Discovery and Structure-Based Design of Potent Covalent PPARγ Inverse-Agonists BAY-4931 and BAY-0069
Orsi, Douglas L., Pook, Elisabeth, Bräuer, Nico, Friberg, Anders, Lienau, Philip, Lemke, Christopher T., Stellfeld, Timo, Brüggemeier, Ulf, Pütter, Vera, Meyer, Hanna, Baco, Maria, Tang, Stephanie, Cherniack, Andrew D., Westlake, Lindsay, Bender, Samantha A., Kocak, Mustafa, Strathdee, Craig A., Meyerson, Matthew, Eis, Knut, Goldstein, Jonathan T.
Published in Journal of medicinal chemistry (10.11.2022)
Published in Journal of medicinal chemistry (10.11.2022)
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Biphenyls as potent vitronectin receptor antagonists. Part 3: Squaric acid amides
Urbahns, Klaus, Härter, Michael, Albers, Markus, Schmidt, Delf, Stelte-Ludwig, Beatrix, Brüggemeier, Ulf, Vaupel, Andrea, Keldenich, Jörg, Lustig, Klemens, Tsujishita, Hideki, Gerdes, Christoph
Published in Bioorganic & medicinal chemistry letters (15.11.2007)
Published in Bioorganic & medicinal chemistry letters (15.11.2007)
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Correction to “Discovery and Structure-Based Design of Potent Covalent PPARγ Inverse-Agonists BAY-4931 and BAY-0069”
Orsi, Douglas L., Pook, Elisabeth, Bräuer, Nico, Friberg, Anders, Lienau, Philip, Lemke, Christopher T., Stellfeld, Timo, Brüggemeier, Ulf, Pütter, Vera, Meyer, Hanna, Baco, Maria, Tang, Stephanie, Cherniack, Andrew D., Westlake, Lindsay, Bender, Samantha A., Kocak, Mustafa, Strathdee, Craig A., Meyerson, Matthew, Eis, Knut, Goldstein, Jonathan T.
Published in Journal of medicinal chemistry (12.01.2023)
Published in Journal of medicinal chemistry (12.01.2023)
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SUBSTITUTED 2-ACETAMIDO-5-ARY1-1,2,4-TRIAZOLONES AND USE THEREOF
DELBECK, MARTINA, TRUBEL, HUBERT, GEIB, VOLKER, FURSTNER, CHANTAL, KRETSCHMER, AXEL, BRUGGEMEIER, ULF, KELDENICH, JORG, KERN, ARMIN, POOK, ELISABETH, SCHMECK, CARSTEN, KOLKHOF, PETER
Year of Publication 31.03.2016
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Year of Publication 31.03.2016
Patent
Substituted 2-acetamido-5-aryl-1,2,4-triazolones and use thereof
GEISS, VOLKER, DELBECK, MARTINA, TRUBEL, HUBERT, FURSTNER, CHANTAL, KRETSCHMER, AXEL, BRUGGEMEIER, ULF, KELDENICH, JORG, KERN, ARMIN, POOK, ELISABETH, SCHMECK, CARSTEN, KOLKHOF, PETER
Year of Publication 06.08.2015
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Year of Publication 06.08.2015
Patent