Clustering of Tadalafil API Samples According to their Manufacturer in the Context of API Falsification Detection
Deconinck, E., Raimondo, M., Borioni, A., Grange, Y., Rebière, H., Mihailova, A., Bøyum, O., Maurin, J.K., Pioruńska-Sędłak, K., Olsen, L. Stengelshøj, Acevska, J., Brezovska, K., Rundlöf, T., Portela, M.J., Meieranz, S., Miquel, M., Bertrand, M.
Published in Journal of pharmaceutical sciences (01.11.2023)
Published in Journal of pharmaceutical sciences (01.11.2023)
Get full text
Journal Article
Behavioral and electrophysiological effects of the adenosine A2A receptor antagonist SCH 58261 in R6/2 Huntington’s disease mice
Domenici, M.R, Scattoni, M.L, Martire, A, Lastoria, G, Potenza, R.L, Borioni, A, Venerosi, A, Calamandrei, G, Popoli, P
Published in Neurobiology of disease (01.11.2007)
Published in Neurobiology of disease (01.11.2007)
Get full text
Journal Article
A new synthetic approach of N-(4-amino-2-methylquinolin-6-yl)-2-(4-ethylphenoxymethyl)benzamide (JTC-801) and its analogues and their pharmacological evaluation as nociceptin receptor (NOP) antagonists
Sestili, Isabella, Borioni, Anna, Mustazza, Carlo, Rodomonte, Andrea, Turchetto, Luciana, Sbraccia, Maria, Riitano, Daniela, Del Giudice, Maria Rosaria
Published in European journal of medicinal chemistry (01.12.2004)
Published in European journal of medicinal chemistry (01.12.2004)
Get full text
Journal Article
Synthesis of imidazo[1,2-c]pyrazolo[4,3-e]pyrimidines, pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines and 1,2,4-triazolo[5,1-i]purines: new potent adenosine A2 receptor antagonists
GATTA, F, DEL GIUDICE, M. R, BORIONI, A, BOREA, P. A, DIONISOTTI, S, ONGINI, E
Published in European journal of medicinal chemistry (1993)
Published in European journal of medicinal chemistry (1993)
Get full text
Journal Article
(E)-1-(Heterocyclyl or cyclohexyl)-2-[1,3,7-trisubstituted (xanthin-8-yl)] ethenes as A2a adenosine receptor antagonists
DEL GIUDICE, M. R, BORIONI, A, MUSTAZZA, C, GATTA, F, DIONISOTTI, S, ZOCCHI, C, ONGINI, E
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
Get full text
Journal Article
Synthesis and Pharmacological Evaluation of 1,2-Dihydrospiro[isoquinoline-4(3H),4′-piperidin]-3-ones as Nociceptin Receptor Agonists
Mustazza, Carlo, Borioni, Anna, Sestili, Isabella, Sbraccia, Maria, Rodomonte, Andrea, Del Giudice, Maria Rosaria
Published in Journal of medicinal chemistry (28.02.2008)
Published in Journal of medicinal chemistry (28.02.2008)
Get full text
Journal Article
Synthesis and Evaluation as NOP Ligands of Some Spiro[piperidine-4,2′(1′H)-quinazolin]-4′(3′H)-ones and Spiro[piperidine-4,5′(6′H)-[1,2,4]triazolo[1,5-c]quinazolines]
Mustazza, Carlo, Borioni, Anna, Sestili, Isabella, Sbraccia, Maria, Rodomonte, Andrea, Ferretti, Rosella, Giudice, Maria Rosaria Del
Published in Chemical & Pharmaceutical Bulletin (2006)
Published in Chemical & Pharmaceutical Bulletin (2006)
Get full text
Journal Article
Behavioral and electrophysiological effects of the adenosine A 2A receptor antagonist SCH 58261 in R6/2 Huntington’s disease mice
Domenici, M.R., Scattoni, M.L., Martire, A., Lastoria, G., Potenza, R.L., Borioni, A., Venerosi, A., Calamandrei, G., Popoli, P.
Published in Neurobiology of disease (2007)
Published in Neurobiology of disease (2007)
Get full text
Journal Article
High resolution NMR conformational studies of new bivalent NOP receptor antagonists in model membrane systems
Borioni, Anna, Bastanzio, Giuditta, Delfini, Maurizio, Mustazza, Carlo, Sciubba, Fabio, Tatti, Massimo, Giudice, Maria Rosaria Del
Published in Bioorganic chemistry (01.02.2011)
Published in Bioorganic chemistry (01.02.2011)
Get full text
Journal Article
Synthesis and cholinesterase activity of phenylcarbamates related to Rivastigmine, a therapeutic agent for Alzheimer's disease
Mustazza, Carlo, Borioni, Anna, Giudice, Maria Rosaria Del, Gatta, Franco, Ferretti, Rosella, Meneguz, Annarita, Volpe, Maria Teresa, Lorenzini, Paola
Published in European journal of medicinal chemistry (01.02.2002)
Published in European journal of medicinal chemistry (01.02.2002)
Get full text
Journal Article
(E)-1-(heterocyclyl or cyclohexyl)-2-[1,3,7-trisubstituted(xantkin-8-yl)] ethenes as A(2a) adenosine receptor antagonists
DelGiudice, MR, Borioni, A, Mustazza, C, Gatta, F, Dionisotti, S, Zocchi, C, Ongini, E
Published in European journal of medicinal chemistry (01.01.1996)
Published in European journal of medicinal chemistry (01.01.1996)
Get full text
Journal Article
Synthesis of 1-Methyl-5-(pyrazol-3- and -5-yl- and 1, 2, 4-triazol-3- and 5-yl)-1, 2, 3, 6-tetrahydropyridine Derivatives and Their Evaluation as Muscarinic Receptor Ligands
Del Giudice, Maria Rosaria, Mustazza, Carlo, Borioni, Anna, Gatta, Franco, Tayebati, Khosrow, Amenta, Francesco, Tucci, Paolo, Pieretti, Stefano
Published in Archiv der Pharmazie (Weinheim) (01.06.2003)
Published in Archiv der Pharmazie (Weinheim) (01.06.2003)
Get full text
Journal Article
( E)-1-(Heterocyclyl or cyclohexyl)-2-[1,3,7-trisubstituted (xanthin-8-yl)] ethenes as A 2a adenosine receptor antagonists
Del Giudice, MR, Borioni, A, Mustazza, C, Gatta, F, Dionisotti, S, Zocchi, C, Ongini, E
Published in European journal of medicinal chemistry (1996)
Published in European journal of medicinal chemistry (1996)
Get full text
Journal Article
NEW[G]-FUSED [1,2,4]TRIAZOLO[1,5-C]PYRIMIDINES - SYNTHESIS OF PYRIDO[3,2-E] AND [4,3-E][1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE, PYRIMIDO[5,4-E][1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE AND [1,2,4]TRIAZOLO[1,5-C]PTERIDINE DERIVATIVES
DELGIUDICE, MR, BORIONI, A, MUSTAZZA, C, GATTA, F
Published in Journal of heterocyclic chemistry (01.11.1994)
Published in Journal of heterocyclic chemistry (01.11.1994)
Get more information
Journal Article
Synthesis of pyrido[2,1-b]- and thiazolo[2,3-b]purines
DelGiudice, MR, Borioni, A, Mustazza, C, Gatta, F
Published in Journal of heterocyclic chemistry (01.11.1995)
Published in Journal of heterocyclic chemistry (01.11.1995)
Get more information
Journal Article