Discovery of Potent Indolyl-Hydrazones as Kinase Inhibitors for Breast Cancer: Synthesis, X-ray Single-Crystal Analysis, and In Vitro and In Vivo Anti-Cancer Activity Evaluation
Salama, Eid E, Youssef, Mohamed F, Aboelmagd, Ahmed, Boraei, Ahmed T A, Nafie, Mohamed S, Haukka, Matti, Barakat, Assem, Sarhan, Ahmed A M
Published in Pharmaceuticals (Basel, Switzerland) (01.12.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.12.2023)
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Synthesis and X-ray Crystal Structure Analysis of Substituted 1,2,4-Triazolo [4’,3’:2,3]pyridazino[4,5-b]indole and Its Precursor
Boraei, Ahmed T. A., Eltamany, Elsayed H., Haukka, Matti, Soliman, Saied M., Barakat, Assem, Sopaih, Manar
Published in Crystals (Basel) (01.07.2023)
Published in Crystals (Basel) (01.07.2023)
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4-Methyl/Phenyl-1,2,5,6-tetraazafluoranthen-3(2H)-ones Synthesis: Mechanistic Pathway Study and Single-Crystal X-ray Analysis of the Intermediates
Sarhan, Ahmed A. M., Haukka, Matti, Barakat, Assem, Soliman, Saied M., Boraei, Ahmed T. A., Sopaih, Manar, Salama, Eid E.
Published in Crystals (Basel) (01.11.2023)
Published in Crystals (Basel) (01.11.2023)
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Journal Article
Synthesis of a Novel Hydrazone of Thieno[2,3-d]pyrimidine Clubbed with Ninhydrin: X-ray Crystal Structure and Computational Investigations
Altowyan, Mezna Saleh, Haukka, Matti, Soliman, Saied M., Barakat, Assem, Boraei, Ahmed T. A., Sopaih, Manar
Published in Crystals (Basel) (01.03.2023)
Published in Crystals (Basel) (01.03.2023)
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Journal Article
Synthesis, Characterization and Single Crystal X-ray Diffraction Analysis of Fused Triazolo/Thiadiazole Clubbed with Indole Scaffold
Altowyan, Mezna Saleh, Haukka, Matti, Soliman, Saied M., Barakat, Assem, Alaswad, Saleh O., Boraei, Ahmed T. A., Gad, Emad M., Youssef, Mohamed F.
Published in Crystals (Basel) (01.03.2023)
Published in Crystals (Basel) (01.03.2023)
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Journal Article
Base-Controlled Regiospecific Mono-Benzylation/Allylation and Diallylation of 4-Aryl-5-indolyl-1,2,4-triazole-3-thione: Thio-Aza Allyl Rearrangement
Salama, Eid E, Youssef, Mohamed F, Boraei, Ahmed T. A, Haukka, Matti, Soliman, Saied M, Barakat, Assem, Sarhan, Ahmed A. M
Published in Crystals (Basel) (01.06.2023)
Published in Crystals (Basel) (01.06.2023)
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Journal Article
Discovery of New Apoptosis-Inducing Agents for Breast Cancer Based on Ethyl 2-Amino-4,5,6,7-Tetra Hydrobenzo[ b ]Thiophene-3-Carboxylate: Synthesis, In Vitro, and In Vivo Activity Evaluation
Gad, Emad M, Nafie, Mohamed S, Eltamany, Elsayed H, Hammad, Magdy S A G, Barakat, Assem, Boraei, Ahmed T A
Published in Molecules (Basel, Switzerland) (28.05.2020)
Published in Molecules (Basel, Switzerland) (28.05.2020)
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Journal Article
Stereoselective Synthesis of New 4-Aryl-5-indolyl-1,2,4-triazole S- and N-β-Galactosides: Characterizations, X-ray Crystal Structure and Hirshfeld Surface Analysis
Altowyan, Mezna Saleh, Haukka, Matti, Soliman, Saied M., Barakat, Assem, Boraei, Ahmed T. A., Aboelmagd, Ahmed
Published in Crystals (Basel) (10.05.2023)
Published in Crystals (Basel) (10.05.2023)
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Journal Article
Synthesis, X-ray Single-Crystal Analysis, and Anticancer Activity Evaluation of New Alkylsulfanyl-Pyridazino[4,5-b]indole Compounds as Multitarget Inhibitors of EGFR and Its Downstream PI3K-AKT Pathway
Salama, Eid E., Althobaiti, Ibrahim O., Haukka, Matti, Boraei, Ahmed T. A.
Published in Crystals (Basel) (01.03.2022)
Published in Crystals (Basel) (01.03.2022)
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Journal Article
Intramolecular Hydrogen Bond, Hirshfeld Analysis, AIM; DFT Studies of Pyran-2,4-dione Derivatives
Boraei, Ahmed T. A., Haukka, Matti, Sarhan, Ahmed A. M., Soliman, Saied M., Barakat, Assem
Published in Crystals (Basel) (01.08.2021)
Published in Crystals (Basel) (01.08.2021)
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Journal Article
Synthesis of New Functionalized Indoles Based on Ethyl Indol-2-carboxylate
Boraei, Ahmed T A, El Ashry, El Sayed H, Barakat, Assem, Ghabbour, Hazem A
Published in Molecules (Basel, Switzerland) (10.03.2016)
Published in Molecules (Basel, Switzerland) (10.03.2016)
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Journal Article
Design and Synthesis of Novel Pyridine-Based Compounds as Potential PIM‑1 Kinase Inhibitors, Apoptosis, and Autophagy Inducers Targeting MCF‑7 Cell Lines: In Vitro and In Vivo Studies
Shaban, Shrouk M., Eltamany, Elsayed H., Boraei, Ahmed T. A., Nafie, Mohamed S., Gad, Emad M.
Published in ACS omega (12.12.2023)
Published in ACS omega (12.12.2023)
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Journal Article
X-ray Single Crystal Structure, Tautomerism Aspect, DFT, NBO, and Hirshfeld Surface Analysis of a New Schiff Bases Based on 4-Amino-5-Indol-2-yl-1,2,4-Triazole-3-Thione Hybrid
Boraei, Ahmed, Soliman, Saied, Haukka, Matti, El Tamany, El, Al-Majid, Abdullah, Barakat, Assem
Published in Crystals (Basel) (01.09.2021)
Published in Crystals (Basel) (01.09.2021)
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Journal Article
Straightforward One-Pot Synthesis of New 4-Phenyl-1,2,5,6-tetraazafluoranthen-3(2H)-one Derivatives: X-ray Single Crystal Structure and Hirshfeld Analyses
Boraei, Ahmed T. A., Haukka, Matti, Sopaih, Manar, Al-Majid, Abdullah Mohammed, Soliman, Saied M., Barakat, Assem, Sarhan, Ahmed A. M.
Published in Crystals (Basel) (01.02.2022)
Published in Crystals (Basel) (01.02.2022)
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Journal Article
Synthesis of C2-Symmetrical Bis-(β-Enamino-Pyran-2,4-dione) Derivative Linked via 1,6-Hexylene Spacer: X-ray Crystal Structures, Hishfeld Studies and DFT Calculations of Mono- and Bis-(Pyran-2,4-diones) Derivatives
Boraei, Ahmed T. A., Haukka, Matti, Sarhan, Ahmed A. M., Soliman, Saied M., Al-Majid, Abdullah Mohammed, Barakat, Assem
Published in Symmetry (Basel) (01.09.2021)
Published in Symmetry (Basel) (01.09.2021)
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