Discovery and Development of Small-Molecule Inhibitors of Glycogen Synthase
Tang, Buyun, Frasinyuk, Mykhaylo S, Chikwana, Vimbai M, Mahalingan, Krishna K, Morgan, Cynthia A, Segvich, Dyann M, Bondarenko, Svitlana P, Mrug, Galyna P, Wyrebek, Przemyslaw, Watt, David S, DePaoli-Roach, Anna A, Roach, Peter J, Hurley, Thomas D
Published in Journal of medicinal chemistry (09.04.2020)
Published in Journal of medicinal chemistry (09.04.2020)
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Journal Article
Aurones: Synthesis and Properties
Popova, Antonina V., Bondarenko, Svitlana P., Frasinyuk, Mykhaylo S.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.05.2019)
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.05.2019)
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Journal Article
Trapping of thermally generated ortho - and para -quinone methides by imidazoles and pyrazoles: a simple route to green synthesis of benzopyrone-azole hybrids and their evaluation as α-glucosidase inhibitors
Myshko, Andrii S., Mrug, Galyna P., Bondarenko, Svitlana P., Kondratyuk, Kostyantyn M., Kobzar, Oleksandr L., Buldenko, Vladyslav M., Kozytskiy, Andriy V., Vovk, Andriy I., Frasinyuk, Mykhaylo S.
Published in RSC advances (29.08.2024)
Published in RSC advances (29.08.2024)
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Journal Article
Developing antineoplastic agents that target peroxisomal enzymes: cytisine-linked isoflavonoids as inhibitors of hydroxysteroid 17-beta-dehydrogenase-4 (HSD17B4)
Frasinyuk, Mykhaylo S., Zhang, Wen, Wyrebek, Przemyslaw, Yu, Tianxin, Xu, Xuehe, Sviripa, Vitaliy M., Bondarenko, Svitlana P., Xie, Yanqi, Ngo, Huy X., Morris, Andrew J., Mohler, James L., Fiandalo, Michael V., Watt, David S., Liu, Chunming
Published in Organic & biomolecular chemistry (20.09.2017)
Published in Organic & biomolecular chemistry (20.09.2017)
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Journal Article
Coumarin-based homoisoflavonoids as precursors in the synthesis of 8-heteroarylmethylcoumarins
Myshko, Nataliia V., Mrug, Galyna P., Kondratyuk, Kostyantyn M., Bondarenko, Svitlana P., Frasinyuk, Mykhaylo S.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.07.2023)
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.07.2023)
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Journal Article
Carboxylated chalcones and related flavonoids as inhibitors of xanthine oxidase
Kobzar, Oleksandr L., Tatarchuk, Alona V., Mrug, Galyna P., Bondarenko, Svitlana P., Demydchuk, Bohdan A., Frasinyuk, Mykhaylo S., Vovk, Andriy I.
Published in Medicinal chemistry research (01.08.2023)
Published in Medicinal chemistry research (01.08.2023)
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Journal Article
Observations from aminomethylation of 7-substituted 6-hydroxyaurones
Bondarenko, Svitlana P., Frasinyuk, Mykhaylo S.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.08.2018)
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.08.2018)
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Journal Article
Semisynthetic aurones inhibit tubulin polymerization at the colchicine-binding site and repress PC-3 tumor xenografts in nude mice and myc-induced T-ALL in zebrafish
Xie, Yanqi, Kril, Liliia M, Yu, Tianxin, Zhang, Wen, Frasinyuk, Mykhaylo S, Bondarenko, Svitlana P, Kondratyuk, Kostyantyn M, Hausman, Elizabeth, Martin, Zachary M, Wyrebek, Przemyslaw P, Liu, Xifu, Deaciuc, Agripina, Dwoskin, Linda P, Chen, Jing, Zhu, Haining, Zhan, Chang-Guo, Sviripa, Vitaliy M, Blackburn, Jessica, Watt, David S, Liu, Chunming
Published in Scientific reports (23.04.2019)
Published in Scientific reports (23.04.2019)
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Journal Article
Chemoselective synthesis of 3-trifluoromethylpyrazole-deoxybenzoin hybrids
Biletska, Iryna M., Mrug, Galyna P., Bondarenko, Svitlana P., Kondratyuk, Kostyantyn M., Prostota, Yaroslav O., Sviripa, Vitaliy M., Frasinyuk, Mykhaylo S.
Published in Journal of fluorine chemistry (01.02.2021)
Published in Journal of fluorine chemistry (01.02.2021)
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Journal Article
A Direct Synthesis of 2‐(ω‐Carboxyalkyl)isoflavones from ortho‐Hydroxylated Deoxybenzoins
Mrug, Galyna P., Demydchuk, Bohdan A., Bondarenko, Svitlana P., Sviripa, Vitaliy M., Wyrebek, Przemyslaw, Mohler, James L., Fiandalo, Michael V., Liu, Chunming, Frasinyuk, Mykhaylo S., Watt, David S.
Published in European journal of organic chemistry (24.10.2018)
Published in European journal of organic chemistry (24.10.2018)
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Journal Article
Synthesis and tautomerization of hydroxylated isoflavones bearing heterocyclic hemi-aminals
Frasinyuk, Mykhaylo S., Bondarenko, Svitlana P., Khilya, Volodymyr P., Liu, Chunming, Watt, David S., Sviripa, Vitaliy M.
Published in Organic & biomolecular chemistry (28.01.2015)
Published in Organic & biomolecular chemistry (28.01.2015)
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Journal Article
Application of Mannich bases to the synthesis of hydroxymethylated isoflavonoids as potential antineoplastic agents
Frasinyuk, Mykhaylo S., Mrug, Galyna P., Bondarenko, Svitlana P., Sviripa, Vitaliy M., Zhang, Wen, Cai, Xianfeng, Fiandalo, Michael V., Mohler, James L., Liu, Chunming, Watt, David S.
Published in Organic & biomolecular chemistry (14.12.2015)
Published in Organic & biomolecular chemistry (14.12.2015)
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Journal Article
Chemoselective aminomethylation of harmol
Bondarenko, Svitlana P., Ishchenko, Vera N., Frasinyuk, Mykhaylo S.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.11.2018)
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.11.2018)
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Journal Article
Antineoplastic Isoflavonoids Derived from Intermediate ortho-Quinone Methides Generated from Mannich Bases
Frasinyuk, Mykhaylo S., Mrug, Galyna P., Bondarenko, Svitlana P., Khilya, Volodymyr P., Sviripa, Vitaliy M., Syrotchuk, Oleksandr A., Zhang, Wen, Cai, Xianfeng, Fiandalo, Michael V., Mohler, James L., Liu, Chunming, Watt, David S.
Published in ChemMedChem (17.03.2016)
Published in ChemMedChem (17.03.2016)
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Journal Article
Development of 6H-chromeno[3,4-c]pyrido[3′,2′:4,5]thieno[2,3-e]pyridazin-6-ones as Par-4 secretagogues
Frasinyuk, Mykhaylo S., Bondarenko, Svitlana P., Sviripa, Vitaliy M., Burikhanov, Ravshan, Rangnekar, Vivek M., Liu, Chunming, Watt, David S.
Published in Tetrahedron letters (03.06.2015)
Published in Tetrahedron letters (03.06.2015)
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