Eribulin Induces Irreversible Mitotic Blockade: Implications of Cell-Based Pharmacodynamics for In vivo Efficacy under Intermittent Dosing Conditions
TOWLE, Murray J, SALVATO, Kathleen A, LITTLEFIELD, Bruce A, WELS, Bruce F, AALFS, Kimberley K, WANJUN ZHENG, SELETSKY, Boris M, XIAOJIE ZHU, LEWIS, Bryan M, KISHI, Yoshito, YU, Melvin J
Published in Cancer research (Chicago, Ill.) (15.01.2011)
Published in Cancer research (Chicago, Ill.) (15.01.2011)
Get full text
Journal Article
Tubulin-based antimitotic mechanism of E7974, a novel analogue of the marine sponge natural product hemiasterlin
Kuznetsov, Galina, TenDyke, Karen, Towle, Murray J, Cheng, Hongsheng, Liu, Junke, Marsh, Joanne P, Schiller, Shawn E R, Spyvee, Mark R, Yang, Hu, Seletsky, Boris M, Shaffer, Christina J, Marceau, Veronique, Yao, Ye, Suh, Edward M, Campagna, Silvio, Fang, Francis G, Kowalczyk, James J, Littlefield, Bruce A
Published in Molecular cancer therapeutics (01.10.2009)
Published in Molecular cancer therapeutics (01.10.2009)
Get full text
Journal Article
Novel second generation analogs of eribulin. Part III: Blood–brain barrier permeability and in vivo activity in a brain tumor model
Narayan, Sridhar, Carlson, Eric M., Cheng, Hongsheng, Condon, Krista, Du, Hong, Eckley, Sean, Hu, Yongbo, Jiang, Yimin, Kumar, Vipul, Lewis, Bryan M., Saxton, Philip, Schuck, Edgar, Seletsky, Boris M., Tendyke, Karen, Zhang, Huiming, Zheng, Wanjun, Littlefield, Bruce A., Towle, Murray J., Yu, Melvin J.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Get full text
Journal Article
Novel second generation analogs of eribulin. Part I: Compounds containing a lipophilic C32 side chain overcome P-glycoprotein susceptibility
Narayan, Sridhar, Carlson, Eric M., Cheng, Hongsheng, Du, Hong, Hu, Yongbo, Jiang, Yimin, Lewis, Bryan M., Seletsky, Boris M., Tendyke, Karen, Zhang, Huiming, Zheng, Wanjun, Littlefield, Bruce A., Towle, Murray J., Yu, Melvin J.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Get full text
Journal Article
Discovery of CC-99677, a selective targeted covalent MAPKAPK2 (MK2) inhibitor for autoimmune disorders
Malona, JOHN, CHUAQUI, CLAUDIO, SELETSKY, BORIS M., BEEBE, LISA, CANTIN, SUSAN, KALKEN, DANIEL VAN, FAHNOE, KELLY, WANG, ZHIGANG, BROWNING, BETH, SZABO, HILARY, KOOPMAN, LOUISE A., ORAVECZ, TAMAS, MCDONALD, JOSEPH J., RAMIREZ-VALLE, FRANCISCO, GAUR, RAJULA, MENSAH, KOFI A., THOMAS, MICHAEL, CONNARN, JAMIE N., HU, HAIQING, ALEXANDER, MATTHEW D., CORIN, ALAN F.
Published in Translational research : the journal of laboratory and clinical medicine (01.11.2022)
Published in Translational research : the journal of laboratory and clinical medicine (01.11.2022)
Get full text
Journal Article
In vitro and in vivo anticancer activities of synthetic macrocyclic ketone analogues of halichondrin B
TOWLE, Murray J, SALVATO, Kathleen A, HABGOOD, Gregory J, SINGER, Lori A, DIPIETRO, Lucian V, YUAN WANG, CHEN, Jack J, QUINCY, David A, DAVIS, Ashley, YOSHIMATSU, Kentaro, KISHI, Yoshito, YU, Melvin J, BUDROW, Jacqueline, LITTLEFIELD, Bruce A, WELS, Bruce F, KUZNETSOV, Galina, AALFS, Kimberley K, WELSH, Susan, WANJUN ZHENG, SELETSKY, Boris M, PALME, Monica H
Published in Cancer research (Chicago, Ill.) (01.02.2001)
Get full text
Published in Cancer research (Chicago, Ill.) (01.02.2001)
Journal Article
Macrocyclic ketone analogues of halichondrin B
Zheng, Wanjun, Seletsky, Boris M., Palme, Monica H., Lydon, Paul J., Singer, Lori A., Chase, Charles E., Lemelin, Charles A., Shen, Yongchun, Davis, Heather, Tremblay, Lynda, Towle, Murray J., Salvato, Kathleen A., Wels, Bruce F., Aalfs, Kimberley K., Kishi, Yoshito, Littlefield, Bruce A., Yu, Melvin J.
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
Get full text
Journal Article
Novel second generation analogs of eribulin. Part II: Orally available and active against resistant tumors in vivo
Narayan, Sridhar, Carlson, Eric M., Cheng, Hongsheng, Condon, Krista, Du, Hong, Eckley, Sean, Hu, Yongbo, Jiang, Yimin, Kumar, Vipul, Lewis, Bryan M., Saxton, Philip, Schuck, Edgar, Seletsky, Boris M., Tendyke, Karen, Zhang, Huiming, Zheng, Wanjun, Littlefield, Bruce A., Towle, Murray J., Yu, Melvin J.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Get full text
Journal Article
Structurally simplified macrolactone analogues of halichondrin B
Seletsky, Boris M., Wang, Yuan, Hawkins, Lynn D., Palme, Monica H., Habgood, Gregory J., DiPietro, Lucian V., Towle, Murray J., Salvato, Kathleen A., Wels, Bruce F., Aalfs, Kimberley K., Kishi, Yoshito, Littlefield, Bruce A., Yu, Melvin J.
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
Published in Bioorganic & medicinal chemistry letters (15.11.2004)
Get full text
Journal Article
Highly syn-Selective Additions of Allylic Stannanes to Protected .alpha.-Amino Aldehydes
Marshall, James A, Seletsky, Boris M, Coan, Paul S
Published in Journal of organic chemistry (01.09.1994)
Published in Journal of organic chemistry (01.09.1994)
Get full text
Journal Article
Abstract 4493: Eribulin recognizes the nucleotide states of soluble tubulin and binds with high-affinity on a site distinct from known tubulin inhibitors
Agarwala, Kishan Lal, Kubara, Kenji, Sagane, Koji, Seletsky, Boris M., Littlefield, Bruce A.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Get full text
Journal Article
HETEROCYCLIC PAD4 INHIBITORS
SELETSKY, Boris M, ROSS, Audrey Graham, GORMISKY, Paul E, MIAO, Guobin, ZHU, Xiao, ANTROPOW, Alyssa H
Year of Publication 30.11.2023
Get full text
Year of Publication 30.11.2023
Patent
HETEROCYCLIC PAD4 INHIBITORS
Selvakumar, Kumaravel, Agarwal, Piyush, Gormisky, Paul E, Paidi, Venkatram, Tino, Joseph A, Zhu, Xiao, Gardner, Daniel S, Cherney, Robert J, Thangathirupathy, Srinivasan, Alajangi, Tirupathi Rao, Duncia, John V, Mahadevu, Krishna, Zhu, Zhengdong, Miao, Guobin, Sura, Mallikarjun Reddy, Seletsky, Boris M, Sistla, Ramesh Kumar, Dhar, T. G. Murali, Morampudi, Ooha, Antropow, Alyssa H, Panda, Manoranjan, Nair, Jalathi S, Ross, Audrey Graham, Subbiah Karuppiah, Arul Mozhi, Cuervo, Julio Herman, Kumar Cm, Vijaya, Niu, Deqiang
Year of Publication 01.06.2023
Get full text
Year of Publication 01.06.2023
Patent
HETEROCYCLIC PAD4 INHIBITORS
SISTLA, Ramesh, Kumar, MAHADEVU, Krishna, CUERVO, Julio, Hernán, ZHU, Zhengdong, SUBBIAH KARUPPIAH, Arul, Mozhi, GORMISKY, Paul, E, AGARWAL, Piyush, ALAJANGI, Tirupathi, Rao, CHERNEY, Robert, J, NIU, Deqiang, GARDNER, Daniel, S, NAIR, Jalathi, S, DHAR, T., G., Murali, KUMAR CM, Vijaya, MORAMPUDI, Ooha, TINO, Joseph, A, ROSS, Audrey, Graham, ZHU, Xiao, SELETSKY, Boris, M, SURA, Mallikarjun, Reddy, SELVAKUMAR, Kumaravel, DUNCIA, John, V, PANDA, Manoranjan, PAIDI, Venkatram Reddy, MIAO, Guobin, THANGATHIRUPATHY, Srinivasan, ANTROPOW, Alyssa, H
Year of Publication 21.12.2022
Get full text
Year of Publication 21.12.2022
Patent
Heterocyclic PAD4 inhibitors
SELETSKY, Boris M, DHAR, T. G. Murali, MAHADEVU, Krishna, SURA, Mallikarjun, ZHU, Zhengdong, AGARWAL, Piyush, SUBBIAH KARUPPIAH, Arul Mozhi, NIU, Deqiang, ALAJANGI, Tirupathi, TINO, Joseph A, GORMISKY, Paul E, NAIR, Jalathi, CUERVO, Julio Hernán, KUMAR CM, Vijaya, MORAMPUDI, Ooha, ZHU, Xiao, ANTROPOW, Alyssa H, SELVAKUMAR, Kumaravel, PANDA, Manoranjan, ROSS, Audrey Graham, PAIDI, Venkatram Reddy, CHERNEY, Robert J, DUNCIA, John V, SISTLA, Ramesh, MIAO, Guobin, GARDNER, Daniel S, THANGATHIRUPATHY, Srinivasan
Year of Publication 06.10.2022
Get full text
Year of Publication 06.10.2022
Patent