Overcoming Wnt-β-catenin dependent anticancer therapy resistance in leukaemia stem cells
Perry, John M, Tao, Fang, Roy, Anuradha, Lin, Tara, He, Xi C, Chen, Shiyuan, Lu, Xiuling, Nemechek, Jacqelyn, Ruan, Linhao, Yu, Xiazhen, Dukes, Debra, Moran, Andrea, Pace, Jennifer, Schroeder, Kealan, Zhao, Meng, Venkatraman, Aparna, Qian, Pengxu, Li, Zhenrui, Hembree, Mark, Paulson, Ariel, He, Zhiquan, Xu, Dong, Tran, Thanh-Huyen, Deshmukh, Prashant, Nguyen, Chi Thanh, Kasi, Rajeswari M, Ryan, Robin, Broward, Melinda, Ding, Sheng, Guest, Erin, August, Keith, Gamis, Alan S, Godwin, Andrew, Sittampalam, G Sitta, Weir, Scott J, Li, Linheng
Published in Nature cell biology (01.06.2020)
Published in Nature cell biology (01.06.2020)
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Drug repurposing for gastrointestinal stromal tumor
Pessetto, Ziyan Y, Weir, Scott J, Sethi, Geetika, Broward, Melinda A, Godwin, Andrew K
Published in Molecular cancer therapeutics (01.07.2013)
Published in Molecular cancer therapeutics (01.07.2013)
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Comparative oncology approach to drug repurposing in osteosarcoma
Parrales, Alejandro, McDonald, Peter, Ottomeyer, Megan, Roy, Anuradha, Shoenen, Frank J, Broward, Melinda, Bruns, Tyce, Thamm, Douglas H, Weir, Scott J, Neville, Kathleen A, Iwakuma, Tomoo, Fulbright, Joy M
Published in PloS one (26.03.2018)
Published in PloS one (26.03.2018)
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Targeting Epithelial-Mesenchymal Transition for Identification of Inhibitors for Pancreatic Cancer Cell Invasion and Tumor Spheres Formation
Polireddy, Kishore, Dong, Ruochen, McDonald, Peter R, Wang, Tao, Luke, Brendan, Chen, Ping, Broward, Melinda, Roy, Anuradha, Chen, Qi
Published in PloS one (20.10.2016)
Published in PloS one (20.10.2016)
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Design, Synthesis, and Evaluation of Duocarmycin O-Amino Phenol Prodrugs Subject to Tunable Reductive Activation
Lajiness, James P, Robertson, William M, Dunwiddie, Irene, Broward, Melinda A, Vielhauer, George A, Weir, Scott J, Boger, Dale L
Published in Journal of medicinal chemistry (11.11.2010)
Published in Journal of medicinal chemistry (11.11.2010)
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A Unique Class of Duocarmycin and CC-1065 Analogues Subject to Reductive Activation
Jin, Wei, Trzupek, John D, Rayl, Thomas J, Broward, Melinda A, Vielhauer, George A, Weir, Scott J, Hwang, Inkyu, Boger, Dale L
Published in Journal of the American Chemical Society (12.12.2007)
Published in Journal of the American Chemical Society (12.12.2007)
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DRES-07. SIGNIFICANT SEX DIFFERENCES IN TEMOZOLOMIDE EFFICACY IN GLIOBLASTOMA (GBM) ARE DETECTABLE IN CELL AND PATIENT BASED EVALUATIONS
Taylor, Sara, Rayfield, Corbin, Kim, Albert, Broward, Melinda, Roy, Anu, Weir, Scott, Swanson, Kristin, Rubin, Joshua
Published in Neuro-oncology (Charlottesville, Va.) (01.11.2016)
Published in Neuro-oncology (Charlottesville, Va.) (01.11.2016)
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Abstract 2903: A novel compound induces synthetic lethality for p53 mutations in osteosarcoma cells
Iwakuma, Tomoo, Parrales, Alejandro, McDonald, Peter, Roy, Anuradha, Braun, Mitchell W., Schoenen, Frank J., Wang, Jenna, Rogers, Steve, Broward, Melinda, Bruns, Tyce, Anant, Shrikant, Dixon, Dan A., Meyer, Fred, Chastain, Katherine M., Thamm, Douglas H., Weir, Scott J., Neville, Kathleen, Fulbright, Joy M.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract 5334: Targeting the KIF15-TPX2 PPI to overcome KIF11 inhibitor resistance in epithelial ovarian cancer
Gibbs, Benjamin K., Douglas, Justin T., Wates, Rebecca J., McDonald, Peter R., Whitaker, Amy M., Ndi, Cornelius N., Pathak, Harsh B., Harned, Laurie A., Neuenswander, Sarah A., Broward, Melinda A., Freudenthal, Bret D., Roy, Anuradha, Schoenen, Frank J., Godwin, Andrew K.
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Abstract 3689: Comparative oncology drug discovery for Osteosarcoma in dogs and humans
Fulbright, Joy M., Neville, Kathleen, Broward, Melinda, Bruns, Tyce A., Roy, Anuradha, McDonald, Peter, Ottomeyer, Megan, Thamm, Douglas H., Iwakuma, Tomoo
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Gender-specific reduction of hepatic Mrp2 expression by high-fat diet protects female mice from ANIT toxicity
Kong, Bo, Csanaky, Iván L., Aleksunes, Lauren M., Patni, Meghan, Chen, Qi, Ma, Xiaochao, Jaeschke, Hartmut, Weir, Scott, Broward, Melinda, Klaassen, Curtis D., Guo, Grace L.
Published in Toxicology and applied pharmacology (01.06.2012)
Published in Toxicology and applied pharmacology (01.06.2012)
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KU-AS-272, a Potential Single-Dose Sterilant for Cats and Dogs, Shows Safety and Ability to Block Spermatogenesis in Testis to Sertoli Cells Only after a Single Subcutaneous Injection in Male Rat
Gupta, Vijayalaxmi G., Roby, Katherine F., Kern, Brian, Hall, Todd, Jakkaraj, Sudhakar, Chakrasali, Ramappa, Georg, Gunda I., Broward, Melinda, Wood, Robyn, Weir, Scott, Tash, Joseph S.
Published in Biology of reproduction (01.08.2012)
Published in Biology of reproduction (01.08.2012)
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Combination Intraperitoneal Chemotherapy Is Superior to Mitomycin C or Oxaliplatin for Colorectal Carcinomatosis In Vivo
Cohen, Mark S., Al-kasspooles, Mazin F., Williamson, Stephen K., Henry, David, Broward, Melinda, Roby, Katherine F.
Published in Annals of surgical oncology (2010)
Published in Annals of surgical oncology (2010)
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Anti-Spermatogenic Efficacy of Nonhormonal Male Contraceptive Agent, H2-Gamendazole, in Mice, Rats, Rabbits, and Nonhuman Primates (Rhesus), and a Multiple Low Dose Oral Regimen That Gives 100% Infertility with Complete Reversibility
Gupta, Vijayalaxmi G., Zelinski, Mary, Steinmetz, Karen, Miklos, Andras, Broward, Melinda, Jakkaraj, Sudhakar, Chakrasali, Ramappa, Georg, Gunda I., Tash, Joseph S.
Published in Biology of reproduction (01.07.2011)
Published in Biology of reproduction (01.07.2011)
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Journal Article
A Unique Class of Duocarmycin and CC-1065 Analogues Subject to Reductive Activation
Jin, Wei, Trzupek, John D, Rayl, Thomas J, Broward, Melinda A, Vielhauer, George A, Weir, Scott J, Hwang, Inkyu, Boger, Dale L
Published in Journal of the American Chemical Society (01.01.2007)
Published in Journal of the American Chemical Society (01.01.2007)
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