GPCRdb: an information system for G protein-coupled receptors
Isberg, Vignir, Mordalski, Stefan, Munk, Christian, Rataj, Krzysztof, Harpsøe, Kasper, Hauser, Alexander S, Vroling, Bas, Bojarski, Andrzej J, Vriend, Gert, Gloriam, David E
Published in Nucleic acids research (04.01.2016)
Published in Nucleic acids research (04.01.2016)
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Journal Article
GPCRdb: the G protein‐coupled receptor database – an introduction
Munk, C, Isberg, V, Mordalski, S, Harpsøe, K, Rataj, K, Hauser, A S, Kolb, P, Bojarski, A J, Vriend, G, Gloriam, D E
Published in British journal of pharmacology (01.07.2016)
Published in British journal of pharmacology (01.07.2016)
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Molecular Modeling of µ Opioid Receptor Ligands with Various Functional Properties: PZM21, SR-17018, Morphine, and Fentanyl-Simulated Interaction Patterns Confronted with Experimental Data
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Published in Molecules (Basel, Switzerland) (12.10.2020)
Published in Molecules (Basel, Switzerland) (12.10.2020)
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Multifunctional Ligands with Glycogen Synthase Kinase 3 Inhibitory Activity as a New Direction in Drug Research for Alzheimer's Disease
Jankowska, Agnieszka, Satała, Grzegorz, Bojarski, Andrzej J, Pawłowski, Maciej, Chłoń-Rzepa, GraŻyna
Published in Current medicinal chemistry (01.01.2021)
Published in Current medicinal chemistry (01.01.2021)
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Exploring protein hotspots by optimized fragment pharmacophores
Bajusz, Dávid, Wade, Warren S, Satała, Grzegorz, Bojarski, Andrzej J, Ilaš, Janez, Ebner, Jessica, Grebien, Florian, Papp, Henrietta, Jakab, Ferenc, Douangamath, Alice, Fearon, Daren, von Delft, Frank, Schuller, Marion, Ahel, Ivan, Wakefield, Amanda, Vajda, Sándor, Gerencsér, János, Pallai, Péter, Keserű, György M
Published in Nature communications (27.05.2021)
Published in Nature communications (27.05.2021)
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GPCRdb in 2018: adding GPCR structure models and ligands
Pándy-Szekeres, Gáspár, Munk, Christian, Tsonkov, Tsonko M, Mordalski, Stefan, Harpsøe, Kasper, Hauser, Alexander S, Bojarski, Andrzej J, Gloriam, David E
Published in Nucleic acids research (04.01.2018)
Published in Nucleic acids research (04.01.2018)
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Ligand-guided homology modelling of the GABAB2 subunit of the GABAB receptor
Freyd, Thibaud, Warszycki, Dawid, Mordalski, Stefan, Bojarski, Andrzej J, Sylte, Ingebrigt, Gabrielsen, Mari
Published in PloS one (01.03.2017)
Published in PloS one (01.03.2017)
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Journal Article
GPCRdb: an information system for G protein-coupled receptors
Isberg, Vignir, Mordalski, Stefan, Munk, Christian, Rataj, Krzysztof, Harpsøe, Kasper, Hauser, Alexander S, Vroling, Bas, Bojarski, Andrzej J, Vriend, Gert, Gloriam, David E
Published in Nucleic acids research (17.03.2017)
Published in Nucleic acids research (17.03.2017)
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Impact of the Substitution Pattern at the Basic Center and Geometry of the Amine Fragment on 5-HT6 and D3R Affinity in the 1H-Pyrrolo[3,2-c]quinoline Series
Grychowska, Katarzyna, Pietruś, Wojciech, Kulawik, Ludmiła, Bento, Ophélie, Satała, Grzegorz, Bantreil, Xavier, Lamaty, Frédéric, Bojarski, Andrzej J., Gołębiowska, Joanna, Nikiforuk, Agnieszka, Marin, Philippe, Chaumont-Dubel, Séverine, Kurczab, Rafał, Zajdel, Paweł
Published in Molecules (Basel, Switzerland) (21.01.2023)
Published in Molecules (Basel, Switzerland) (21.01.2023)
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An Algorithm to Identify Target-Selective Ligands - A Case Study of 5-HT7/5-HT1A Receptor Selectivity
Kurczab, Rafał, Canale, Vittorio, Zajdel, Paweł, Bojarski, Andrzej J
Published in PloS one (07.06.2016)
Published in PloS one (07.06.2016)
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Activation of the 5-HT7 receptor and MMP-9 signaling module in the hippocampal CA1 region is necessary for the development of depressive-like behavior
Bijata, Monika, Bączyńska, Ewa, Müller, Franziska E., Bijata, Krystian, Masternak, Julia, Krzystyniak, Adam, Szewczyk, Bernadeta, Siwiec, Marcin, Antoniuk, Svitlana, Roszkowska, Matylda, Figiel, Izabela, Magnowska, Marta, Olszyński, Krzysztof H., Wardak, Agnieszka D., Hogendorf, Adam, Ruszczycki, Błażej, Gorinski, Nataliya, Labus, Josephine, Stępień, Tomasz, Tarka, Sylwia, Bojarski, Andrzej J., Tokarski, Krzysztof, Filipkowski, Robert K., Ponimaskin, Evgeni, Wlodarczyk, Jakub
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Published in Cell reports (Cambridge) (15.03.2022)
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Published in International journal of molecular sciences (05.07.2021)
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In Silico Methods for the Discovery of Orthosteric GABAB Receptor Compounds
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Published in Molecules (Basel, Switzerland) (07.03.2019)
Published in Molecules (Basel, Switzerland) (07.03.2019)
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Substructural Connectivity Fingerprint and Extreme Entropy Machines-A New Method of Compound Representation and Analysis
Rataj, Krzysztof, Czarnecki, Wojciech, Podlewska, Sabina, Pocha, Agnieszka, Bojarski, Andrzej J
Published in Molecules (Basel, Switzerland) (23.05.2018)
Published in Molecules (Basel, Switzerland) (23.05.2018)
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