Fourier Transform Mass Spectrometry and Nuclear Magnetic Resonance Analysis for the Rapid and Accurate Characterization of Hexacosanoylceramide
Ross, Charles W, Simonsick, William J, Bogusky, Michael J, Celikay, Recep W, Guare, James P, Newton, Randall C
Published in International journal of molecular sciences (01.07.2016)
Published in International journal of molecular sciences (01.07.2016)
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Conformational analysis of N,N-disubstituted-1,4-diazepane orexin receptor antagonists and implications for receptor binding
Cox, Christopher D., McGaughey, Georgia B., Bogusky, Michael J., Whitman, David B., Ball, Richard G., Winrow, Christopher J., Renger, John J., Coleman, Paul J.
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
Published in Bioorganic & medicinal chemistry letters (01.06.2009)
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Two Tarantula Peptides Inhibit Activation of Multiple Sodium Channels
Middleton, Richard E, Warren, Vivien A, Kraus, Richard L, Hwang, Jeremy C, Liu, Chou J, Dai, Ge, Brochu, Richard M, Kohler, Martin G, Gao, Ying-Duo, Garsky, Victor M, Bogusky, Michael J, Mehl, John T, Cohen, Charles J, Smith, McHardy M
Published in Biochemistry (Easton) (17.12.2002)
Published in Biochemistry (Easton) (17.12.2002)
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Discovery of a Potent, CNS‐Penetrant Orexin Receptor Antagonist Based on an N,N‐Disubstituted‐1,4‐diazepane Scaffold that Promotes Sleep in Rats
Whitman, David B., Cox, Christopher D., Breslin, Michael J., Brashear, Karen M., Schreier, John D., Bogusky, Michael J., Bednar, Rodney A., Lemaire, Wei, Bruno, Joseph G., Hartman, George D., Reiss , Duane R., Harrell, C. Meacham, Kraus, Richard L., Li, Yuxing, Garson, Susan L., Doran, Scott M., Prueksaritanont, Thomayant, Li, Chunze, Winrow, Christopher J., Koblan, Kenneth S., Renger, John J., Coleman, Paul J.
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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Discovery of the Dual Orexin Receptor Antagonist [(7R)-4-(5-Chloro-1,3-benzoxazol-2-yl)-7-methyl-1,4-diazepan-1-yl][5-methyl-2-(2H-1,2,3-triazol-2-yl)phenyl]methanone (MK-4305) for the Treatment of Insomnia
Cox, Christopher D, Breslin, Michael J, Whitman, David B, Schreier, John D, McGaughey, Georgia B, Bogusky, Michael J, Roecker, Anthony J, Mercer, Swati P, Bednar, Rodney A, Lemaire, Wei, Bruno, Joseph G, Reiss, Duane R, Harrell, C. Meacham, Murphy, Kathy L, Garson, Susan L, Doran, Scott M, Prueksaritanont, Thomayant, Anderson, Wayne B, Tang, Cuyue, Roller, Shane, Cabalu, Tamara D, Cui, Donghui, Hartman, George D, Young, Steven D, Koblan, Ken S, Winrow, Christopher J, Renger, John J, Coleman, Paul J
Published in Journal of medicinal chemistry (22.07.2010)
Published in Journal of medicinal chemistry (22.07.2010)
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Conformational Restriction of Flexible Ligands Guided by the Transferred NOE Experiment: Potent Macrocyclic Inhibitors of Farnesyltransferase
Dinsmore, Christopher J, Bogusky, Michael J, Culberson, J. Christopher, Bergman, Jeffrey M, Homnick, Carl F, Zartman, C. Blair, Mosser, Scott D, Schaber, Michael D, Robinson, Ronald G, Koblan, Kenneth S, Huber, Hans E, Graham, Samuel L, Hartman, George D, Huff, Joel R, Williams, Theresa M
Published in Journal of the American Chemical Society (07.03.2001)
Published in Journal of the American Chemical Society (07.03.2001)
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Discovery of [(2R,5R)-5-{[(5-Fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl][5-methyl-2-(pyrimidin-2-yl)phenyl]methanone (MK-6096): A Dual Orexin Receptor Antagonist with Potent Sleep-Promoting Properties
Coleman, Paul J., Schreier, John D., Cox, Christopher D., Breslin, Michael J., Whitman, David B., Bogusky, Michael J., McGaughey, Georgia B., Bednar, Rodney A., Lemaire, Wei, Doran, Scott M., Fox, Steven V., Garson, Susan L., Gotter, Anthony L., Harrell, C. Meacham, Reiss, Duane R., Cabalu, Tamara D., Cui, Donghui, Prueksaritanont, Thomayant, Stevens, Joanne, Tannenbaum, Pamela L., Ball, Richard G., Stellabott, Joyce, Young, Steven D., Hartman, George D., Winrow, Christopher J., Renger, John J.
Published in ChemMedChem (05.03.2012)
Published in ChemMedChem (05.03.2012)
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Structure-Function Relationships in the Neuropeptide S Receptor: MOLECULAR CONSEQUENCES OF THE ASTHMA-ASSOCIATED MUTATION N107I
Bernier, Virginie, Stocco, Rino, Bogusky, Michael J, Joyce, Joseph G, Parachoniak, Christine, Grenier, Karl, Arget, Michael, Mathieu, Marie-Claude, O'Neill, Gary P, Slipetz, Deborah, Crackower, Michael A, Tan, Christopher M, Therien, Alex G
Published in The Journal of biological chemistry (25.08.2006)
Published in The Journal of biological chemistry (25.08.2006)
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Enhancement of alpha -helicity in the HIV-1 inhibitory peptide DP178 leads to an increased affinity for human monoclonal antibody 2F5 but does not elicit neutralizing responses in vitro. Implications for vaccine design
Joyce, Joseph G, Hurni, William M, Bogusky, Michael J, Garsky, Victor M, Liang, Xiaoping, Citron, Michael P, Danzeisen, Renee C, Miller, Michael D, Shiver, John W, Keller, Paul M
Published in The Journal of biological chemistry (29.11.2002)
Published in The Journal of biological chemistry (29.11.2002)
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Design and synthesis of conformationally constrained N,N-disubstituted 1,4-diazepanes as potent orexin receptor antagonists
Coleman, Paul J., Schreier, John D., McGaughey, Georgia B., Bogusky, Michael J., Cox, Christopher D., Hartman, George D., Ball, Richard G., Harrell, C. Meacham, Reiss, Duane R., Prueksaritanont, Thomayant, Winrow, Christopher J., Renger, John J.
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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3-Aminopyrrolidinone Farnesyltransferase Inhibitors: Design of Macrocyclic Compounds with Improved Pharmacokinetics and Excellent Cell Potency
Bell, Ian M, Gallicchio, Steven N, Abrams, Marc, Beese, Lorena S, Beshore, Douglas C, Bhimnathwala, Hema, Bogusky, Michael J, Buser, Carolyn A, Culberson, J. Christopher, Davide, Joseph, Ellis-Hutchings, Michelle, Fernandes, Christine, Gibbs, Jackson B, Graham, Samuel L, Hamilton, Kelly A, Hartman, George D, Heimbrook, David C, Homnick, Carl F, Huber, Hans E, Huff, Joel R, Kassahun, Kelem, Koblan, Kenneth S, Kohl, Nancy E, Lobell, Robert B, Lynch, Joseph J, Robinson, Ronald, Rodrigues, A. David, Taylor, Jeffrey S, Walsh, Eileen S, Williams, Theresa M, Zartman, C. Blair
Published in Journal of medicinal chemistry (06.06.2002)
Published in Journal of medicinal chemistry (06.06.2002)
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Synthesis and biological evaluation of unnatural canthine alkaloids
Lindsley, Craig W., Bogusky, Michael J., Leister, William H., McClain, Ray T., Robinson, Ronald G., Barnett, Stanley F., Defeo-Jones, Deborah, Ross, Charles W., Hartman, George D.
Published in Tetrahedron letters (18.04.2005)
Published in Tetrahedron letters (18.04.2005)
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Cover Picture: Discovery of [(2R,5R)-5-{[(5-Fluoropyridin-2-yl)oxy]methyl}-2-methylpiperidin-1-yl][5-methyl-2-(pyrimidin-2-yl)phenyl]methanone (MK-6096): A Dual Orexin Receptor Antagonist with Potent Sleep-Promoting Properties (ChemMedChem 3/2012)
Coleman, Paul J., Schreier, John D., Cox, Christopher D., Breslin, Michael J., Whitman, David B., Bogusky, Michael J., McGaughey, Georgia B., Bednar, Rodney A., Lemaire, Wei, Doran, Scott M., Fox, Steven V., Garson, Susan L., Gotter, Anthony L., Harrell, C. Meacham, Reiss, Duane R., Cabalu, Tamara D., Cui, Donghui, Prueksaritanont, Thomayant, Stevens, Joanne, Tannenbaum, Pamela L., Ball, Richard G., Stellabott, Joyce, Young, Steven D., Hartman, George D., Winrow, Christopher J., Renger, John J.
Published in ChemMedChem (05.03.2012)
Published in ChemMedChem (05.03.2012)
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Cyclopsychotride A, a Biologically Active, 31-Residue Cyclic Peptide Isolated from Psychotria longipes
Witherup, Keith M, Bogusky, Michael J, Anderson, Paul S, Ramjit, Harri, Ransom, Richard W, Wood, Theresa, Sardana, Mohinder
Published in Journal of natural products (Washington, D.C.) (01.12.1994)
Published in Journal of natural products (Washington, D.C.) (01.12.1994)
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Potent antagonists of the Kv1.5 potassium channel: Synthesis and evaluation of analogous N, N-diisopropyl-2-(pyridine-3-yl)acetamides
Nanda, Kausik K., Brad Nolt, M., Cato, Matthew J., Kane, Stefanie A., Kiss, Laszlo, Spencer, Robert H., Wang, Jixin, Lynch, Joseph J., Regan, Christopher P., Stump, Gary L., Li, Bing, White, Rebecca, Yeh, Suzie, Bogusky, Michael J., Bilodeau, Mark T., Dinsmore, Christopher J., Lindsley, Craig W., Hartman, George D., Wolkenberg, Scott E., Wesley Trotter, B.
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
Published in Bioorganic & medicinal chemistry letters (15.11.2006)
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Journal Article
Structure-Function Relationships in the Neuropeptide S Receptor
Bernier, Virginie, Stocco, Rino, Bogusky, Michael J., Joyce, Joseph G., Parachoniak, Christine, Grenier, Karl, Arget, Michael, Mathieu, Marie-Claude, O'Neill, Gary P., Slipetz, Deborah, Crackower, Michael A., Tan, Christopher M., Therien, Alex G.
Published in The Journal of biological chemistry (25.08.2006)
Published in The Journal of biological chemistry (25.08.2006)
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Progress towards the development of a HIV-1 gp41-directed vaccine
McGaughey, Georgia B, Barbato, Gaetano, Bianchi, Elisabetta, Freidinger, Roger M, Garsky, Victor M, Hurni, William M, Joyce, Joseph G, Liang, Xiaoping, Miller, Michael D, Pessi, Antonello, Shiver, John W, Bogusky, Michael J
Published in Current HIV research (01.04.2004)
Published in Current HIV research (01.04.2004)
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3,8-Diazabicyclo[3.2.1]octan-2-one Peptide Mimetics: Synthesis of a Conformationally Restricted Inhibitor of Farnesyltransferase
Dinsmore, Christopher J, Bergman, Jeffrey M, Bogusky, Michael J, Culberson, J. Christopher, Hamilton, Kelly A, Graham, Samuel L
Published in Organic letters (22.03.2001)
Published in Organic letters (22.03.2001)
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Journal Article
N-Arylpiperazinone Inhibitors of Farnesyltransferase: Discovery and Biological Activity
Williams, Theresa M, Bergman, Jeffrey M, Brashear, Karen, Breslin, Michael J, Dinsmore, Christopher J, Hutchinson, John H, MacTough, Suzanne C, Stump, Craig A, Wei, Donna D, Zartman, C. Blair, Bogusky, Michael J, Culberson, J. Christopher, Buser-Doepner, Carolyn, Davide, Joseph, Greenberg, Ian B, Hamilton, Kelly A, Koblan, Kenneth S, Kohl, Nancy E, Liu, Dongming, Lobell, Robert B, Mosser, Scott D, O'Neill, Timothy J, Rands, Elaine, Schaber, Michael D, Wilson, Francine, Senderak, Edith, Motzel, Sherri L, Gibbs, Jackson B, Graham, Samuel L, Heimbrook, David C, Hartman, George D, Oliff, Allen I, Huff, Joel R
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Dynamics of the multidomain fibrinolytic protein urokinase from two-dimensional NMR
Oswald, R E, Bogusky, M J, Bamberger, M, Smith, R A, Dobson, C M
Published in Nature (London) (09.02.1989)
Published in Nature (London) (09.02.1989)
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