Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H2R and D3R
Biselli, Sabrina, Bresinsky, Merlin, Tropmann, Katharina, Forster, Lisa, Honisch, Claudia, Buschauer, Armin, Bernhardt, Günther, Pockes, Steffen
Published in European journal of medicinal chemistry (15.03.2021)
Published in European journal of medicinal chemistry (15.03.2021)
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Journal Article
Abolishing Dopamine D-2long/D-3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H-2 Receptor Agonists
Tropmann, Katharina, Bresinsky, Merlin, Forster, Lisa, Moennich, Denise, Buschauer, Armin, Wittmann, Hans-Joachim, Huebner, Harald, Gmeiner, Peter, Pockes, Steffen, Strasser, Andrea
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
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Journal Article
Cardiac Effects of Novel Histamine H 2 Receptor Agonists
Gergs, Ulrich, Büxel, Maren L, Bresinsky, Merlin, Kirchhefer, Uwe, Fehse, Charlotte, Höring, Carina, Hofmann, Britt, Marušáková, Margaréta, Čináková, Aneta, Schwarz, Rebecca, Pockes, Steffen, Neumann, Joachim
Published in The Journal of pharmacology and experimental therapeutics (01.12.2021)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2021)
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Journal Article
Abolishing Dopamine D2long/D3 Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H2 Receptor Agonists
Tropmann, Katharina, Bresinsky, Merlin, Forster, Lisa, Mönnich, Denise, Buschauer, Armin, Wittmann, Hans-Joachim, Hübner, Harald, Gmeiner, Peter, Pockes, Steffen, Strasser, Andrea
Published in Journal of medicinal chemistry (24.06.2021)
Published in Journal of medicinal chemistry (24.06.2021)
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Journal Article
Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent
Szczepańska, Katarzyna, Pockes, Steffen, Podlewska, Sabina, Höring, Carina, Mika, Kamil, Latacz, Gniewomir, Bednarski, Marek, Siwek, Agata, Karcz, Tadeusz, Nagl, Martin, Bresinsky, Merlin, Mönnich, Denise, Seibel, Ulla, Kuder, Kamil J., Kotańska, Magdalena, Stark, Holger, Elz, Sigurd, Kieć-Kononowicz, Katarzyna
Published in European journal of medicinal chemistry (05.03.2021)
Published in European journal of medicinal chemistry (05.03.2021)
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Journal Article
Structural modifications in the distal, regulatory region of histamine H-3 receptor antagonists leading to the identification of a potent anti-obesity agent
Szczepanska, Katarzyna, Pockes, Steffen, Podlewska, Sabina, Horing, Carina, Mika, Kamil, Latacz, Gniewomir, Bednarski, Marek, Siwek, Agata, Karcz, Tadeusz, Nagl, Martin, Bresinsky, Merlin, Monnich, Denise, Seibel, Ulla, Kuder, Kamil J., Kotanska, Magdalena, Stark, Holger, Elz, Sigurd, Kiec-Kononowicz, Katarzyna
Published in European journal of medicinal chemistry (05.03.2021)
Published in European journal of medicinal chemistry (05.03.2021)
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Journal Article
Characterization of caspase‐2 inhibitors based on specific sites of caspase‐2‐mediated proteolysis
Bresinsky, Merlin, Strasser, Jessica M., Hubmann, Alexander, Vallaster, Bernadette, McCue, William M., Fuller, Jessica, Singh, Gurpreet, Nelson, Kathryn M., Cuellar, Matthew E., Finzel, Barry C., Ashe, Karen H., Walters, Michael A., Pockes, Steffen
Published in Archiv der Pharmazie (Weinheim) (01.09.2022)
Published in Archiv der Pharmazie (Weinheim) (01.09.2022)
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Journal Article
Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H 2 R and D 3 R
Biselli, Sabrina, Bresinsky, Merlin, Tropmann, Katharina, Forster, Lisa, Honisch, Claudia, Buschauer, Armin, Bernhardt, Günther, Pockes, Steffen
Published in European journal of medicinal chemistry (15.03.2021)
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Published in European journal of medicinal chemistry (15.03.2021)
Journal Article
Caspase‑2 Inhibitor Blocks Tau Truncation and Restores Excitatory Neurotransmission in Neurons Modeling FTDP-17 Tauopathy
Singh, Gurpreet, Liu, Peng, Yao, Katherine R., Strasser, Jessica M., Hlynialuk, Chris, Leinonen-Wright, Kailee, Teravskis, Peter J., Choquette, Jessica M., Ikramuddin, Junaid, Bresinsky, Merlin, Nelson, Kathryn M., Liao, Dezhi, Ashe, Karen H., Walters, Michael A., Pockes, Steffen
Published in ACS chemical neuroscience (18.05.2022)
Published in ACS chemical neuroscience (18.05.2022)
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Journal Article
Structure-Based Design and Biological Evaluation of Novel Caspase‑2 Inhibitors Based on the Peptide AcVDVAD-CHO and the Caspase-2-Mediated Tau Cleavage Sequence YKPVD314
Bresinsky, Merlin, Strasser, Jessica M, Vallaster, Bernadette, Liu, Peng, McCue, William M, Fuller, Jessica, Hubmann, Alexander, Singh, Gurpreet, Nelson, Kathryn M, Cuellar, Matthew E, Wilmot, Carrie M, Finzel, Barry C, Ashe, Karen H, Walters, Michael A, Pockes, Steffen
Published in ACS pharmacology & translational science (14.01.2022)
Published in ACS pharmacology & translational science (14.01.2022)
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Journal Article
PROTEASE INHIBITORS
WALTERS, Michael A, ASHE, Karen, HUBMANN, Alexander, POCKES, Steffen, BRESINSKY, Merlin, LIAO, Dezhi, SINGH, Gurpreet
Year of Publication 31.08.2023
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Year of Publication 31.08.2023
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