First-in-class multifunctional TYMS nonclassical antifolate inhibitor with potent in vivo activity that prolongs survival
Guijarro, Maria V, Kellish, Patrick C, Dib, Peter E, Paciaroni, Nicholas G, Nawab, Akbar, Andring, Jacob, Kulemina, Lidia, Borrero, Nicholas V, Modenutti, Carlos, Feely, Michael, Nasri, Elham, Seifert, Robert P, Luo, Xiaoping, Bennett, Richard L, Shabashvili, Daniil, Licht, Jonathan D, McKenna, Robert, Roitberg, Adrian, Huigens, 3rd, Robert W, Kaye, Frederic J, Zajac-Kaye, Maria
Published in JCI insight (22.05.2023)
Published in JCI insight (22.05.2023)
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Journal Article
Phenazine antibiotic inspired discovery of potent bromophenazine antibacterial agents against Staphylococcus aureus and Staphylococcus epidermidis
Borrero, Nicholas V., Bai, Fang, Perez, Cristian, Duong, Benjamin Q., Rocca, James R., Jin, Shouguang, Huigens, Robert W.
Published in Organic & biomolecular chemistry (14.02.2014)
Published in Organic & biomolecular chemistry (14.02.2014)
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Phenazine antibiotic inspired discovery of potent bromophenazine antibacterial agents against Staphylococcus aureus and Staphylococcus epidermidisElectronic supplementary information (ESI) available. See DOI: 10.1039/c3ob42416b
Borrero, Nicholas V, Bai, Fang, Perez, Cristian, Duong, Benjamin Q, Rocca, James R, Jin, Shouguang, Huigens III, Robert W
Year of Publication 14.01.2014
Year of Publication 14.01.2014
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Abstract 4055: First in class multifunctional non classical antifolates inhibits thymidylate synthase and extends survival in pancreatic cancer model
Guijarro, Maria V., Kellish, Patrick C., Dib, Peter E., Paciaroni, Nicholas G., Nawab, Akbar, Andring, Jacob, Kulemina, Lidia, Borrero, Nicholas V., Modenutti, Carlos, Bennett, Richard L., Shabashvili, Daniil, Licht, Jonathan D., McKenna, Robert, Roitberg, Adrian, Huigens, Robert W., Kaye, Frederic J., Zajac-Kaye, Maria
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Journal Article
Phenazine antibiotic inspired discovery of potent bromophenazine antibacterial agents against Staphylococcus aureusand Staphylococcus epidermidis
Borrero, Nicholas V, Bai, Fang, Perez, Cristian, Duong, Benjamin Q, Rocca, James R, Jin, Shouguang, Huigens, Robert W
Published in Organic & biomolecular chemistry (01.01.2014)
Published in Organic & biomolecular chemistry (01.01.2014)
Get full text
Journal Article