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Published in Neuropsychopharmacology (New York, N.Y.) (01.06.2014)
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Synthesis and Structure–Activity Relationships of Allosteric Potentiators of the M4 Muscarinic Acetylcholine Receptor
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Published in ChemMedChem (05.10.2009)
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Wood, Michael R, Hopkins, Corey R, Brogan, John T, Conn, P. Jeffrey, Lindsley, Craig W
Published in Biochemistry (Easton) (05.04.2011)
Published in Biochemistry (Easton) (05.04.2011)
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Chemical Modulation of Mutant mGlu1 Receptors Derived from Deleterious GRM1 Mutations Found in Schizophrenics
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Published in ACS chemical biology (17.10.2014)
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The Discovery and Characterization of ML218: A Novel, Centrally Active T-Type Calcium Channel Inhibitor with Robust Effects in STN Neurons and in a Rodent Model of Parkinson’s Disease
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Published in ACS chemical neuroscience (21.12.2011)
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Optimization of a small molecule probe that restores e-cadherin expression
Brogan, John T., Stoops, Sydney L., Brady, Suzanne, An, Hanbing, Weaver, Connie, Daniels, J. Scott, Beauchamp, R. Daniel, Lindsley, Craig W., Waterson, Alex G.
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Total Synthesis and Biological Evaluation of the Marine Bromopyrrole Alkaloid Dispyrin: Elucidation of Discrete Molecular Targets with Therapeutic Potential
Kennedy, J. Phillip, Brogan, John T, Lindsley, Craig W
Published in Journal of natural products (Washington, D.C.) (01.10.2008)
Published in Journal of natural products (Washington, D.C.) (01.10.2008)
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Synthesis and SAR of analogues of the M1 allosteric agonist TBPB. Part I: Exploration of alternative benzyl and privileged structure moieties
Bridges, Thomas M., Brady, Ashley E., Phillip Kennedy, J., Nathan Daniels, R., Miller, Nicole R., Kim, Kwango, Breininger, Micah L., Gentry, Patrick R., Brogan, John T., Jones, Carrie K., Jeffrey Conn, P., Lindsley, Craig W.
Published in Bioorganic & medicinal chemistry (15.10.2008)
Published in Bioorganic & medicinal chemistry (15.10.2008)
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Synthesis and Structure–Activity Relationships of Allosteric Potentiators of the M 4 Muscarinic Acetylcholine Receptor
Kennedy, J. Phillip, Bridges, Thomas M., Gentry, Patrick R., Brogan, John T., Kane, Alexander S., Jones, Carrie K., Brady, Ashley E., Shirey, Jana K., Conn, P. Jeffrey, Lindsley, Craig W.
Published in ChemMedChem (05.10.2009)
Published in ChemMedChem (05.10.2009)
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Total Synthesis of (+)-7-Bromotrypargine and Unnatural Analogues: Biological Evaluation Uncovers Activity at CNS Targets of Therapeutic Relevance
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Published in ACS chemical neuroscience (16.11.2011)
Published in ACS chemical neuroscience (16.11.2011)
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Antipsychotic Drug-Like Effects of the Selective M sub(4) Muscarinic Acetylcholine Receptor Positive Allosteric Modulator VU0152100
Byun, Nellie E, Grannan, Michael, Bubser, Michael, Barry, Robert L, Thompson, Analisa, Rosanelli, John, Gowrishankar, Raajaram, Kelm, Nathaniel D, Damon, Stephen, Bridges, Thomas M, Melancon, Bruce J, Tarr, James C, Brogan, John T, Avison, Malcolm J, Deutch, Ariel Y, Wess, Juergen, Wood, Michael R, Lindsley, Craig W, Gore, John C, Conn, P Jeffrey, Jones, Carrie K
Published in Neuropsychopharmacology (New York, N.Y.) (01.06.2014)
Published in Neuropsychopharmacology (New York, N.Y.) (01.06.2014)
Get full text
Journal Article
Chemical Modulation of Mutant mGlu 1 Receptors Derived from Deleterious GRM1 Mutations Found in Schizophrenics
Cho, Hyekyung P., Garcia-Barrantes, Pedro M., Brogan, John T., Hopkins, Corey R., Niswender, Colleen M., Rodriguez, Alice L., Venable, Daryl F., Morrison, Ryan D., Bubser, Michael, Daniels, J. Scott, Jones, Carrie K., Conn, P. Jeffrey, Lindsley, Craig W.
Published in ACS chemical biology (17.10.2014)
Published in ACS chemical biology (17.10.2014)
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Synthesis and SAR of analogues of the Ml allosteric agonist TBPB. Part I: Exploration of alternative benzyl and privileged structure moieties
BRIDGES, Thomas M, BRADY, Ashley E, CONNA, P. Jeffrey, LINDSLEY, Craig W, KENNEDY, J. Phillip, DANIELS, R. Nathan, MILLER, Nicole R, KIM, Kwango, BREININGER, Micah L, GENTRY, Patrick R, BROGAN, John T, JONES, Carrie K
Published in Bioorganic & medicinal chemistry letters (2008)
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Published in Bioorganic & medicinal chemistry letters (2008)
Journal Article
Synthesis and structure-activity relationships of allosteric potentiators of the m(4) muscarinic acetylcholine receptor
Kennedy, J Phillip, Bridges, Thomas M, Gentry, Patrick R, Brogan, John T, Kane, Alexander S, Jones, Carrie K, Brady, Ashley E, Shirey, Jana K, Conn, P Jeffrey, Lindsley, Craig W
Published in ChemMedChem (01.10.2009)
Published in ChemMedChem (01.10.2009)
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UNNATURAL DISPYRIN ANALOGUES, PREPARATION AND USES THEREOF
LINDSLEY, CRAIG, W, BROGAN, JOHN, T, KENNEDY, PHILLIP, J, CONN, JEFFREY, P
Year of Publication 17.12.2009
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Year of Publication 17.12.2009
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