Functionalization of Planar Chiral Fused Arene Ruthenium Complexes: Synthesis, X-ray Structures, and Spectroscopic Characterization of Monodentate Triarylphosphines
Buchgraber, Philipp, Mercier, Audrey, Yeo, Wee Chuan, Besnard, Céline, Kündig, E. Peter
Published in Organometallics (28.11.2011)
Published in Organometallics (28.11.2011)
Get full text
Journal Article
Discovery of YAP1/TAZ pathway inhibitors through phenotypic screening with potent anti-tumor activity via blockade of Rho-GTPase signaling
Graham, Keith, Lienau, Philip, Bader, Benjamin, Prechtl, Stefan, Naujoks, Jan, Lesche, Ralf, Weiske, Joerg, Kuehnlenz, Julia, Brzezinka, Krzysztof, Potze, Lisette, Zanconato, Francesca, Nicke, Barbara, Montebaur, Anna, Bone, Wilhelm, Golfier, Sven, Kaulfuss, Stefan, Kopitz, Charlotte, Pilari, Sabine, Steuber, Holger, Hayat, Sikander, Kamburov, Atanas, Steffen, Andreas, Schlicker, Andreas, Buchgraber, Philipp, Braeuer, Nico, Font, Nuria Aiguabella, Heinrich, Tobias, Kuhnke, Lara, Nowak-Reppel, Katrin, Stresemann, Carlo, Steigemann, Patrick, Walter, Annette O., Blotta, Simona, Ocker, Matthias, Lakner, Ashley, von Nussbaum, Franz, Mumberg, Dominik, Eis, Knut, Piccolo, Stefano, Lange, Martin
Published in Cell chemical biology (18.07.2024)
Published in Cell chemical biology (18.07.2024)
Get full text
Journal Article
New Generation of sGC Stimulators: Discovery of Imidazo[1,2‑a]pyridine Carboxamide BAY 1165747 (BAY-747), a Long-Acting Soluble Guanylate Cyclase Stimulator for the Treatment of Resistant Hypertension
Vakalopoulos, Alexandros, Wunder, Frank, Hartung, Ingo V., Redlich, Gorden, Jautelat, Rolf, Buchgraber, Philipp, Hassfeld, Jorma, Gromov, Alexey V., Lindner, Niels, Bierer, Donald, Gries, Jörg, Kroh, Walter, Paulsen, Holger, Mittendorf, Joachim, Lang, Dieter, Becker-Pelster, Eva, Brockschnieder, Damian, Geiss, Volker, Li, Volkhart, Straub, Alexander, Knorr, Andreas, Mondritzki, Thomas, Trübel, Hubert, Raschke, Marian, Schaefer, Martina, Thomas, Dirk, Sandner, Peter, Stasch, Johannes-Peter, Follmann, Markus
Published in Journal of medicinal chemistry (08.06.2023)
Published in Journal of medicinal chemistry (08.06.2023)
Get full text
Journal Article
BAY-8400: A Novel Potent and Selective DNA-PK Inhibitor which Shows Synergistic Efficacy in Combination with Targeted Alpha Therapies
Berger, Markus, Wortmann, Lars, Buchgraber, Philipp, Lücking, Ulrich, Zitzmann-Kolbe, Sabine, Wengner, Antje M, Bader, Benjamin, Bömer, Ulf, Briem, Hans, Eis, Knut, Rehwinkel, Hartmut, Bartels, Florian, Moosmayer, Dieter, Eberspächer, Uwe, Lienau, Philip, Hammer, Stefanie, Schatz, Christoph A, Wang, Qiuwen, Wang, Qi, Mumberg, Dominik, Nising, Carl F, Siemeister, Gerhard
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
Get full text
Journal Article
Total Synthesis of Berkelic Acid
Snaddon, Thomas N., Buchgraber, Philipp, Schulthoff, Saskia, Wirtz, Conny, Mynott, Richard, Fürstner, Alois
Published in Chemistry : a European journal (25.10.2010)
Published in Chemistry : a European journal (25.10.2010)
Get full text
Journal Article
Synthesis-driven mapping of the dictyodendrin alkaloids
Buchgraber, Philipp, Domostoj, Mathias M., Scheiper, Bodo, Wirtz, Conny, Mynott, Richard, Rust, Jörg, Fürstner, Alois
Published in Tetrahedron (15.08.2009)
Published in Tetrahedron (15.08.2009)
Get full text
Journal Article
Synthesis-Driven Structure Revision of Berkelic Acid Methyl Ester
Buchgraber, Philipp, Snaddon, Thomas N, Wirtz, Conny, Mynott, Richard, Goddard, Richard, Fürstner, Alois
Published in Angewandte Chemie (International ed.) (20.10.2008)
Published in Angewandte Chemie (International ed.) (20.10.2008)
Get full text
Journal Article
Abstract 4584: Novel YAP1/TAZ pathway inhibitors identified through phenotypic screening with potent anti-tumor activity via blockade of GGTase-I and Rho-GTPase signaling
Graham, Keith, Lienau, Philip, Bader, Benjamin, Prechtl, Stefan, Naujoks, Jan, Lesche, Ralf, Nicke, Barbara, Bone, Wilhelm, Golfier, Sven, Brzezinka, Krzysztof, Kaulfuss, Stefan, Kopitz, Charlotte, Steuber, Holger, Braeuer, Nico, Nowak-Reppel, Katrin, Stresemann, Carlo, Steigemann, Patrick, Kuehnlenz, Julia, Potze, Lisette, Zanconato, Francesca, Montebaur, Anna, Pilari, Sabine, Hayat, Sikander, Kamburov, Atanas, Steffen, Andreas, Schlicker, Andreas, Buchgraber, Philipp, Font, Nuria Aiguabella, Heinrich, Tobias, Kuhnke, Lara, Walter, Annette O., Blotta, Simona, Ocker, Matthias, Lakner, Ashley, Mumberg, Dominik, Eis, Knut, Piccolo, Stefano, Lange, Martin
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Get full text
Journal Article
아드레날린수용체 ADRAC2의 억제제
DELBECK MARTINA, DIETZ LISA, BUCHGRABER PHILIPP, MEIBOM DANIEL, PLATZK MAGDALENA, BECKER PELSTER EVA MARIA, HAHN MICHAEL, MUELLER THOMAS, SCHMECK CARSTEN, LINDNER NIELS
Year of Publication 11.07.2022
Get full text
Year of Publication 11.07.2022
Patent
Synthesis-driven mapping of the dictyodendrin alkaloids: 2008 Tetrahedron Prize for Creativity in Organic Chemistry. The Art of Synthesis: Methods, Strategies and Applications
BUCHGRABER, Philipp, DOMOSTOJ, Mathias M, SCHEIPER, Bodo, WIRTZ, Conny, MYNOTT, Richard, RUST, Jörg, FÜRSTNER, Alois
Published in Tetrahedron (2009)
Get full text
Published in Tetrahedron (2009)
Journal Article
아미도-치환된 시클로헥산 유도체
SIEGEL FRANZISKA, LIENAU PHILIP, KOPPITZ MARCUS, BUCHGRABER PHILIPP, BENDER ECKHARD, VON NUSSBAUM FRANZ, LIU NINGSHU, EIS KNUT, SUELZLE DETLEV, BAIRLEIN MICHAELA, LI VOLKHART, ACKERSTAFF JENS, WAGNER SARAH, HOLTON SIMON, HERBERT SIMON ANTHONY
Year of Publication 08.01.2018
Get full text
Year of Publication 08.01.2018
Patent
TNKS1 / TNKS2 - AMIDO-SUBSTITUTED AZOLE COMPOUNDS AS INHIBITORS OF TNKS1 AND/OR TNKS2
LIENAU PHILIP, SIEGEL FRANZISKA, GOLZ STEFAN, BENDER ECKHARD, BUCHGRABER PHILIPP, LIU NINGSHU, EIS KNUT, BAUSER MARCUS, SUELZLE DETLEV, BAIRLEIN MICHAELA, ACKERSTAFF JENS, WAGNER SARAH, BASTING DANIEL, HOLTON SIMON, LI VOLKHART MIN JIAN, BALINT JOZSEF
Year of Publication 21.11.2016
Get full text
Year of Publication 21.11.2016
Patent
SUBSTITUTED PIPERIDINYL-TETRAHYDROQUINOLINES
KAST RAIMUND, GOELLER ANDREAS, KNORR ANDREAS, LANG DIETER, BUCHGRABER PHILIPP, BECKER PELSTER EVA MARIA, ENGEL KAREN, HIMMEL HERBERT, WUNDER FRANK, REDLICH GORDEN, TINEL HANNA, BUCHMUELLER ANJA, SCHMECK CARSTEN, GEISS VOLKER
Year of Publication 18.08.2016
Get full text
Year of Publication 18.08.2016
Patent
SUBSTITUTED PIPERIDINYL-TETRAHYDROQUINOLINES AND THEIR USE AS ALPHA-2C ADRENORECEPTOR ANTAGONISTS
KAST RAIMUND, GOELLER ANDREAS, KNORR ANDREAS, LANG DIETER, BUCHGRABER PHILIPP, BECKER PELSTER EVA MARIA, ENGEL KAREN, HIMMEL HERBERT, WUNDER FRANK, REDLICH GORDEN, TINEL HANNA, BUCHMUELLER ANJA, SCHMECK CARSTEN, GEISS VOLKER
Year of Publication 18.08.2016
Get full text
Year of Publication 18.08.2016
Patent
AMINO-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINECARBOXAMIDES AND THEIR USE
KNORR ANDREAS, BUCHGRABER PHILIPP, JAUTELAT ROLF, BECKER PELSTER EVA MARIA, FOLLMANN MARKUS, LINDNER NIELS, WUNDER FRANK, REDLICH GORDEN, HARTUNG INGO, VAKALOPOULOS ALEXANDROS, GROMOV ALEXEY, LI VOLKHART MIN JIAN, HASSFELD JORMA
Year of Publication 13.07.2015
Get full text
Year of Publication 13.07.2015
Patent
A Synthesis-Driven Structure Revision of Berkelic Acid Methyl Ester
Buchgraber, Philipp, Snaddon, Thomas N., Wirtz, Conny, Mynott, Richard, Goddard, Richard, Fürstner, Alois
Published in Angewandte Chemie (20.10.2008)
Published in Angewandte Chemie (20.10.2008)
Get full text
Journal Article
INHIBITORS OF ADRENORECEPTOR ADRAC2
BECKER-PELSTER, Eva Maria, DIETZ, Lisa, LINDNER, Niels, MÜLLER, Thomas, SCHMECK, Carsten, MEIBOM, Daniel, BUCHGRABER, Philipp, PLATZK, Magdalena, HAHN, Michael, DELBECK, Martina
Year of Publication 10.07.2024
Get full text
Year of Publication 10.07.2024
Patent
BICYCLIC TRIAZINE DERIVATIVES FOR THE TREATMENT OF CANCER
STEIGEMANN, Patrick, THEDE, Kai, BUCHGRABER, Philipp, DIETER, Sebastian, WENGNER, Antje Margret, KRETH, Sina, LIENAU, Philip, HERBST-NOWROUZI, Friederike, SIEMEISTER, Gerhard, BÖMER, Ulf, GLIMM, Hanno, WESTERMANN, Frank
Year of Publication 04.07.2024
Get full text
Year of Publication 04.07.2024
Patent