KLS-13019, a novel structural analogue of cannabidiol (CBD) and GPR55 receptor antagonist, Prevents and Reverses Chemotherapy-Induced Peripheral Neuropathy (CIPN) in Rats
Ippolito, Michael J, Kinney, William, Brenneman, Douglas E, Ward, Sara Jane, Hayduk, Sean A
Published in The Journal of pharmacology and experimental therapeutics (12.08.2024)
Published in The Journal of pharmacology and experimental therapeutics (12.08.2024)
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Knockdown siRNA Targeting the Mitochondrial Sodium-Calcium Exchanger-1 Inhibits the Protective Effects of Two Cannabinoids Against Acute Paclitaxel Toxicity
Brenneman, Douglas E., Kinney, William A., Ward, Sara Jane
Published in Journal of molecular neuroscience (01.08.2019)
Published in Journal of molecular neuroscience (01.08.2019)
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Pharmacological Comparisons Between Cannabidiol and KLS-13019
Brenneman, Douglas E., Petkanas, Dean, Kinney, William A.
Published in Journal of molecular neuroscience (01.09.2018)
Published in Journal of molecular neuroscience (01.09.2018)
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Behavioural and pharmacological effects of cannabidiol (CBD) and the cannabidiol analogue KLS‐13019 in mouse models of pain and reinforcement
Foss, Jeffery D., Farkas, Daniel J., Huynh, Lana M., Kinney, William A., Brenneman, Douglas E., Ward, Sara Jane
Published in British journal of pharmacology (01.08.2021)
Published in British journal of pharmacology (01.08.2021)
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Knockdown siRNA Targeting GPR55 Reveals Significant Differences Between the Anti-inflammatory Actions of KLS-13019 and Cannabidiol
Brenneman, Douglas E., Kinney, William A., McDonnell, Mark E., Ippolito, Michael J., Ward, Sara Jane
Published in Journal of molecular neuroscience (11.04.2024)
Published in Journal of molecular neuroscience (11.04.2024)
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Anti-Inflammatory Properties of KLS-13019: a Novel GPR55 Antagonist for Dorsal Root Ganglion and Hippocampal Cultures
Brenneman, Douglas E., Kinney, William A., McDonnell, Mark E., Zhao, Pingei, Abood, Mary E., Ward, Sara Jane
Published in Journal of molecular neuroscience (01.09.2022)
Published in Journal of molecular neuroscience (01.09.2022)
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Discovery of KLS-13019, a Cannabidiol-Derived Neuroprotective Agent, with Improved Potency, Safety, and Permeability
Kinney, William A, McDonnell, Mark E, Zhong, Hua Marlon, Liu, Chaomin, Yang, Lanyi, Ling, Wei, Qian, Tao, Chen, Yu, Cai, Zhijie, Petkanas, Dean, Brenneman, Douglas E
Published in ACS medicinal chemistry letters (14.04.2016)
Published in ACS medicinal chemistry letters (14.04.2016)
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NAP and ADNF-9 Protect Normal and Downs Syndrome Cortical Neurons from Oxidative Damage and Apoptosis
Busciglio, Jorge, Pelsman, Alejandra, Helguera, Pablo, Ashur-Fabian, Osnat, Pinhasov, Albert, Brenneman, Douglas E, Gozes, Illana
Published in Current pharmaceutical design (01.04.2007)
Published in Current pharmaceutical design (01.04.2007)
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2-Amino-3,4-dihydroquinazolines as Inhibitors of BACE-1 (β-Site APP Cleaving Enzyme): Use of Structure Based Design to Convert a Micromolar Hit into a Nanomolar Lead
Baxter, Ellen W, Conway, Kelly A, Kennis, Ludo, Bischoff, François, Mercken, Marc H, De Winter, Hans L, Reynolds, Charles H, Tounge, Brett A, Luo, Chi, Scott, Malcolm K, Huang, Yifang, Braeken, Mirielle, Pieters, Serge M. A, Berthelot, Didier J. C, Masure, Stefan, Bruinzeel, Wouter D, Jordan, Alfonzo D, Parker, Michael H, Boyd, Robert E, Qu, Junya, Alexander, Richard S, Brenneman, Douglas E, Reitz, Allen B
Published in Journal of medicinal chemistry (06.09.2007)
Published in Journal of medicinal chemistry (06.09.2007)
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Novel, Broad-Spectrum Anticonvulsants Containing a Sulfamide Group: Pharmacological Properties of (S)‑N‑[(6-Chloro-2,3-dihydrobenzo[1,4]dioxin-2-yl)methyl]sulfamide (JNJ-26489112)
McComsey, David F, Smith-Swintosky, Virginia L, Parker, Michael H, Brenneman, Douglas E, Malatynska, Ewa, White, H. Steve, Klein, Brian D, Wilcox, Karen S, Milewski, Michael E, Herb, Mark, Finley, Michael F. A, Liu, Yi, Lubin, Mary Lou, Qin, Ning, Reitz, Allen B, Maryanoff, Bruce E
Published in Journal of medicinal chemistry (27.11.2013)
Published in Journal of medicinal chemistry (27.11.2013)
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The expression of activity-dependent neuroprotective protein (ADNP) is regulated by brain damage and treatment of mice with the ADNP derived peptide, NAP, reduces the severity of traumatic head injury
Gozes, Illana, Zaltzman, Roy, Hauser, Janet, Brenneman, Douglas E, Shohami, Esther, Hill, Joanna M
Published in Current Alzheimer research (01.04.2005)
Published in Current Alzheimer research (01.04.2005)
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A Glia-Derived Signal Regulating Neuronal Differentiation
Blondel, Olivier, Collin, Carlos, McCarran, William J, Zhu, Shiaoping, Zamostiano, Rachel, Gozes, Illana, Brenneman, Douglas E, McKay, Ronald D. G
Published in The Journal of neuroscience (01.11.2000)
Published in The Journal of neuroscience (01.11.2000)
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NAP, a femtomolar-acting peptide, protects the brain against ischemic injury by reducing apoptotic death
LEKER, Ronen R, TEICHNER, Angella, GRIGORIADIS, Nikolas, OVADIA, Haim, BRENNEMAN, Douglas E, FRIDKIN, Mati, GILADI, Eli, ROMANO, Jacob, GOZES, Illana
Published in Stroke (1970) (01.04.2002)
Published in Stroke (1970) (01.04.2002)
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Differential Effects of Ethanol Antagonism and Neuroprotection in Peptide Fragment NAPVSIPQ Prevention of Ethanol-Induced Developmental Toxicity
Wilkemeyer, Michael F., Chen, Shao-yu, Menkari, Carrie E., Brenneman, Douglas E., Sulik, Kathleen K., Charness, Michael E.
Published in Proceedings of the National Academy of Sciences - PNAS (08.07.2003)
Published in Proceedings of the National Academy of Sciences - PNAS (08.07.2003)
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Carisbamate, a novel neuromodulator, inhibits voltage-gated sodium channels and action potential firing of rat hippocampal neurons
Liu, Yi, Yohrling, George J, Wang, Yan, Hutchinson, Tasha L, Brenneman, Douglas E, Flores, Christopher M, Zhao, Boyu
Published in Epilepsy research (01.01.2009)
Published in Epilepsy research (01.01.2009)
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Reduction of dominant or submissive behaviors as models for antimanic or antidepressant drug testing: Technical considerations
Malatynska, Ewa, Pinhasov, Albert, Crooke, Jeffrey J., Smith-Swintosky, Virginia L., Brenneman, Douglas E.
Published in Journal of neuroscience methods (30.09.2007)
Published in Journal of neuroscience methods (30.09.2007)
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