Synthesis of Mono- and Difluoronaphthoic Acids
Tagat, Jayaram R, McCombie, Stuart W, Nazareno, Dennis V, Boyle, Craig D, Kozlowski, Joseph A, Chackalamannil, Samuel, Josien, Hubert, Wang, Yuguang, Zhou, Guowei
Published in Journal of organic chemistry (22.02.2002)
Published in Journal of organic chemistry (22.02.2002)
Get full text
Journal Article
Azabicyclic sulfonamides as potent 11β-HSD1 inhibitors
Shah, Unmesh, Boyle, Craig D., Chackalamannil, Samuel, Baker, Hana, Kowalski, Timothy, Lee, Julie, Terracina, Giuseppe, Zhang, Lili
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Get full text
Journal Article
Design, synthesis, and evaluation of fused heterocyclic analogs of SCH 58261 as adenosine A2A receptor antagonists
SHAH, Unmesh, LANKIN, Claire M, HONGTAO ZHANG, LACHOWICZ, Jean E, BOYLE, Craig D, CHACKALAMANNIL, Samuel, GREENLEE, William J, NEUSTADT, Bernard R, COHEN-WILLIAMS, Mary E, HIGGINS, Guy A, NG, Kwokei, VARTY, Geoffrey B
Published in Bioorganic & medicinal chemistry letters (01.07.2008)
Published in Bioorganic & medicinal chemistry letters (01.07.2008)
Get full text
Journal Article
Design, synthesis, and evaluation of fused heterocyclic analogs of SCH 58261 as adenosine A2A receptor antagonists
Shah, Unmesh, Lankin, Claire M, Boyle, Craig D, Chackalamannil, Samuel, Greenlee, William J, Neustadt, Bernard R, Cohen-Williams, Mary E, Higgins, Guy A, Ng, Kwokei, Varty, Geoffrey B, Zhang, Hongtao, Lachowicz, Jean E
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Get full text
Journal Article
Biaryl and heteroaryl derivatives of SCH 58261 as potent and selective adenosine A2A receptor antagonists
SHAH, Unmesh, BOYLE, Craig D, SHIYONG WANG, MONOPOLI, Angela, LACHOWICZ, Jean E, CHACKALAMANNIL, Samuel, NEUSTADT, Bernard R, LINDO, Neil, GREENLEE, William J, FOSTER, Carolyn, ARIK, Leyla, YING ZHAI, NG, Kwokei
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Get full text
Journal Article
Optimization of purine based PDE1/PDE5 inhibitors to a potent and selective PDE5 inhibitor for the treatment of male ED
Boyle, Craig D., Xu, Ruo, Asberom, Theodros, Chackalamannil, Samuel, Clader, John W., Greenlee, William J., Guzik, Henry, Hu, Yuequing, Hu, Zhiyong, Lankin, Claire M., Pissarnitski, Dmitri A., Stamford, Andrew W., Wang, Yuguang, Skell, Jeffrey, Kurowski, Stanley, Vemulapalli, Subbarao, Palamanda, Jairam, Chintala, Madhu, Wu, Ping, Myers, Joyce, Wang, Peng
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Get full text
Journal Article
SAR development of polycyclic guanine derivatives targeted to the discovery of a selective PDE5 inhibitor for treatment of erectile dysfunction
PISSARNITSKI, Dmitri A, ASBEROM, Theodros, PALAMANDA, Jairam, STAMFORD, Andrew W, VEMULAPALLI, Subbarao, YUGUANG WANG, PENG WANG, PING WU, RUO XU, BOYLE, Craig D, CHACKALAMANNIL, Samuel, CHINTALA, Madhu, CLADER, John W, GREENLEE, William J, YUEQING HU, KUROWSKI, Stanley, MYERS, Joyce
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Published in Bioorganic & medicinal chemistry letters (08.03.2004)
Get full text
Journal Article
Novel Structure Elucidation of AAL Toxin TA Backbone
Boyle, Craig D, Harmange, Jean-Christophe, Kishi, Yoshito
Published in Journal of the American Chemical Society (01.06.1994)
Published in Journal of the American Chemical Society (01.06.1994)
Get full text
Journal Article
Design and synthesis of xanthine analogues as potent and selective PDE5 inhibitors
Wang, Yuguang, Chackalamannil, Samuel, Hu, Zhiyong, Boyle, Craig D, Lankin, Claire M, Xia, Yan, Xu, Ruo, Asberom, Theodros, Pissarnitski, Dmitri, Stamford, Andrew W, Greenlee, William J, Skell, Jeffrey, Kurowski, Stanley, Vemulapalli, Subbarao, Palamanda, Jairam, Chintala, Madhu, Wu, Ping, Myers, Joyce, Wang, Peng
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Get full text
Journal Article
Improving the Oral Efficacy of CNS Drug Candidates: Discovery of Highly Orally Efficacious Piperidinyl Piperidine M2 Muscarinic Receptor Antagonists
Wang, Yuguang, Chackalamannil, Samuel, Hu, Zhiyong, Greenlee, William J, Clader, John, Boyle, Craig D, Kaminski, James J, Billard, William, Binch, Crosby, Gordon, Ruperto, Vilma, Duffy, Ruth A, Cohen-Williams, Mary, Coffin, Vicki L, Cox, Kathleen A, Grotz, Diane E, Lachowicz, Jean E
Published in Journal of medicinal chemistry (05.12.2002)
Published in Journal of medicinal chemistry (05.12.2002)
Get full text
Journal Article
Enhancement of pharmacokinetic properties and in vivo efficacy of benzylidene ketal M2 muscarinic receptor antagonists via benzamide modification
BOYLE, Craig D, VICE, Susan F, COFFIN, Vicki L, COX, Kathleen A, GROTZ, Diane E, DUFFY, Ruth A, RUPERTO, Vilma, LACHOWICZ, Jean E, CAMPION, Jennifer, CHACKALAMANNIL, Samuel, LANKIN, Claire M, MCCOMBIE, Stuart W, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, WILLIAMS, Mary-Cohen
Published in Bioorganic & medicinal chemistry letters (01.12.2002)
Published in Bioorganic & medicinal chemistry letters (01.12.2002)
Get full text
Journal Article
Metabolic stabilization of benzylidene ketal M2 muscarinic receptor antagonists via halonaphthoic acid substitution
BOYLE, Craig D, CHACKALAMANNIL, Samuel, YUGUANG WANG, GUOWEI ZHOU, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, COHEN-WILLIAMS, Mary, COFFIN, Vicki L, COX, Kathleen A, GROTZ, Diane E, DUFFY, Ruth A, CLADER, John W, RUPERTO, Vilma, LACHOWICZ, Jean E, GREENLEE, William J, JOSIEN, Hubert B, KAMINSKI, James J, KOZLOWSKI, Joseph A, MCCOMBIE, Stuart W, NAZARENO, Dennis V, TAGAT, Jayaram R
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Get full text
Journal Article
Benzylidene ketal derivatives as M2 muscarinic receptor antagonists
BOYLE, Craig D, CHACKALAMANNIL, Samuel, DUFFY, Ruth A, RUPERTO, Vilma, LACHOWICZ, Jean E, CHEN, Lian-Yong, DUGAR, Sundeep, PUSHPAVANAM, Pradeep, BILLARD, William, BINCH, Herbert III, CROSBY, Gordon, COHEN-WILLIAMS, Mary, COFFIN, Vicki L
Published in Bioorganic & medicinal chemistry letters (18.12.2000)
Published in Bioorganic & medicinal chemistry letters (18.12.2000)
Get full text
Journal Article
BICYCLIC HETEROCYCLE DERIVATIVES AND THEIR USE AS MODULATORS OF THE ACTIVITY OF GPR119
CHACKALAMANNIL SAMUEL, SHAH UNMESH G, LANKIN CLAIRE M, BOYLE CRAIG D, DAI XING, HARRIS JOEL M, XIA YAN, GREENLEE WILLIAM J, LIU HONG, STAMFORD ANDREW W, NEUSTADT BERNARD R, NEELAMKAVIL SANTHOSH FRANCIS, JAYNE CHARLES LEE
Year of Publication 02.07.2010
Get full text
Year of Publication 02.07.2010
Patent
Azabicyclic sulfonamides as potent 11b-HSD1 inhibitors
Shah, Unmesh, Boyle, Craig D, Chackalamannil, Samuel, Baker, Hana, Kowalski, Timothy, Lee, Julie, Terracina, Giuseppe, Zhang, Lili
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Get full text
Journal Article
Relative and absolute stereochemistry of the fumonisin B2 backbone
Harmange, Jean-Christophe, Boyle, Craig D., Kishi, Yoshito
Published in Tetrahedron letters (01.09.1994)
Published in Tetrahedron letters (01.09.1994)
Get full text
Journal Article