Structural Modeling of TRPA1 Ion Channel-Determination of the Binding Site for Antagonists
Gawalska, Alicja, Kołaczkowski, Marcin, Bucki, Adam
Published in Molecules (Basel, Switzerland) (11.05.2022)
Published in Molecules (Basel, Switzerland) (11.05.2022)
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Metabolic carbonyl reduction of anthracyclines — role in cardiotoxicity and cancer resistance. Reducing enzymes as putative targets for novel cardioprotective and chemosensitizing agents
Piska, Kamil, Koczurkiewicz, Paulina, Bucki, Adam, Wójcik-Pszczoła, Katarzyna, Kołaczkowski, Marcin, Pękala, Elżbieta
Published in Investigational new drugs (01.06.2017)
Published in Investigational new drugs (01.06.2017)
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Advances in Discovery of PDE10A Inhibitors for CNS-Related Disorders. Part 1: Overview of the Chemical and Biological Research
Jankowska, Agnieszka, Świerczek, Artur, Wyska, Elżbieta, Gawalska, Alicja, Bucki, Adam, Pawłowski, Maciej, Chłoń-Rzepa, Grażyna
Published in Current drug targets (01.01.2019)
Published in Current drug targets (01.01.2019)
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In Silico and In Vitro Assessment of Carbonyl Reductase 1 Inhibition Using ASP9521-A Potent Aldo-Keto Reductase 1C3 Inhibitor with the Potential to Support Anticancer Therapy Using Anthracycline Antibiotics
Jamrozik, Marek, Piska, Kamil, Bucki, Adam, Koczurkiewicz-Adamczyk, Paulina, Sapa, Michał, Władyka, Benedykt, Pękala, Elżbieta, Kołaczkowski, Marcin
Published in Molecules (Basel, Switzerland) (27.04.2023)
Published in Molecules (Basel, Switzerland) (27.04.2023)
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Serotonin 5-HT6 Receptor Ligands and Butyrylcholinesterase Inhibitors Displaying Antioxidant Activity—Design, Synthesis and Biological Evaluation of Multifunctional Agents against Alzheimer’s Disease
Więckowski, Krzysztof, Szałaj, Natalia, Gryzło, Beata, Wichur, Tomasz, Góral, Izabella, Sługocka, Emilia, Sniecikowska, Joanna, Latacz, Gniewomir, Siwek, Agata, Godyń, Justyna, Bucki, Adam, Kołaczkowski, Marcin, Więckowska, Anna
Published in International journal of molecular sciences (21.08.2022)
Published in International journal of molecular sciences (21.08.2022)
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Impact of N-Alkylamino Substituents on Serotonin Receptor (5-HTR) Affinity and Phosphodiesterase 10A (PDE10A) Inhibition of Isoindole-1,3-dione Derivatives
Czopek, Anna, Partyka, Anna, Bucki, Adam, Pawłowski, Maciej, Kołaczkowski, Marcin, Siwek, Agata, Głuch-Lutwin, Monika, Koczurkiewicz, Paulina, Pękala, Elżbieta, Jaromin, Anna, Tyliszczak, Bożena, Wesołowska, Anna, Zagórska, Agnieszka
Published in Molecules (Basel, Switzerland) (25.08.2020)
Published in Molecules (Basel, Switzerland) (25.08.2020)
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Neuroprotective Activity of Enantiomers of Salsolinol and N‑Methyl‑(R)‑salsolinol: In Vitro and In Silico Studies
Kurnik-Łucka, Magdalena, Latacz, Gniewomir, Bucki, Adam, Rivera-Meza, Mario, Khan, Nadia, Konwar, Jahnobi, Skowron, Kamil, Kołaczkowski, Marcin, Gil, Krzysztof
Published in ACS omega (17.10.2023)
Published in ACS omega (17.10.2023)
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Synthesis and biological evaluation of N-arylpiperazine derivatives of 4,4-dimethylisoquinoline-1,3(2H,4H)-dione as potential antiplatelet agents
Marcinkowska, Monika, Kotańska, Magdalena, Zagórska, Agnieszka, Śniecikowska, Joanna, Kubacka, Monika, Siwek, Agata, Bucki, Adam, Pawłowski, Maciej, Bednarski, Marek, Sapa, Jacek, Starek, Małgorzata, Dąbrowska, Monika, Kołaczkowski, Marcin
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2018)
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Rapid erosion of soft sediments by tidewater glacier advance: Taku Glacier, Alaska, USA
Motyka, Roman J., Truffer, Martin, Kuriger, Elsbeth M., Bucki, Adam K.
Published in Geophysical research letters (01.12.2006)
Published in Geophysical research letters (01.12.2006)
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Application of automated machine learning in the identification of multi‐target‐directed ligands blocking PDE4B, PDE8A, and TRPA1 with potential use in the treatment of asthma and COPD
Gawalska, Alicja, Czub, Natalia, Sapa, Michał, Kołaczkowski, Marcin, Bucki, Adam, Mendyk, Aleksander
Published in Molecular informatics (01.07.2023)
Published in Molecular informatics (01.07.2023)
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Comparative study on ABCB1-dependent efflux of anthracyclines and their metabolites: consequences for cancer resistance
Piska, Kamil, Koczurkiewicz-Adamczyk, Paulina, Jamrozik, Marek, Bucki, Adam, Kołaczkowski, Marcin, Pękala, Elżbieta
Published in Xenobiotica (03.07.2023)
Published in Xenobiotica (03.07.2023)
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Novel drug-like fluorenyl derivatives as selective butyrylcholinesterase and β-amyloid inhibitors for the treatment of Alzheimer’s disease
Pasieka, Anna, Panek, Dawid, Zaręba, Paula, Sługocka, Emilia, Gucwa, Natalia, Espargaró, Alba, Latacz, Gniewomir, Khan, Nadia, Bucki, Adam, Sabaté, Raimon, Więckowska, Anna, Malawska, Barbara
Published in Bioorganic & medicinal chemistry (06.06.2023)
Published in Bioorganic & medicinal chemistry (06.06.2023)
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Idalopirdine, a selective 5-HT6 receptor antagonist, reduces food intake and body weight in a model of excessive eating
Kotańska, Magdalena, Lustyk, Klaudia, Bucki, Adam, Marcinkowska, Monika, Śniecikowska, Joanna, Kołaczkowski, Marcin
Published in Metabolic brain disease (01.06.2018)
Published in Metabolic brain disease (01.06.2018)
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Novel serotonin 5-HT 2A receptor antagonists derived from 4-phenylcyclohexane-5-spiro-and 5-methyl-5-phenyl-hydantoin, for use as potential antiplatelet agents
Czopek, Anna, Kubacka, Monika, Bucki, Adam, Siwek, Agata, Filipek, Barbara, Pawłowski, Maciej, Kołaczkowski, Marcin
Published in Pharmacological reports (01.10.2021)
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Published in Pharmacological reports (01.10.2021)
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