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Zhou, Hao, Topiol, Sidney W., Grenon, Michel, Jimenez, Hermogenes N., Uberti, Michelle A., Smith, Daniel G., Brodbeck, Robbin M., Chandrasena, Gamini, Pedersen, Henrik, Madsen, Jens Christian, Doller, Darío, Li, Guiying
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
Published in Bioorganic & medicinal chemistry letters (01.03.2013)
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Identification and Characterization of NDT 9513727 [N,N-bis(1,3-Benzodioxol-5-ylmethyl)-1-butyl-2,4-diphenyl-1H-imidazole-5-methanamine], a Novel, Orally Bioavailable C5a Receptor Inverse Agonist
Brodbeck, Robbin M, Cortright, Daniel N, Kieltyka, Andrzej P, Yu, Jianying, Baltazar, Carolyn O, Buck, Marianne E, Meade, Robin, Maynard, George D, Thurkauf, Andrew, Chien, Du-Shieng, Hutchison, Alan J, Krause, James E
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Published in The Journal of pharmacology and experimental therapeutics (01.12.2008)
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P2X7 receptor-mediated release of microglial prostanoids and miRNAs correlates with reversal of neuropathic hypersensitivity in rats
Staal, Roland, Khayrullina, Tanzilya, Christensen, Rie, Hestehave, Sara, Zhou, Hua, Cajina, Manuel, Nattini, Megan E, Gandhi, Adarsh, Fallon, Shaun M, Schmidt, Megan, Zorn, Stevin H, Brodbeck, Robbin M, Chandrasena, Gamini, Segerdahl, Märta, Breysse, Nathalie, Hopper, Allen T, Möller, Thomas, Munro, Gordon
Published in European journal of pain (01.07.2022)
Published in European journal of pain (01.07.2022)
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Leukocyte Effects of C5a-Receptor Blockade During Simulated Extracorporeal Circulation
Rinder, Christine S., MD, Smith, Michael J., PhD, Rinder, Henry M., MD, Cortright, Daniel N., PhD, Brodbeck, Robbin M., PhD, Krause, James E., PhD, Smith, Brian R., MD
Published in The Annals of thoracic surgery (2007)
Published in The Annals of thoracic surgery (2007)
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Molecular Characterization of the Gerbil C5a Receptor and Identification of a Transmembrane Domain V Amino Acid That Is Crucial for Small Molecule Antagonist Interaction
Waters, Stephen M., Brodbeck, Robbin M., Steflik, Jeremy, Yu, Jianying, Baltazar, Carolyn, Peck, Amy E., Severance, Daniel, Zhang, Lu Yan, Currie, Kevin, Chenard, Bertrand L., Hutchison, Alan J., Maynard, George, Krause, James E.
Published in The Journal of biological chemistry (09.12.2005)
Published in The Journal of biological chemistry (09.12.2005)
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Efficacy switching SAR of mGluR5 allosteric modulators: Highly potent positive and negative modulators from one chemotype
Sams, Anette Graven, Mikkelsen, Gitte Kobberøe, Brodbeck, Robbin M., Pu, Xiaosui, Ritzén, Andreas
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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C5L2, a Nonsignaling C5A Binding Protein
Okinaga, Shoji, Slattery, Dubhfeasa, Humbles, Alison, Zsengeller, Zsusanna, Morteau, Olivier, Kinrade, Michele Bennett, Brodbeck, Robbin M, Krause, James E, Choe, Hye-Ryun, Gerard, Norma P, Gerard, Craig
Published in Biochemistry (Easton) (12.08.2003)
Published in Biochemistry (Easton) (12.08.2003)
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N-Aryl pyrrolidinonyl oxadiazoles as potent mGluR5 positive allosteric modulators
Packiarajan, Mathivanan, Mazza Ferreira, Christine G., Hong, Sang-Phyo, White, Andrew D., Chandrasena, Gamini, Pu, Xiaosui, Brodbeck, Robbin M., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Fused thiazolyl alkynes as potent mGlu5 receptor positive allosteric modulators
Packiarajan, Mathivanan, Grenon, Michel, Zorn, Samuel, Hopper, Allen T., White, Andrew D., Chandrasena, Gamini, Pu, Xiaosui, Brodbeck, Robbin M., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
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Azetidinyl oxadiazoles as potent mGluR5 positive allosteric modulators
Packiarajan, Mathivanan, Ferreira, Christine G. Mazza, Hong, Sang-Phyo, White, Andrew D., Chandrasena, Gamini, Pu, Xiaosui, Brodbeck, Robbin M., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (15.10.2012)
Published in Bioorganic & medicinal chemistry letters (15.10.2012)
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Novel heterocyclic compounds as mGlu5 antagonists: WO2009015897
Doller, Dario, Li, Guiying, Brodbeck, Robbin M, Thomsen, Christian
Published in Expert opinion on therapeutic patents (01.03.2010)
Published in Expert opinion on therapeutic patents (01.03.2010)
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Aminopyrazine CB1 receptor inverse agonists
Wustrow, David J., Maynard, George D., Yuan, Jun, Zhao, He, Mao, Jianmin, Guo, Qin, Kershaw, Mark, Hammer, Jack, Brodbeck, Robbin M., Near, Kristen E., Zhou, Dan, Beers, David S., Chenard, Bertrand L., Krause, James E., Hutchison, Alan J.
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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Fused thiazolyl alkynes as potent mGlu(5) receptor positive allosteric modulators
Packiarajan, Mathivanan, Grenon, Michel, Zorn, Samuel, Hopper, Allen T., White, Andrew D., Chandrasena, Gamini, Pu, Xiaosui, Brodbeck, Robbin M., Robichaud, Albert J.
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
Published in Bioorganic & medicinal chemistry letters (15.07.2013)
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Leukocyte effects of C5a-receptor blockade during simulated extracorporeal circulation. Commentary
RINDER, Christine S, SMITH, Michael J, RINDER, Henry M, CORTRIGHT, Daniel N, BRODBECK, Robbin M, KRAUSE, James E, SMITH, Brian R, LAPPEGARD, Knut Tore
Published in The Annals of thoracic surgery (2007)
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Published in The Annals of thoracic surgery (2007)
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Molecular characterization of the gerbil C5a receptor and identification of a transmembrane domain V amino acid that is crucial for small molecule antagonist interaction. VOLUME 280 (2005) PAGES 40617-40623
Waters, Stephen M., Brodbeck, Robbin M., Steflik, Jeremy, Yu, Jianying, Baltazar, Carolyn, Peck, Amy E., Severance, Daniel, Zhang, Lu Yan, Currie, Kevin, Chenard, Bertrand L., Hutchison, Alan J., Maynard, George, Krause, James E.
Published in The Journal of biological chemistry (10.02.2006)
Published in The Journal of biological chemistry (10.02.2006)
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Circulatory Half-Life but not Interaction with the Lutropin/Chorionic Gonadotropin Receptor is Modulated by Sulfation of Bovine Lutropin Oligosaccharides
Baenziger, Jacques U., Swatantar Kuma r, Brodbeck, Robbin M., Smith, Peter L., Beranek, Mary C.
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1992)
Published in Proceedings of the National Academy of Sciences - PNAS (01.01.1992)
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