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Published in Journal of medicinal chemistry (24.02.2005)
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Discovery and Clinical Evaluation of 1-{N-[2-(Amidinoaminooxy)ethyl]amino}carbonylmethyl-6-methyl-3-[2,2-difluoro-2-phenylethylamino]pyrazinone (RWJ-671818), a Thrombin Inhibitor with an Oxyguanidine P1 Motif
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Published in Journal of medicinal chemistry (25.02.2010)
Published in Journal of medicinal chemistry (25.02.2010)
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Design and synthesis of polyethylene glycol-modified biphenylsulfonyl-thiophene-carboxamidine inhibitors of the complement component C1s
Subasinghe, Nalin L., Khalil, Ehab, Travins, Jeremy M., Ali, Farah, Ballentine, Shelley K., Hufnagel, Heather R., Pan, Wenxi, Leonard, Kristi, Bone, Roger F., Soll, Richard M., Crysler, Carl S., Ninan, Nisha, Kirkpatrick, Jennifer, Kolpak, Michael X., Diloreto, Karen A., Eisennagel, Stephen H., Huebert, Norman D., Molloy, Christopher J., Tomczuk, Bruce E., Gaul, Michael D.
Published in Bioorganic & medicinal chemistry letters (15.08.2012)
Published in Bioorganic & medicinal chemistry letters (15.08.2012)
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Corrections to Discovery and Clinical Evaluation of 1-{N-[2-(Amidinoaminooxy)ethyl]amino}carbonylmethyl-6-methyl-3-[2,2-difluoro-2-phenylethylamino]pyrazinone (RWJ-671818), a Thrombin Inhibitor with an Oxyguanidine P1 Motif
Lu, Tianbao, Markotan, Thomas, Ballentine, Shelley K, Giardino, Edward C, Spurlino, John, Brown, Kathryn, Maryanoff, Bruce E, Tomczuk, Bruce E, Damiano, Bruce P, Shukla, Umesh, End, David, Andrade-Gordon, Patricia, Bone, Roger F, Player, Mark R
Published in Journal of medicinal chemistry (22.04.2010)
Published in Journal of medicinal chemistry (22.04.2010)
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Biphenylsulfonyl-thiophene-carboxamidine inhibitors of the complement component C1s
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Published in Bioorganic & medicinal chemistry (01.03.2008)
Published in Bioorganic & medicinal chemistry (01.03.2008)
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A novel series of arylsulfonylthiophene-2-carboxamidine inhibitors of the complement component C1s
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Published in Bioorganic & medicinal chemistry letters (15.04.2006)
Published in Bioorganic & medicinal chemistry letters (15.04.2006)
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A novel series of potent and selective small molecule inhibitors of the complement component C1s
Subasinghe, Nalin L., Ali, Farah, Illig, Carl R., Jonathan Rudolph, M., Klein, Scott, Khalil, Ehab, Soll, Richard M., Bone, Roger F., Spurlino, John C., DesJarlais, Renee L., Crysler, Carl S., Cummings, Maxwell D., Morris, Philip E., Kilpatrick, John M., Sudhakara Babu, Y.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)
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Amino acid transport in suspension-cultured plant cells. III. Common carrier system for the uptake of L-arginine, L-aspartic acid, L-histidine, L-leucine, and L-phenylalanine
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Published in Plant physiology (Bethesda) (1982)
Published in Plant physiology (Bethesda) (1982)
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CRYSTAL STRUCTURE OF THE PRO FORM OF A MATRIX METALLOPROTEINASE AND AN ALLOSTERIC PROCESSING INHIBITOR
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Year of Publication 26.07.2017
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METHOD FOR THE IDENTIFICATION OF LIGANDS
ASKARI, HOSSEIN, SPRINGER, BARRY, A, RENTZEPERIS, DIONISIOS, BONE, ROGER, F
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Methods of treatment using allosteric processing inhibitors for matrix metalloproteinases
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Year of Publication 11.11.2014
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Year of Publication 11.11.2014
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