Recent Advances on Small-Molecule Antagonists Targeting TLR7
Zheng, Haoyang, Wu, Peiyang, Bonnet, Pierre-Antoine
Published in Molecules (Basel, Switzerland) (07.01.2023)
Published in Molecules (Basel, Switzerland) (07.01.2023)
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Agonist and antagonist ligands of toll-like receptors 7 and 8: Ingenious tools for therapeutic purposes
Patinote, Cindy, Karroum, Nour Bou, Moarbess, Georges, Cirnat, Natalina, Kassab, Issam, Bonnet, Pierre-Antoine, Deleuze-Masquéfa, Carine
Published in European journal of medicinal chemistry (01.05.2020)
Published in European journal of medicinal chemistry (01.05.2020)
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Journal Article
Anticoagulant Activity of Sulfated Ulvan Isolated from the Green Macroalga Ulva rigida
Adrien, Amandine, Bonnet, Antoine, Dufour, Delphine, Baudouin, Stanislas, Maugard, Thierry, Bridiau, Nicolas
Published in Marine drugs (14.05.2019)
Published in Marine drugs (14.05.2019)
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[1,2,4]triazolo[4,3- a ]quinoxaline as Novel Scaffold in the Imiqualines Family: Candidates with Cytotoxic Activities on Melanoma Cell Lines
Patinote, Cindy, Raevens, Sandy, Baumann, Amélie, Pellegrin, Eloise, Bonnet, Pierre-Antoine, Deleuze-Masquéfa, Carine
Published in Molecules (Basel, Switzerland) (18.07.2023)
Published in Molecules (Basel, Switzerland) (18.07.2023)
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Bixin, an apocarotenoid isolated from Bixa orellana L., sensitizes human melanoma cells to dacarbazine-induced apoptosis through ROS-mediated cytotoxicity
de Oliveira Júnior, Raimundo Gonçalves, Bonnet, Antoine, Braconnier, Estelle, Groult, Hugo, Prunier, Grégoire, Beaugeard, Laureen, Grougnet, Raphäel, da Silva Almeida, Jackson Roberto Guedes, Ferraz, Christiane Adrielly Alves, Picot, Laurent
Published in Food and chemical toxicology (01.03.2019)
Published in Food and chemical toxicology (01.03.2019)
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Imidazoquinoxaline derivative EAPB0503: A promising drug targeting mutant nucleophosmin 1 in acute myeloid leukemia
Nabbouh, Ali I., Hleihel, Rita S., Saliba, Jessica L., Karam, Martin M., Hamie, Maguy H., Wu, Hsin‐Chieh J. M., Berthier, Caroline P., Tawil, Nadim M., Bonnet, Pierre‐Antoine A., Deleuze‐Masquefa, Carine, El Hajj, Hiba A.
Published in Cancer (01.05.2017)
Published in Cancer (01.05.2017)
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EAPB0503, an Imidazoquinoxaline Derivative Modulates SENP3/ARF Mediated SUMOylation, and Induces NPM1c Degradation in NPM1 Mutant AML
Skayneh, Hala, Jishi, Batoul, Hleihel, Rita, Hamie, Maguy, El Hajj, Rana, Deleuze-Masquefa, Carine, Bonnet, Pierre-Antoine, El Sabban, Marwan, El Hajj, Hiba
Published in International journal of molecular sciences (22.03.2022)
Published in International journal of molecular sciences (22.03.2022)
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EAPB0503: An Imiquimod analog with potent in vitro activity against cutaneous leishmaniasis caused by Leishmania major and Leishmania tropica
El Hajj, Rana, Bou Youness, Hanady, Lachaud, Laurence, Bastien, Patrick, Masquefa, Carine, Bonnet, Pierre-Antoine, El Hajj, Hiba, Khalifeh, Ibrahim
Published in PLoS neglected tropical diseases (01.11.2018)
Published in PLoS neglected tropical diseases (01.11.2018)
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Journal Article
A novel route for the synthesis of androgen receptor antagonist enzalutamide
Meng, Xiangguo, Bi, Siju, Jin, Shixin, Wu, Kai, Wu, Shanchao, Shao, Lei, Bonnet, Pierre-Antoine, Sheng, Chunquan
Published in Chinese chemical letters (01.06.2023)
Published in Chinese chemical letters (01.06.2023)
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Journal Article
Imiquimod Targets Toxoplasmosis Through Modulating Host Toll-Like Receptor-MyD88 Signaling
Hamie, Maguy, Najm, Rania, Deleuze-Masquefa, Carine, Bonnet, Pierre Antoine, Dubremetz, Jean-François, El Sabban, Marwan, El Hajj, Hiba
Published in Frontiers in immunology (09.03.2021)
Published in Frontiers in immunology (09.03.2021)
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HMOX1 and NQO1 Genes are Upregulated in Response to Contact Sensitizers in Dendritic Cells and THP-1 Cell Line: Role of the Keap1/Nrf2 Pathway
Ade, Nadège, Leon, Fanny, Pallardy, Marc, Peiffer, Jean-Luc, Kerdine-Romer, Saadia, Tissier, Marie-Hélène, Bonnet, Pierre-Antoine, Fabre, Isabelle, Ourlin, Jean-Claude
Published in Toxicological sciences (01.02.2009)
Published in Toxicological sciences (01.02.2009)
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Substantial Cellular Penetration of Fluorescent Imidazoquinoxalines
Patinote, Cindy, Cirnat, Natalina, Hadj-Kaddour, Kamel, Cuq, Pierre, Bonnet, Pierre-Antoine, Deleuze-Masquéfa, Carine
Published in Journal of fluorescence (01.12.2020)
Published in Journal of fluorescence (01.12.2020)
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Journal Article
Identification of ace inhibitory cryptides in Tilapia protein hydrolysate by UPLC–MS/MS coupled to database analysis
Yesmine, Ben Henda, Antoine, Bonnet, da Silva Ortência Leocádia, Nunes Gonzalez, Rogério, Boscolo Wilson, Ingrid, Arnaudin, Nicolas, Bridiau, Thierry, Maugard, Jean-Marie, Piot, Frédéric, Sannier, Stéphanie, Bordenave-Juchereau
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.05.2017)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.05.2017)
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Post-treatment positron emission tomography-computed tomography is highly predictive of outcome in Plasmablastic lymphoma
Al Tabaa, Yassine, Tchernonog, Emmanuelle, Faurie, Pierre, Cottereau, Anne Ségolène, Monjanel, Hélène, Bonnet, Antoine, Le Gouill, Steven, Gyan, Emmanuel, Ghesquieres, Hervé, Mariano-Goulart, Denis, Cartron, Guillaume
Published in European journal of nuclear medicine and molecular imaging (01.09.2018)
Published in European journal of nuclear medicine and molecular imaging (01.09.2018)
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Journal Article
FLT3 ligand plasma levels in acute myeloid leukemia
Peterlin, Pierre, Gaschet, Joelle, Guillaume, Thierry, Garnier, Alice, Eveillard, Marion, Le Bourgeois, Amandine, Cherel, Michel, Debord, Camille, Le Bris, Yannick, Theisen, Olivier, Mahé, Béatrice, Dubruille, Viviane, Godon, Catherine, Robillard, Nelly, Wuilleme, Soraya, Touzeau, Cyrille, Gastinne, Thomas, Blin, Nicolas, Lok, Anne, Bonnet, Antoine, Le Gouill, Steven, Moreau, Philippe, Béné, Marie-C, Chevallier, Patrice
Published in Haematologica (Roma) (01.06.2019)
Published in Haematologica (Roma) (01.06.2019)
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Synthesis of 2-Mercapto-(2-Oxoindolin-3-Ylidene)Acetonitriles from 3-(4-Chloro-5 H -1,2,3-Dithiazol-5-Ylidene)Indolin-2-ones
Letribot, Boris, Delatouche, Régis, Rouillard, Hervé, Bonnet, Antoine, Chérouvrier, Jean-René, Domon, Lisianne, Besson, Thierry, Thiéry, Valérie
Published in Molecules (Basel, Switzerland) (08.06.2018)
Published in Molecules (Basel, Switzerland) (08.06.2018)
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UPLC-MSE profiling of Phytoplankton metabolites: application to the identification of pigments and structural analysis of metabolites in Porphyridium purpureum
Juin, Camille, Bonnet, Antoine, Nicolau, Elodie, Bérard, Jean-Baptiste, Devillers, Romain, Thiéry, Valérie, Cadoret, Jean-Paul, Picot, Laurent
Published in Marine drugs (22.04.2015)
Published in Marine drugs (22.04.2015)
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