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SABNIS, Gauri J, GOLOUBEVA, Olga, CHUMSRI, Saranya, NGUYEN, Nguyen, SUKUMAR, Saraswati, BRODIE, Angela M. H
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Published in Cancer research (Chicago, Ill.) (01.03.2011)
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Inhibition of estrogen signaling activates the NRF2 pathway in breast cancer
Yao, Yuan, Brodie, Angela M. H, Davidson, Nancy E, Kensler, Thomas W, Zhou, Qun
Published in Breast cancer research and treatment (01.11.2010)
Published in Breast cancer research and treatment (01.11.2010)
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Novel C-17-Heteroaryl Steroidal CYP17 Inhibitors/Antiandrogens: Synthesis, in Vitro Biological Activity, Pharmacokinetics, and Antitumor Activity in the LAPC4 Human Prostate Cancer Xenograft Model
Handratta, Venkatesh D, Vasaitis, Tadas S, Njar, Vincent C. O, Gediya, Lalji K, Kataria, Ritesh, Chopra, Pankaj, Newman, Donnell, Farquhar, Rena, Guo, Zhiyong, Qiu, Yun, Brodie, Angela M. H
Published in Journal of medicinal chemistry (21.04.2005)
Published in Journal of medicinal chemistry (21.04.2005)
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A Novel Androgen Receptor Splice Variant Is Up-regulated during Prostate Cancer Progression and Promotes Androgen Depletion-Resistant Growth
ZHIYONG GUO, XI YANG, KUNG, Hsing-Jien, BRODIE, Angela M. H, EDWARDS, Joanne, YUN QIU, FENG SUN, JIANG, Richeng, LINN, Douglas E, HEGE CHEN, HEGANG CHEN, XIANGTIAN KONG, MELAMED, Jonathan, TEPPER, Clifford G
Published in Cancer research (Chicago, Ill.) (15.03.2009)
Published in Cancer research (Chicago, Ill.) (15.03.2009)
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Aromatase inhibitors and xenograft studies
Chumsri, Saranya, Sabnis, Gauri J., Howes, Timothy, Brodie, Angela M.H.
Published in Steroids (01.07.2011)
Published in Steroids (01.07.2011)
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Conference Proceeding
Synthesis and biological evaluations of putative metabolically stable analogs of VN/124-1 (TOK-001): Head to head anti-tumor efficacy evaluation of VN/124-1 (TOK-001) and abiraterone in LAPC-4 human prostate cancer xenograft model
Bruno, Robert D., Vasaitis, Tadas S., Gediya, Lalji K., Purushottamachar, Puranik, Godbole, Abhijit M., Ates-Alagoz, Zeynep, Brodie, Angela M.H., Njar, Vincent C.O.
Published in Steroids (01.11.2011)
Published in Steroids (01.11.2011)
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Aromatase Inhibitors: Are There Differences Between Steroidal and Nonsteroidal Aromatase Inhibitors and Do They Matter?
Miller, William R., Bartlett, John, Brodie, Angela M. H., Brueggemeier, Robert W., di Salle, Enrico, Lønning, Per Eystein, Llombart, Antonio, Maass, Nicolai, Maudelonde, Thierry, Sasano, Hironobu, Goss, Paul E.
Published in The oncologist (Dayton, Ohio) (01.08.2008)
Published in The oncologist (Dayton, Ohio) (01.08.2008)
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Stopping treatment can reverse acquired resistance to letrozole
Sabnis, Gauri J, Macedo, Luciana F, Goloubeva, Olga, Schayowitz, Adam, Brodie, Angela M H
Published in Cancer research (Chicago, Ill.) (15.06.2008)
Published in Cancer research (Chicago, Ill.) (15.06.2008)
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Activation of mitogen-activated protein kinase in xenografts and cells during prolonged treatment with aromatase inhibitor letrozole
JELOVAC, Danijela, SABNIS, Gauri, LONG, Brian J, MACEDO, Luciana, GOLOUBEVA, Olga G, BRODIE, Angela M. H
Published in Cancer research (Chicago, Ill.) (15.06.2005)
Published in Cancer research (Chicago, Ill.) (15.06.2005)
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Synergistic effect of a novel antiandrogen, VN/124-1, and signal transduction inhibitors in prostate cancer progression to hormone independence in vitro
Schayowitz, Adam, Sabnis, Gauri, Njar, Vincent C O, Brodie, Angela M H
Published in Molecular cancer therapeutics (01.01.2008)
Published in Molecular cancer therapeutics (01.01.2008)
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Three Dimensional Pharmacophore Modeling of Human CYP17 Inhibitors. Potential Agents for Prostate Cancer Therapy
Clement, Omoshile O, Freeman, Clive M, Hartmann, Rolf W, Handratta, Venkatesh D, Vasaitis, Tadas S, Brodie, Angela M. H, Njar, Vincent C. O
Published in Journal of medicinal chemistry (05.06.2003)
Published in Journal of medicinal chemistry (05.06.2003)
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Novel Retinoic Acid Metabolism Blocking Agents Endowed with Multiple Biological Activities Are Efficient Growth Inhibitors of Human Breast and Prostate Cancer Cells in Vitro and a Human Breast Tumor Xenograft in Nude Mice
Patel, Jyoti B, Huynh, Carlic K, Handratta, Venkatesh D, Gediya, Lalji K, Brodie, Angela M. H, Goloubeva, Olga G, Clement, Omoshile O, Nanne, Ivo P, Soprano, Dianne Robert, Njar, Vincent C. O
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
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Novel Membrane-associated Androgen Receptor Splice Variant Potentiates Proliferative and Survival Responses in Prostate Cancer Cells
Yang, Xi, Guo, Zhiyong, Sun, Feng, Li, Wei, Alfano, Alan, Shimelis, Hermela, Chen, Mingyuan, Brodie, Angela M.H., Chen, Hegang, Xiao, Zhen, Veenstra, Timothy D., Qiu, Yun
Published in The Journal of biological chemistry (14.10.2011)
Published in The Journal of biological chemistry (14.10.2011)
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Regulation of androgen receptor activity by tyrosine phosphorylation
Guo, Zhiyong, Dai, Bojie, Jiang, Tianyun, Xu, Kexin, Xie, Yingqiu, Kim, Oekyung, Nesheiwat, Issa, Kong, Xiangtian, Melamed, Jonathan, Handratta, Venkatesh D., Njar, Vincent C.O., Brodie, Angela M.H., Yu, Li-Rong, Veenstra, Timothy D., Chen, Hegang, Qiu, Yun
Published in Cancer cell (01.10.2006)
Published in Cancer cell (01.10.2006)
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Additive antitumor effect of aromatase inhibitor letrozole and antiestrogen fulvestrant in a postmenopausal breast cancer model
JELOVAC, Danijela, MACEDO, Luciana, GOLOUBEVA, Olga G, HANDRATTA, Venkatesh, BRODIE, Angela M. H
Published in Cancer research (Chicago, Ill.) (15.06.2005)
Published in Cancer research (Chicago, Ill.) (15.06.2005)
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