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Published in Scientia pharmaceutica (18.11.2021)
Published in Scientia pharmaceutica (18.11.2021)
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Synthesis, in silico and in vitro antimicrobial activity of N-(benzyl)-5-methyl-4-oxo-3,4-dihydrothieno[2,3-d]pyrimidine-6-carboxamides
Vlasov, Sergiy V, Borysov, Oleksandr V, Severina, Hanna I, Vlasov, Vitaliy S, Abu Sharkh, Amjad Ibrahim M, Georgiyants, Victoriya A
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Published in Farmacija (29.01.2024)
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Synthesis and Antimicrobial Evaluation of 2-(6-Imidazo[1,2-a]pyridin-2-yl-5-methyl-2,4-dioxo-3-phenyl-3,4-dihydrothieno[2,3-d]pyrimidin-1(2H)-yl)-N-arylacetamide Derivatives
Vlasov, Sergiy V., Severina, Hanna I., Borysov, Oleksandr V., Krolenko, Konstantin Yu, Shynkarenko, Pavlo E., Saidov, Narzullo B., Vlasov, Vitaliy S., Georgiyants, Victoriya A.
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Published in MolBank (01.03.2022)
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Spiropyran‐Based Photoisomerizable α‐Amino Acid for Membrane‐Active Peptide Modification
Hrebonkin, Andrii, Afonin, Sergii, Nikitjuka, Anna, Borysov, Oleksandr V., Leitis, Gundars, Babii, Oleg, Koniev, Serhii, Lorig, Theo, Grage, Stephan L., Nick, Peter, Ulrich, Anne S., Jirgensons, Aigars, Komarov, Igor V.
Published in Chemistry : a European journal (16.04.2024)
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Fragment-Based Discovery of 2‑Aminoquinazolin-4(3H)‑ones As Novel Class Nonpeptidomimetic Inhibitors of the Plasmepsins I, II, and IV
Rasina, Dace, Otikovs, Martins, Leitans, Janis, Recacha, Rosario, Borysov, Oleksandr V, Kanepe-Lapsa, Iveta, Domraceva, Ilona, Pantelejevs, Teodors, Tars, Kaspars, Blackman, Michael J, Jaudzems, Kristaps, Jirgensons, Aigars
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Published in Journal of medicinal chemistry (14.01.2016)
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Synthesis of 5‑(Fluoroalkyl)isoxazole Building Blocks by Regioselective Reactions of Functionalized Halogenoximes
Chalyk, Bohdan A, Hrebeniuk, Kateryna V, Fil, Yulia V, Gavrilenko, Konstantin S, Rozhenko, Alexander B, Vashchenko, Bohdan V, Borysov, Oleksandr V, Biitseva, Angelina V, Lebed, Pavlo S, Bakanovych, Iulia, Moroz, Yurii S, Grygorenko, Oleksandr O
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Published in Journal of organic chemistry (20.12.2019)
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Electrochemical Scaled‐up Synthesis of Cyclic Enecarbamates as Starting Materials for Medicinal Chemistry Relevant Building Bocks
Tereshchenko, Oleksandr D., Perebiynis, Maryana Y., Knysh, Irina V., Vasylets, Olesia V., Sorochenko, Anna A., Slobodyanyuk, Eugeniy Y., Rusanov, Eduard B., Borysov, Oleksandr V., Kolotilov, Sergey V., Ryabukhin, Sergey V., Volochnyuk, Dmitriy M.
Published in Advanced synthesis & catalysis (04.08.2020)
Published in Advanced synthesis & catalysis (04.08.2020)
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Consistency of phenolic profiles with taxonomic distribution and adaptation of birch species ( Betula L.) to environmental conditions
Likhanov, Artur F, Vasylyshyn, Roman D, Marchuk, Yurii M, Kurdyuk, Oleksandr M, Honchar, Hanna Yu, Borysov, Oleksandr V, Bilous, Svitlana Yu, Yakubenko, Borys Ye, Al Naggar, Yahya
Published in Botany (01.10.2023)
Published in Botany (01.10.2023)
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Synthesis of methotrexate-betulonic acid hybrids and evaluation of their effect on artificial and Caco-2 cell membranes
Semenenko, Olexander M., Lipson, Victoria V., Sadchenko, Alina O., Vashchenko, Olga V., Kasian, Natalia A., Sviechnikova, Liliia, Lisetski, Longin M., Babak, Mykola L., Vakula, Volodymyr M., Borysov, Oleksandr, Holota, Yuliia, Zozulya, Sergey O., Borysko, Petro O., Mazepa, Olexander
Published in Steroids (01.01.2024)
Published in Steroids (01.01.2024)
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2-Aminoquinazolin-4(3H)-one based plasmepsin inhibitors with improved hydrophilicity and selectivity
Rasina, Dace, Stakanovs, Georgijs, Borysov, Oleksandr V., Pantelejevs, Teodors, Bobrovs, Raitis, Kanepe-Lapsa, Iveta, Tars, Kaspars, Jaudzems, Kristaps, Jirgensons, Aigars
Published in Bioorganic & medicinal chemistry (15.05.2018)
Published in Bioorganic & medicinal chemistry (15.05.2018)
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Focused small molecule library of 5,6,7,8-tetrahydro[1,2,4]triazolo-[4,3-a]pyrazines: a brick for the house of medicinal chemistry
Borysov, Oleksandr V., Voloshchuk, Volodymyr V., Nechayev, Maksym A., Lysenko, Viacheslav A., Nikolaychuk, Mykola M., Portiankin, Anton O., Oliinyk, Oleksandra V., Lega, Dmitry A., Volochnyuk, Dmitriy M., Ryabukhin, Sergey V.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.07.2023)
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.07.2023)
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The synthesis, antimicrobial activity and docking studies of 6-(1H-benzimidazol-2-yl)-5-methylthieno[2,3-d]pyrimidin- 4(3H)-ones with acetamide and 1,2,4-oxadiazol-5-ylmethyl substituents
Vlasov, Sergiy V., Borysov, Oleksandr V., Severina, Hanna I., Kovalenko, Sergiy M., Osolodchenko, Tetiana P., Vlasov, Vitaliy S., Georgiyants, Victoriya A.
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Published in Z͡h︡urnal orhanichnoï ta farmat͡s︡evtychnoï khimiï (20.10.2021)
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Straightforward Synthesis of Functionalized 4,5,6,7‐Tetrahydro‐pyrazolo[1,5‐a]pyrazines – Important Building Blocks for Medicinal Chemistry
Bozhanov, Vladimir I., Bohdan, Dmytro P., Borysov, Oleksandr V., Silin, Aleksey V., Zaremba, Oleg V., Avramenko, Mykola M., Volochnyuk, Dmitriy M., Ryabukhin, Sergey V., Gavrilenko, Konstantin S.
Published in ChemistrySelect (Weinheim) (07.06.2022)
Published in ChemistrySelect (Weinheim) (07.06.2022)
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