Ruthenium Half-Sandwich Type Complexes with Bidentate Monosaccharide Ligands Show Antineoplastic Activity in Ovarian Cancer Cell Models through Reactive Oxygen Species Production
Kacsir, István, Sipos, Adrienn, Ujlaki, Gyula, Buglyó, Péter, Somsák, László, Bai, Péter, Bokor, Éva
Published in International journal of molecular sciences (01.10.2021)
Published in International journal of molecular sciences (01.10.2021)
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Reactive Oxygen Species Production Is Responsible for Antineoplastic Activity of Osmium, Ruthenium, Iridium and Rhodium Half-Sandwich Type Complexes with Bidentate Glycosyl Heterocyclic Ligands in Various Cancer Cell Models
Kacsir, István, Sipos, Adrienn, Bényei, Attila, Janka, Eszter, Buglyó, Péter, Somsák, László, Bai, Péter, Bokor, Éva
Published in International journal of molecular sciences (12.01.2022)
Published in International journal of molecular sciences (12.01.2022)
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Synthesis of New C- and N-β-d-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase
Kun, Sándor, Bokor, Éva, Sipos, Ádám, Docsa, Tibor, Somsák, László
Published in Molecules (Basel, Switzerland) (15.03.2018)
Published in Molecules (Basel, Switzerland) (15.03.2018)
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C‑Glucopyranosyl-1,2,4-triazoles As New Potent Inhibitors of Glycogen Phosphorylase
Bokor, Éva, Docsa, Tibor, Gergely, Pál, Somsák, László
Published in ACS medicinal chemistry letters (11.07.2013)
Published in ACS medicinal chemistry letters (11.07.2013)
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Amide-1,2,3-triazole bioisosterism: the glycogen phosphorylase case
Chrysina, Evangelia D., Bokor, Eva, Alexacou, Kyra-Melinda, Charavgi, Maria-Despoina, Oikonomakos, George N., Zographos, Spyros E., Leonidas, Demetres D., Oikonomakos, Nikos G., Laszlo, Somsak
Published in Tetrahedron: asymmetry (07.05.2009)
Published in Tetrahedron: asymmetry (07.05.2009)
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Toxic metal phytoextraction potential and health-risk parameters of some cultivated plants when grown in metal-contaminated river sediment of Danube, near an industrial town
Kovács-Bokor, Éva, Domokos, Endre, Biró, Borbála
Published in Environmental geochemistry and health (01.06.2021)
Published in Environmental geochemistry and health (01.06.2021)
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Half-Sandwich Type Platinum-Group Metal Complexes of C -Glucosaminyl Azines: Synthesis and Antineoplastic and Antimicrobial Activities
Kacsir, István, Sipos, Adrienn, Major, Evelin, Bajusz, Nikolett, Bényei, Attila, Buglyó, Péter, Somsák, László, Kardos, Gábor, Bai, Péter, Bokor, Éva
Published in Molecules (Basel, Switzerland) (29.03.2023)
Published in Molecules (Basel, Switzerland) (29.03.2023)
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Synthesis of C-β-d-glucopyranosyl derivatives of some fused azoles for the inhibition of glycogen phosphorylase
Szennyes, Eszter, Bokor, Éva, Docsa, Tibor, Sipos, Ádám, Somsák, László
Published in Carbohydrate research (15.01.2019)
Published in Carbohydrate research (15.01.2019)
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First representatives of C-glycosyl 1,2,4,5-tetrazines: synthesis of 3-beta-d-glucopyranosyl 1,2,4,5-tetrazines and their transformation into 3-beta-d-glucopyranosyl pyridazines
Bokor, Eva, Kecskes, Dora T., Gombas, Ferenc, Feher, Alexandra, Kardos, Eszter, Dabian, Akram, Vonza, Zsofia, Szennyes, Eszter, Somsak, Laszlo
Published in New journal of chemistry (19.12.2022)
Published in New journal of chemistry (19.12.2022)
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Identification of C‑β‑d‑Glucopyranosyl Azole-Type Inhibitors of Glycogen Phosphorylase That Reduce Glycogenolysis in Hepatocytes: In Silico Design, Synthesis, in Vitro Kinetics, and ex Vivo Studies
Barr, Daniel, Szennyes, Eszter, Bokor, Éva, Al-Oanzi, Ziad H, Moffatt, Colin, Kun, Sándor, Docsa, Tibor, Sipos, Ádám, Davies, Matthew P, Mathomes, Rachel T, Snape, Timothy J, Agius, Loranne, Somsák, László, Hayes, Joseph M
Published in ACS chemical biology (19.07.2019)
Published in ACS chemical biology (19.07.2019)
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Glycogen phosphorylase inhibition improves beta cell function
Nagy, Lilla, Márton, Judit, Vida, András, Kis, Gréta, Bokor, Éva, Kun, Sándor, Gönczi, Mónika, Docsa, Tibor, Tóth, Attila, Antal, Miklós, Gergely, Pál, Csóka, Balázs, Pacher, Pal, Somsák, László, Bai, Péter
Published in British journal of pharmacology (01.01.2018)
Published in British journal of pharmacology (01.01.2018)
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Nanomolar Inhibitors of Glycogen Phosphorylase Based on β‑d‑Glucosaminyl Heterocycles: A Combined Synthetic, Enzyme Kinetic, and Protein Crystallography Study
Bokor, Éva, Kyriakis, Efthimios, Solovou, Theodora G.A, Koppány, Csenge, Kantsadi, Anastassia L, Szabó, Katalin E, Szakács, Andrea, Stravodimos, George A, Docsa, Tibor, Skamnaki, Vassiliki T, Zographos, Spyros E, Gergely, Pál, Leonidas, Demetres D, Somsák, László
Published in Journal of medicinal chemistry (22.11.2017)
Published in Journal of medicinal chemistry (22.11.2017)
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New synthesis of 3-(β-D-glucopyranosyl)-5-substituted-1,2,4-triazoles, nanomolar inhibitors of glycogen phosphorylase
Kun, Sándor, Bokor, Éva, Varga, Gergely, Szőcs, Béla, Páhi, András, Czifrák, Katalin, Tóth, Marietta, Juhász, László, Docsa, Tibor, Gergely, Pál, Somsák, László
Published in European journal of medicinal chemistry (09.04.2014)
Published in European journal of medicinal chemistry (09.04.2014)
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Half sandwich-type osmium, ruthenium, iridium and rhodium complexes with bidentate glycosyl heterocyclic ligands induce cytostasis in platinum-resistant ovarian cancer cells and bacteriostasis in Gram-positive multiresistant bacteria
Kacsir, István, Sipos, Adrienn, Kiss, Tímea, Major, Evelin, Bajusz, Nikolett, Tóth, Emese, Buglyó, Péter, Somsák, László, Kardos, Gábor, Bai, Péter, Bokor, Éva
Published in Frontiers in chemistry (30.01.2023)
Published in Frontiers in chemistry (30.01.2023)
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Dual-Target Compounds against Type 2 Diabetes Mellitus : Proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors
Sipos, Ádám, Szennyes, Eszter, Hajnal, Nikolett Éva, Kun, Sándor, Szabó, Katalin E, Uray, Karen, Somsák, László, Docsa, Tibor, Bokor, Éva
Published in Pharmaceuticals (Basel, Switzerland) (15.04.2021)
Published in Pharmaceuticals (Basel, Switzerland) (15.04.2021)
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