IRC‐083864, a novel bis quinone inhibitor of CDC25 phosphatases active against human cancer cells
Brezak, Marie‐Christine, Valette, Annie, Quaranta, Muriel, Contour‐Galcera, Marie‐Odile, Jullien, Denis, Lavergne, Olivier, Frongia, Céline, Bigg, Dennis, Kasprzyk, Philip G., Prevost, Grégoire Pierre, Ducommun, Bernard
Published in International journal of cancer (15.03.2009)
Published in International journal of cancer (15.03.2009)
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Inhibition of human tumor cell growth in vivo by an orally bioavailable inhibitor of CDC25 phosphatases
Brezak, Marie-Christine, Quaranta, Muriel, Contour-Galcera, Marie-Odile, Lavergne, Olivier, Mondesert, Odile, Auvray, Pierrïck, Kasprzyk, Philip G, Prevost, Gregoire P, Ducommun, Bernard
Published in Molecular cancer therapeutics (01.09.2005)
Published in Molecular cancer therapeutics (01.09.2005)
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Journal Article
Pharmacologic inhibition of CDC25 phosphatases impairs interphase microtubule dynamics and mitotic spindle assembly
Cazales, Martine, Boutros, Rose, Brezak, Marie-Christine, Chaumeron, Sophie, Prevost, Grégoire, Ducommun, Bernard
Published in Molecular cancer therapeutics (01.01.2007)
Published in Molecular cancer therapeutics (01.01.2007)
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Journal Article
Synthesis and biological evaluation of novel heterocyclic quinones as inhibitors of the dual specificity protein phosphatase CDC25C
Lavergne, Olivier, Fernandes, Anne-Cécile, Bréhu, Laetitia, Sidhu, Alban, Brézak, Marie-Christine, Prévost, Grégoire, Ducommun, Bernard, Contour-Galcera, Marie-Odile
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Inhibition of human tumor cell growth in vivo by an orally bioavailable inhibitor of human farnesyltransferase, BIM‐46228
Prevost, Grégoire P., Pradines, Anne, Brezak, Marie‐Christine, Lonchampt, Marie‐Odile, Viossat, Isabelle, Ader, Isabelle, Toulas, Christine, Kasprzyk, Philip, Gordon, Thomas, Favre, Gilles, Morgan, Barry
Published in International journal of cancer (01.03.2001)
Published in International journal of cancer (01.03.2001)
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A novel synthetic inhibitor of CDC25 phosphatases: BN82002
BREZAK, Marie-Christine, QUARANTA, Muriel, LANCO, Christophe, KASPRZYK, Philip G, PREVOST, Gregoire P, DUCOMMUN, Bernard, MONDESERT, Odile, GALCERA, Marie-Odile, LAVERGNE, Olivier, ALBY, Frédéric, CAZALES, Martine, BALDIN, Véronique, THURIEAU, Christophe, HARNETT, Jeremiath
Published in Cancer research (Chicago, Ill.) (01.05.2004)
Published in Cancer research (Chicago, Ill.) (01.05.2004)
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Apoptosis and TRAF-1 cleavage in Epstein-Barr virus-positive nasopharyngeal carcinoma cells treated with doxorubicin combined with a farnesyl-transferase inhibitor
Vicat, Jean-Michel, Ardila-Osorio, Hector, Khabir, Abdelmajid, Brezak, Marie-Christine, Viossat, Isabelle, Kasprzyk, Philip, Jlidi, Rachid, Opolon, Paule, Ooka, Tadamassa, Prevost, Grégoire, Huang, Dolly P., Busson, Pierre
Published in Biochemical pharmacology (01.02.2003)
Published in Biochemical pharmacology (01.02.2003)
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A Novel Synthetic Inhibitor of CDC25 Phosphatases
Brezak, Marie-Christine, Quaranta, Muriel, Mondésert, Odile, Galcera, Marie-Odile, Lavergne, Olivier, Alby, Frédéric, Cazales, Martine, Baldin, Véronique, Thurieau, Christophe, Harnett, Jeremiath, Lanco, Christophe, Kasprzyk, Philip G., Prevost, Gregoire P., Ducommun, Bernard
Published in Cancer research (Chicago, Ill.) (01.05.2004)
Published in Cancer research (Chicago, Ill.) (01.05.2004)
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Inhibition of human tumor cell growth In vitro and In vivo by a specific inhibitor of human farnesyltransferase: BIM‐46068
Prevost, Grégoire P., Pradines, Anne, Viossat, Isabelle, Brezak, Marie‐Christine, Miquel, Karine, Lonchampt, Marie‐Odile, Kasprzyk, Philip, Favre, Gilles, Pignol, Bernadette, Le Breton, Christine, Dong, Jesse, Morgan, Barry
Published in International journal of cancer (08.10.1999)
Published in International journal of cancer (08.10.1999)
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Inhibitors of the CDC25 phosphatases
Prevost, Grégoire Pierre, Brezak, Marie-Christine, Goubin, Françoise, Mondesert, Odile, Galcera, Marie-Odile, Quaranta, Muriel, Alby, Frédéric, Lavergne, Olivier, Ducommun, Bernard
Published in Progress in cell cycle research (2003)
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Published in Progress in cell cycle research (2003)
Journal Article
Synthesis and Biological Evaluation of Novel Heterocyclic Quinones as Inhibitors of the Dual Specificity Protein Phosphatase CDC25C
Lavergne, Olivier, Fernandes, Anne-Cecile, Brehu, Laetitia, Sidhu, Alban, Brezak, Marie-Christine, Prevost, Gregoire, Ducommun, Bernard, Contour-Galcera, Marie-Odile
Published in ChemInform (04.04.2006)
Published in ChemInform (04.04.2006)
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Inhibition of human tumor cell growthin vivo by an orally bioavailable inhibitor of human farnesyltransferase, BIM-46228
Prevost, Grégoire P., Pradines, Anne, Brezak, Marie-Christine, Lonchampt, Marie-Odile, Viossat, Isabelle, Ader, Isabelle, Toulas, Christine, Kasprzyk, Philip, Gordon, Thomas, Favre, Gilles, Morgan, Barry
Published in International journal of cancer (01.03.2001)
Published in International journal of cancer (01.03.2001)
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Journal Article
Inhibition of human tumor cell growthIn vitro andIn vivo by a specific inhibitor of human farnesyltransferase: BIM-46068
Prevost, Gr goire P., Pradines, Anne, Viossat, Isabelle, Brezak, Marie-Christine, Miquel, Karine, Lonchampt, Marie-Odile, Kasprzyk, Philip, Favre, Gilles, Pignol, Bernadette, Le Breton, Christine, Dong, Jesse, Morgan, Barry
Published in International journal of cancer (08.10.1999)
Published in International journal of cancer (08.10.1999)
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Journal Article
Inhibitors of Cdc25 phosphatases
MARIE-ODILE GALCERA CONTOUR, CHRISTOPHE LANCO, FRANCOISE GOUBIN-GRAMMATICA, BERNARD DUCOMMUN, GREGOIRE PREVOST, MARIE- CHRISTINE BREZAK PANNETIER, CHRISTOPHE THURIEAU
Year of Publication 09.11.2006
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Year of Publication 09.11.2006
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