Influence of Transporter Polymorphisms on Drug Disposition and Response: A Perspective From the International Transporter Consortium
Yee, Sook Wah, Brackman, Deanna J, Ennis, Elizabeth A, Sugiyama, Yuichi, Kamdem, Landry K, Blanchard, Rebecca, Galetin, Aleksandra, Zhang, Lei, Giacomini, Kathleen M
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Journal Article
A conserved role of the insulin-like signaling pathway in diet-dependent uric acid pathologies in Drosophila melanogaster
Lang, Sven, Hilsabeck, Tyler A, Wilson, Kenneth A, Sharma, Amit, Bose, Neelanjan, Brackman, Deanna J, Beck, Jennifer N, Chen, Ling, Watson, Mark A, Killilea, David W, Ho, Sunita, Kahn, Arnold, Giacomini, Kathleen, Stoller, Marshall L, Chi, Thomas, Kapahi, Pankaj
Published in PLoS genetics (15.08.2019)
Published in PLoS genetics (15.08.2019)
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Journal Article
Reverse Translational Research of ABCG2 (BCRP) in Human Disease and Drug Response
Brackman, Deanna J, Giacomini, Kathleen M
Published in Clinical pharmacology and therapeutics (01.02.2018)
Published in Clinical pharmacology and therapeutics (01.02.2018)
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Journal Article
Venetoclax Plus Gilteritinib for FLT3 -Mutated Relapsed/Refractory Acute Myeloid Leukemia
Daver, Naval, Perl, Alexander E, Maly, Joseph, Levis, Mark, Ritchie, Ellen, Litzow, Mark, McCloskey, James, Smith, Catherine C, Schiller, Gary, Bradley, Terrence, Tiu, Ramon V, Naqvi, Kiran, Dail, Monique, Brackman, Deanna, Siddani, Satya, Wang, Jing, Chyla, Brenda, Lee, Paul, Altman, Jessica K
Published in Journal of clinical oncology (10.12.2022)
Published in Journal of clinical oncology (10.12.2022)
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Journal Article
Impact of Multiple Concomitant CYP3A Inhibitors on Venetoclax Pharmacokinetics: A PBPK and Population PK-Informed Analysis
Mukherjee, Dwaipayan, Brackman, Deanna J, Suleiman, Ahmed A, Zha, Jiuhong, Menon, Rajeev M, Salem, Ahmed Hamed
Published in Journal of clinical pharmacology (01.01.2023)
Published in Journal of clinical pharmacology (01.01.2023)
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Journal Article
PharmGKB summary: very important pharmacogene information for ABCG2
Fohner, Alison E, Brackman, Deanna J, Giacomini, Kathleen M, Altman, Russ B, Klein, Teri E
Published in Pharmacogenetics and genomics (01.11.2017)
Published in Pharmacogenetics and genomics (01.11.2017)
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Journal Article
Genome-Wide Association and Functional Studies Reveal Novel Pharmacological Mechanisms for Allopurinol
Brackman, Deanna J, Yee, Sook Wah, Enogieru, Osatohanmwen J, Shaffer, Christian, Ranatunga, Dilrini, Denny, Joshua C, Wei, Wei-Qi, Kamatani, Yoichiro, Kubo, Michiaki, Roden, Dan M, Jorgenson, Eric, Giacomini, Kathleen M
Published in Clinical pharmacology and therapeutics (01.09.2019)
Published in Clinical pharmacology and therapeutics (01.09.2019)
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Journal Article
Oxypurinol pharmacokinetics and pharmacodynamics in healthy volunteers: Influence of BCRP Q141K polymorphism and patient characteristics
Vora, Bianca, Brackman, Deanna J., Zou, Ling, Garcia‐Cremades, Maria, Sirota, Marina, Savic, Radojka M., Giacomini, Kathleen M.
Published in Clinical and translational science (01.07.2021)
Published in Clinical and translational science (01.07.2021)
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Journal Article
Efficient Delivery of the Toll-like Receptor Agonists Polyinosinic:Polycytidylic Acid and CpG to Macrophages by Acetalated Dextran Microparticles
Peine, Kevin J, Bachelder, Eric M, Vangundy, Zachary, Papenfuss, Tracy, Brackman, Deanna J, Gallovic, Mathew D, Schully, Kevin, Pesce, John, Keane-Myers, Andrea, Ainslie, Kristy M
Published in Molecular pharmaceutics (05.08.2013)
Published in Molecular pharmaceutics (05.08.2013)
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Journal Article
Electrospun Acetalated Dextran Scaffolds for Temporal Release of Therapeutics
Borteh, Hassan M, Gallovic, Matthew D, Sharma, Sadhana, Peine, Kevin J, Miao, Simeng, Brackman, Deanna J, Gregg, Katie, Xu, Yanyi, Guo, Xiaolei, Guan, Jianjun, Bachelder, Eric M, Ainslie, Kristy M
Published in Langmuir (25.06.2013)
Published in Langmuir (25.06.2013)
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Journal Article
A First-in-Human Phase 1 Study of Abbv-319, an Antibody-Drug Conjugate Composed of a CD19 Antibody Linked to a Potent Proprietary Glucocorticoid Receptor Modulator, in Patients with Relapsed or Refractory B-Cell Malignancies
Levy, Moshe, Gustafson, Carl, Purcell, James, Freise, Kevin J., Assaily, Wissam, Brackman, Deanna, Henner, William R., McDevitt, Michael, Kuruvilla, John
Published in Blood (15.11.2022)
Published in Blood (15.11.2022)
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Journal Article
Two Phase 1b Studies Evaluating the Safety and Tolerability of BET Inhibitors, ABBV-744 and Mivebresib, as Monotherapies and in Combination with Ruxolitinib or Navitoclax in Patients with Myelofibrosis
Mascarenhas, John, Saab, Rabih, Brackman, Deanna, Modi, Dimple A., Abraham, Linu, Ward, James E., Verstovsek, Srdan
Published in Blood (05.11.2020)
Published in Blood (05.11.2020)
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Journal Article
Venetoclax Exposure-Efficacy and Exposure-Safety Relationships in Subjects with Treatment-Naïve Acute Myeloid Leukemia Who Are Ineligible for Intensive Chemotherapy
Eckert, Doerthe, Brackman, Deanna, Menon, Rajeev, Salem, Ahmed Hamed, Potluri, Jalaja, Smith, B. Douglas, Wei, Andrew H., Hayslip, John, Miles, Dale, Mensing, Sven, Gopalakrishnan, Sathej, Zha, Jiuhong
Published in Blood (05.11.2020)
Published in Blood (05.11.2020)
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Journal Article
Risk-Based Pharmacokinetic and Drug-Drug Interaction Characterization of Antibody-Drug Conjugates in Oncology Clinical Development: An International Consortium for Innovation and Quality in Pharmaceutical Development Perspective
Li, Chunze, Menon, Rajeev, Walles, Markus, Singh, Renu, Upreti, Vijay V, Brackman, Deanna, Lee, Anthony J, Endres, Christopher J, Kumar, Seema, Zhang, Donglu, Barletta, Frank, Suri, Ajit, Hainzl, Dominik, Liao, Kai H, Lalovic, Bojan, Beaumont, Maribel, Zuo, Peiying, Mayer, Andrew P, Wei, Dong
Published in Clinical pharmacology and therapeutics (01.10.2022)
Published in Clinical pharmacology and therapeutics (01.10.2022)
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Journal Article
Postremission cytopenia management in patients with acute myeloid leukemia treated with venetoclax and azacitidine in VIALE‐A
Pratz, Keith W., DiNardo, Courtney D., Selleslag, Dominik, Li, Junmin, Yamamoto, Kazuhito, Konopleva, Marina, Stevens, Don, Kantarjian, Hagop, Traina, Fabiola, Venditti, Adriano, Mayer, Jiri, Montez, Melissa, Jin, Huan, Duan, Yinghui, Brackman, Deanna, Zha, Jiuhong, Potluri, Jalaja, Werner, Michael, Jonas, Brian A.
Published in American journal of hematology (01.11.2022)
Published in American journal of hematology (01.11.2022)
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Journal Article
Venetoclax exposure‐efficacy and exposure‐safety relationships in patients with treatment‐naïve acute myeloid leukemia who are ineligible for intensive chemotherapy
Brackman, Deanna, Eckert, Doerthe, Menon, Rajeev, Salem, Ahmed Hamed, Potluri, Jalaja, Smith, B. Douglas, Wei, Andrew H., Hayslip, John, Miles, Dale, Mensing, Sven, Gopalakrishnan, Sathej, Zha, Jiuhong
Published in Hematological oncology (01.04.2022)
Published in Hematological oncology (01.04.2022)
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Journal Article
A phase 1b study of venetoclax and alvocidib in patients with relapsed/refractory acute myeloid leukemia
Jonas, Brian A, Hou, Jing-Zhou, Roboz, Gail J, Alvares, Caroline L, Jeyakumar, Deepa, Edwards, John R, Erba, Harry P, Kelly, Richard J, Röllig, Christoph, Fiedler, Walter, Brackman, Deanna, Siddani, Satya R, Chyla, Brenda, Hilger-Rolfe, Jacqueline, Watts, Justin M
Published in Hematological oncology (01.10.2023)
Published in Hematological oncology (01.10.2023)
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