Ligands for Glutamate Receptors: Design and Therapeutic Prospects
Bräuner-Osborne, Hans, Egebjerg, Jan, Nielsen, Elsebet Ø, Madsen, Ulf, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (13.07.2000)
Published in Journal of medicinal chemistry (13.07.2000)
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The GPCR, class C, group 6, subtype A (GPRC6A) receptor: from cloning to physiological function
Clemmensen, C, Smajilovic, S, Wellendorph, P, Bräuner‐Osborne, H
Published in British journal of pharmacology (01.03.2014)
Published in British journal of pharmacology (01.03.2014)
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The orthosteric GABAA receptor ligand Thio‐4‐PIOL displays distinctly different functional properties at synaptic and extrasynaptic receptors
Hoestgaard‐Jensen, K, O'Connor, R M, Dalby, N O, Simonsen, C, Finger, B C, Golubeva, A, Hammer, H, Bergmann, M L, Kristiansen, U, Krogsgaard‐Larsen, P, Bräuner‐Osborne, H, Ebert, B, Frølund, B, Cryan, J F, Jensen, A A
Published in British journal of pharmacology (01.10.2013)
Published in British journal of pharmacology (01.10.2013)
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Journal Article
1,2,3-Triazolyl amino acids as AMPA receptor ligands
Stanley, N.J., Pedersen, D. Sejer, Nielsen, B., Kvist, T., Mathiesen, J.M., Bräuner-Osborne, H., Taylor, D.K., Abell, A.D.
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
Published in Bioorganic & medicinal chemistry letters (15.12.2010)
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Agonists and Inverse Agonists for the Herpesvirus 8-encoded Constitutively Active Seven-transmembrane Oncogene Product, ORF-74
Rosenkilde, Mette M., Kledal, Thomas N., Bräuner-Osborne, Hans, Schwartz, Thue W.
Published in The Journal of biological chemistry (08.01.1999)
Published in The Journal of biological chemistry (08.01.1999)
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Journal Article
Synthesis and Pharmacology of a New AMPA−Kainate Receptor Agonist with Potent Convulsant Activity
Conti, Paola, De Amici, Marco, De Sarro, Giovambattista, Stensbøl, Tine Bryan, Bräuner-Osborne, Hans, Madsen, Ulf, De Micheli, Carlo
Published in Journal of medicinal chemistry (24.09.1998)
Published in Journal of medicinal chemistry (24.09.1998)
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Functional importance of the Ala(116)-Pro(136) region in the calcium-sensing receptor. Constitutive activity and inverse agonism in a family C G-protein-coupled receptor
Jensen, A A, Spalding, T A, Burstein, E S, Sheppard, P O, O'Hara, P J, Brann, M R, Krogsgaard-Larsen, P, Bräuner-Osborne, H
Published in The Journal of biological chemistry (22.09.2000)
Published in The Journal of biological chemistry (22.09.2000)
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Journal Article
Synthesis and Enantiopharmacology of New AMPA-Kainate Receptor Agonists
Conti, Paola, De Amici, Marco, De Sarro, Giovambattista, Rizzo, Milena, Stensbøl, Tine Bryan, Bräuner-Osborne, Hans, Madsen, Ulf, Toma, Lucio, De Micheli, Carlo
Published in Journal of medicinal chemistry (07.10.1999)
Published in Journal of medicinal chemistry (07.10.1999)
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Journal Article
A New Highly Selective Metabotropic Excitatory Amino Acid Agonist: 2-Amino-4-(3-hydroxy-5-methylisoxazol-4-yl)butyric Acid
Bräuner-Osborne, Hans, Sløk, Frank A, Skjærbæk, Niels, Ebert, Bjarke, Sekiyama, Naohiro, Nakanishi, Shigetada, Krogsgaard-Larsen, Povl
Published in Journal of medicinal chemistry (02.08.1996)
Published in Journal of medicinal chemistry (02.08.1996)
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