Mehlin, Christopher, DeTitta, George, Lauricella, Angela, Anderson, Lori, Kalyuzhniy, Oleksandr, Zucker, Frank, Schoenfeld, Lori W., Earnest, Thomas N., Hol, Wim G. J., Merritt, Ethan A.
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2006)
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.05.2006)
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Journal Article
Protein structure-based design of anti-protozoal drugs
Verlinde, Christophe L. M. J., Bressi, Jerome C., Choe, Jungwoo, Suresh, Stephen, Buckner, Frederick S., Van Voorhis, Wesley C., Michels, Paul A. M., Gelb, Michael H., Hol, Wim G. J.
Published in Journal of the Brazilian Chemical Society (01.11.2002)
Published in Journal of the Brazilian Chemical Society (01.11.2002)
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Journal Article
Structure of the conserved hypothetical protein MAL13P1.257 from Plasmodium falciparum
Holmes, Margaret A., Buckner, Frederick S., Van Voorhis, Wesley C., Mehlin, Christopher, Boni, Erica, Earnest, Thomas N., DeTitta, George, Luft, Joseph, Lauricella, Angela, Anderson, Lori, Kalyuzhniy, Oleksandr, Zucker, Frank, Schoenfeld, Lori W., Hol, Wim G. J., Merritt, Ethan A.
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.03.2006)
Published in Acta crystallographica. Section F, Structural biology and crystallization communications (01.03.2006)
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