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Identification and Preclinical Development of a 2,5,6-Trisubstituted Fluorinated Pyridine Derivative as a Radioligand for the Positron Emission Tomography Imaging of Cannabinoid Type 2 Receptors
Haider, Achi, Gobbi, Luca, Kretz, Julian, Ullmer, Christoph, Brink, Andreas, Honer, Michael, Woltering, Thomas J., Muri, Dieter, Iding, Hans, Bürkler, Markus, Binder, Martin, Bartelmus, Christian, Knuesel, Irene, Pacher, Pal, Herde, Adrienne Müller, Spinelli, Francesco, Ahmed, Hazem, Atz, Kenneth, Keller, Claudia, Weber, Markus, Schibli, Roger, Mu, Linjing, Grether, Uwe, Ametamey, Simon M.
Published in Journal of medicinal chemistry (24.09.2020)
Published in Journal of medicinal chemistry (24.09.2020)
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Structure–Activity Relationship Studies of Pyridine-Based Ligands and Identification of a Fluorinated Derivative for Positron Emission Tomography Imaging of Cannabinoid Type 2 Receptors
Haider, Achi, Kretz, Julian, Gobbi, Luca, Ahmed, Hazem, Atz, Kenneth, Bürkler, Markus, Bartelmus, Christian, Fingerle, Jürgen, Guba, Wolfgang, Ullmer, Christoph, Honer, Michael, Knuesel, Irene, Weber, Markus, Brink, Andreas, Herde, Adrienne Müller, Keller, Claudia, Schibli, Roger, Mu, Linjing, Grether, Uwe, Ametamey, Simon M.
Published in Journal of medicinal chemistry (26.12.2019)
Published in Journal of medicinal chemistry (26.12.2019)
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Structure-Guided Discovery of cis-Hexahydro-pyrido-oxazinones as Reversible, Drug-like Monoacylglycerol Lipase Inhibitors
Kuhn, Bernd, Ritter, Martin, Hornsperger, Benoit, Bell, Charles, Kocer, Buelent, Rombach, Didier, Lutz, Marius D. R., Gobbi, Luca, Kuratli, Martin, Bartelmus, Christian, Bürkler, Markus, Koller, Raffael, Tosatti, Paolo, Ruf, Iris, Guerard, Melanie, Pavlovic, Anto, Stephanus, Juliane, O’Hara, Fionn, Wetzl, Dennis, Saal, Wiebke, Stihle, Martine, Roth, Doris, Hug, Melanie, Huber, Sylwia, Heer, Dominik, Kroll, Carsten, Topp, Andreas, Schneider, Manfred, Gertsch, Jürg, Glasmacher, Sandra, van der Stelt, Mario, Martella, Andrea, Wittwer, Matthias Beat, Collin, Ludovic, Benz, Jörg, Richter, Hans, Grether, Uwe
Published in Journal of medicinal chemistry (24.10.2024)
Published in Journal of medicinal chemistry (24.10.2024)
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Synthesis of potential drug metabolites by a modified Udenfriend reaction
Slavik, Roger, Peters, Jens-Uwe, Giger, Rudolf, Bürkler, Markus, Bald, Eric
Published in Tetrahedron letters (16.02.2011)
Published in Tetrahedron letters (16.02.2011)
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Expediting hit-to-lead progression in drug discovery through reaction prediction and multi-objective molecular optimization
Nippa, David F., Atz, Kenneth, Stenzhorn, Yannick, Müller, Alex T., Tosstorff, Andreas, Benz, Jörg, Binch, Hayley, Bürkler, Markus, Haider, Achi, Heer, Dominik, Hochstrasser, Remo, Kramer, Christian, Reutlinger, Michael, Schneider, Petra, Shema, Thierry, Topp, Andreas, Walter, Alexander, Wittwer, Matthias B., Wolfard, Jens, Kuhn, Bernd, van der Stelt, Mario, Martin, Rainer E., Grether, Uwe, Schneider, Gisbert
Published in ChemRxiv
Published in ChemRxiv
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METHOD AND DEVICE FOR CALIBRATING LIQUID METERS
SCHOLL, RALPH THORSTEN, BUERKLER, MARKUS, THORN, FRANK, MAIER, ANDREAS
Year of Publication 28.10.2010
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Year of Publication 28.10.2010
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POSITION-RELATED EMISSION CONTROL
SCHOLL, RALPH, THORSTEN, BUERKLER, MARKUS, THORN, FRANK, VINCENT, MICHAEL, GRANGE, MAIER, ANDREAS
Year of Publication 28.10.2010
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Year of Publication 28.10.2010
Patent