Discovery of new inhibitors of the bacterial peptidoglycan biosynthesis enzymes MurD and MurF by structure-based virtual screening
Turk, Samo, Kovač, Andreja, Boniface, Audrey, Bostock, Julieanne M., Chopra, Ian, Blanot, Didier, Gobec, Stanislav
Published in Bioorganic & medicinal chemistry (01.03.2009)
Published in Bioorganic & medicinal chemistry (01.03.2009)
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Journal Article
nature of Staphylococcus aureus MurA and MurZ and approaches for detection of peptidoglycan biosynthesis inhibitors
Blake, Katy L, O'Neill, Alex J, Mengin-Lecreulx, Dominique, Henderson, Peter J.F, Bostock, Julieanne M, Dunsmore, Colin J, Simmons, Katie J, Fishwick, Colin W.G, Leeds, Jennifer A, Chopra, Ian
Published in Molecular microbiology (01.04.2009)
Published in Molecular microbiology (01.04.2009)
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Journal Article
Diazenedicarboxamides as inhibitors of d-alanine- d-alanine ligase (Ddl)
Kovač, Andreja, Majce, Vita, Lenaršič, Roman, Bombek, Sergeja, Bostock, Julieanne M., Chopra, Ian, Polanc, Slovenko, Gobec, Stanislav
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
Published in Bioorganic & medicinal chemistry letters (01.04.2007)
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Journal Article
A De Novo Designed Inhibitor of D-Ala-D-Ala Ligase from E. coli
Besong, Gilbert E., Bostock, Julieanne M., Stubbings, Will, Chopra, Ian, Roper, David I., Lloyd, Adrian J., Fishwick, Colin W. G., Johnson, A. Peter
Published in Angewandte Chemie (International ed.) (07.10.2005)
Published in Angewandte Chemie (International ed.) (07.10.2005)
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Journal Article
Evolution of extended-spectrum β-lactamases in a MutS-deficient Pseudomonas aeruginosa hypermutator
Driffield, Kiersten L., Bostock, Julieanne M., Miller, Keith, O'Neill, Alexander J., Hobbs, Joanne K., Chopra, Ian
Published in Journal of antimicrobial chemotherapy (01.10.2006)
Published in Journal of antimicrobial chemotherapy (01.10.2006)
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Journal Article
Macrocyclic inhibitors of the bacterial cell wall biosynthesis enzyme mur D
Horton, James R., Bostock, Julieanne M., Chopra, Ian, Hesse, Lars, Phillips, Simon E.V., Adams, David J., Johnson, A.Peter, Fishwick, Colin W.G.
Published in Bioorganic & medicinal chemistry letters (05.05.2003)
Published in Bioorganic & medicinal chemistry letters (05.05.2003)
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Journal Article
Mecillinam has potent in vitro activity against Chlamydophila pneumoniae ATCC VR1310
Bostock, Julieanne M., Geary, Ian, Eley, Adrian, Chopra, Ian
Published in Journal of antimicrobial chemotherapy (01.06.2004)
Published in Journal of antimicrobial chemotherapy (01.06.2004)
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Journal Article
Zeocin resistance suppresses mutation in hypermutable Escherichia coli
Bostock, Julieanne M, Miller, Keith, O'Neill, Alexander J, Chopra, Ian
Published in Microbiology (Society for General Microbiology) (01.04.2003)
Published in Microbiology (Society for General Microbiology) (01.04.2003)
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Journal Article
Evolution of extended-spectrum b-lactamases in a MutS-deficient Pseudomonas aeruginosa hypermutator
Driffield, Kiersten L, Bostock, Julieanne M, Miller, Keith, O'Neill, Alexander J, Hobbs, Joanne K, Chopra, Ian
Published in Journal of antimicrobial chemotherapy (01.10.2006)
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Published in Journal of antimicrobial chemotherapy (01.10.2006)
Journal Article
Macrocyclic inhibitors of the bacterial cell wall biosynthesis enzyme MurD
Horton, James R, Bostock, Julieanne M, Chopra, Ian, Hesse, Lars, Phillips, Simon E V, Adams, David J, Johnson, A Peter, Fishwick, Colin W G
Published in Bioorganic & medicinal chemistry letters (05.05.2003)
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Published in Bioorganic & medicinal chemistry letters (05.05.2003)
Journal Article
A De Novo Designed Inhibitor of D-Ala-D-Ala Ligase from E. coli
Besong, Gilbert E., Bostock, Julieanne M., Stubbings, Will, Chopra, Ian, Roper, David I., Lloyd, Adrian J., Fishwick, Colin W. G., Johnson, A. Peter
Published in Angewandte Chemie (07.10.2005)
Published in Angewandte Chemie (07.10.2005)
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Journal Article
A De Novo Designed Inhibitor of D ‐Ala– D ‐Ala Ligase from E. coli
Besong, Gilbert E., Bostock, Julieanne M., Stubbings, Will, Chopra, Ian, Roper, David I., Lloyd, Adrian J., Fishwick, Colin W. G., Johnson, A. Peter
Published in Angewandte Chemie (07.10.2005)
Published in Angewandte Chemie (07.10.2005)
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Journal Article
Macrocyclic Inhibitors of the Bacterial Cell Wall Biosynthesis Enzyme MurD
Horton, James R., Bostock, Julieanne M., Chopra, Ian, Hesse, Lars, Phillips, Simon E. V., Adams, David J., Johnson, A. Peter, Fishwick, Colin W. G.
Published in ChemInform (29.07.2003)
Published in ChemInform (29.07.2003)
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