Synthesis, structure-property relationships and pharmacokinetic evaluation of ethyl 6-aminonicotinate sulfonylureas as antagonists of the P2Y(12) receptor
Bach, Peter, Bostrom, Jonas, Brickmann, Kay, van Giezen, J. J. J., Groneberg, Robert D., Harvey, Darren M., O'Sullivan, Michael, Zetterberg, Fredrik
Published in European journal of medicinal chemistry (01.07.2013)
Published in European journal of medicinal chemistry (01.07.2013)
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Synthesis, structure–property relationships and pharmacokinetic evaluation of ethyl 6-aminonicotinate sulfonylureas as antagonists of the P2Y12 receptor
Bach, Peter, Boström, Jonas, Brickmann, Kay, van Giezen, J.J.J., Groneberg, Robert D., Harvey, Darren M., O'Sullivan, Michael, Zetterberg, Fredrik
Published in European journal of medicinal chemistry (01.07.2013)
Published in European journal of medicinal chemistry (01.07.2013)
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A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y12 receptor
BACH, Peter, BOSTROM, Jonas, BRICKMANN, Kay, VAN GIEZEN, J. J. J, HOVLAND, Ragnar, PETERSSON, Annika U, RAY, Asim, ZETTERBERG, Fredrik
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Design of small molecule inhibitors of acetyl-CoA carboxylase 1 and 2 showing reduction of hepatic malonyl-CoA levels in vivo in obese Zucker rats
Bengtsson, Christoffer, Blaho, Stefan, Saitton, David Blomberg, Brickmann, Kay, Broddefalk, Johan, Davidsson, Öjvind, Drmota, Tomas, Folmer, Rutger, Hallberg, Kenth, Hallén, Stefan, Hovland, Ragnar, Isin, Emre, Johannesson, Petra, Kull, Bengt, Larsson, Lars-Olof, Löfgren, Lars, Nilsson, Kristina E., Noeske, Tobias, Oakes, Nick, Plowright, Alleyn T., Schnecke, Volker, Ståhlberg, Pernilla, Sörme, Pernilla, Wan, Hong, Wellner, Eric, Öster, Linda
Published in Bioorganic & medicinal chemistry (15.05.2011)
Published in Bioorganic & medicinal chemistry (15.05.2011)
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Journal Article
A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y sub(12 receptor)
Bach, Peter, Bostroem, Jonas, Brickmann, Kay, Van Giezen, JJJ, Hovland, Ragnar, Petersson, Annika U, Ray, Asim, Zetterberg, Fredrik
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Journal Article
A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y 12 receptor
Bach, Peter, Boström, Jonas, Brickmann, Kay, van Giezen, J.J.J., Hovland, Ragnar, Petersson, Annika U., Ray, Asim, Zetterberg, Fredrik
Published in Bioorganic & medicinal chemistry letters (2011)
Published in Bioorganic & medicinal chemistry letters (2011)
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5-alkyl-1,3-oxazole derivatives of 6-amino-nicotinic acids as alkyl ester bioisosteres are antagonists of the P2Y12 receptor
Bach, Peter, Boström, Jonas, Brickmann, Kay, Burgess, Laurence E, Clarke, David, Groneberg, Robert D, Harvey, Darren M, Laird, Ellen R, O'Sullivan, Michael, Zetterberg, Fredrik
Published in Future medicinal chemistry (01.11.2013)
Published in Future medicinal chemistry (01.11.2013)
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Journal Article
Synthesis and biological evaluation of leucine enkephalin turn mimetics
Blomberg, D, Kreye, P, Fowler, C, Brickmann, K, Kihlberg, J
Published in Organic & biomolecular chemistry (07.02.2006)
Published in Organic & biomolecular chemistry (07.02.2006)
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Synthesis and Conformational Studies of a β-Turn Mimetic Incorporated in Leu-enkephalin
Blomberg, David, Hedenström, Mattias, Kreye, Paul, Sethson, Ingmar, Brickmann, Kay, Kihlberg, Jan
Published in Journal of organic chemistry (14.05.2004)
Published in Journal of organic chemistry (14.05.2004)
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Journal Article
Synthesis and Pharmacological Evaluation of an Analogue of the Peptide Hormone Oxytocin That Contains a Mimetic of an Inverse γ-Turn
Yuan, ZhongQing, Blomberg, David, Sethson, Ingmar, Brickmann, Kay, Ekholm, Kjell, Johansson, Birgitta, Nilsson, Anders, Kihlberg, Jan
Published in Journal of medicinal chemistry (06.06.2002)
Published in Journal of medicinal chemistry (06.06.2002)
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Synthesis of Conformationally Restricted Mimetics of γ-Turns and Incorporation into Desmopressin, an Analogue of the Peptide Hormone Vasopressin
Brickmann, Kay, Yuan, ZhongQing, Sethson, Ingmar, Somfai, Peter, Kihlberg, Jan
Published in Chemistry : a European journal (02.08.1999)
Published in Chemistry : a European journal (02.08.1999)
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Conformations and Receptor Activity of Desmopressin Analogues, Which Contain γ-Turn Mimetics or a Ψ[CH2O] Isostere
Hedenström, Mattias, Yuan, Brickmann, Kay, Carlsson, Jolanta, Ekholm, Kjell, Johansson, Birgitta, Kreutz, Eva, Nilsson, Anders, Sethson, Ingmar, Kihlberg, Jan
Published in Journal of medicinal chemistry (06.06.2002)
Published in Journal of medicinal chemistry (06.06.2002)
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