Structure–Activity Relationship of Inositol Thiophosphate Analogs as Allosteric Activators of Clostridioides difficile Toxin B
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Published in Journal of medicinal chemistry (26.09.2024)
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Novel Quinazoline Derivatives as Highly Effective A2A Adenosine Receptor Antagonists
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Published in Molecules (Basel, Switzerland) (14.08.2024)
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High ligand efficiency quinazoline compounds as novel A2A adenosine receptor antagonists
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Published in European journal of medicinal chemistry (05.11.2022)
Published in European journal of medicinal chemistry (05.11.2022)
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Quinazoline and phthalazine derivatives as novel melatonin receptor ligands analogues of agomelatine
Bolteau, Raphaël, Descamps, Florian, Ettaoussi, Mohamed, Caignard, Daniel H., Delagrange, Philippe, Melnyk, Patricia, Yous, Saïd
Published in European journal of medicinal chemistry (01.03.2020)
Published in European journal of medicinal chemistry (01.03.2020)
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Design and synthesis of 2,6-disubstituted-8-amino imidazo[1,2a]pyridines, a promising privileged structure
Boulahjar, Rajaa, Rincon Arias, Angela, Bolteau, Raphaël, Renault, Nicolas, Coevoet, Mathilde, Barczyk, Amélie, Duroux, Romain, Yous, Saïd, Melnyk, Patricia, Agouridas, Laurence
Published in Bioorganic & medicinal chemistry (23.07.2018)
Published in Bioorganic & medicinal chemistry (23.07.2018)
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High ligand efficiency quinazoline compounds as novel A(2A) adenosine receptor antagonists
Bolteau, Raphael, Duroux, Romain, Laversin, Amelie, Vreulz, Brandon, Shiriaeva, Anna, Stauch, Benjamin, Han, Gye Won, Cherezov, Vadim, Renault, Nicolas, Barczyk, Amelie, Ravez, Severine, Coevoet, Mathilde, Melnyk, Patricia, Liberelle, Maxime, Yous, Said
Published in European journal of medicinal chemistry (05.11.2022)
Published in European journal of medicinal chemistry (05.11.2022)
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