Synthesis of water-soluble (aminoalkyl)camptothecin analogs: inhibition of topoisomerase I and antitumor activity
Kingsbury, William D, Boehm, Jeffrey C, Jakas, Dalia R, Holden, Kenneth G, Hecht, Sidney M, Gallagher, Gregory, Caranfa, Mary Jo, McCabe, Francis L, Faucette, Leo F, Johnson, Randall K, Hertzberg, Robert P
Published in Journal of medicinal chemistry (01.01.1991)
Published in Journal of medicinal chemistry (01.01.1991)
Get full text
Journal Article
1-Substituted 4-Aryl-5-pyridinylimidazoles: A New Class of Cytokine Suppressive Drugs with Low 5-Lipoxygenase and Cyclooxygenase Inhibitory Potency
Boehm, Jeffrey C, Smietana, Juanita M, Sorenson, Margaret E, Garigipati, Ravi S, Gallagher, Timothy F, Sheldrake, Peter L, Bradbeer, Jeremy, Badger, Alison M, Laydon, Jeffrey T, Lee, John C, Hillegass, Leonard M, Griswold, Donald E, Breton, John J, Chabot-Fletcher, Marie C, Adams, Jerry L
Published in Journal of medicinal chemistry (27.09.1996)
Published in Journal of medicinal chemistry (27.09.1996)
Get full text
Journal Article
Structural basis of inhibitor selectivity in MAP kinases
Wang, Zhulun, Canagarajah, Bertram J, Boehm, Jeffrey C, Kassisà, Skouki, Cobb, Melanie H, Young, Peter R, Abdel-Meguid, Sherin, Adams, Jerry L, Goldsmith, Elizabeth J
Published in Structure (London) (15.09.1998)
Published in Structure (London) (15.09.1998)
Get full text
Journal Article
Pyrimidinylimidazole inhibitors of CSBP/P38 kinase demonstrating decreased inhibition of hepatic cytochrome P450 enzymes
Adams, Jerry L., Boehm, Jeffrey C., Kassis, Shouki, Gorycki, Peter D., Webb, Edward F., Hall, Ralph, Sorenson, Margaret, Lee, John C., Ayrton, Andrew, Griswold, Don E., Gallagher, Timothy F.
Published in Bioorganic & medicinal chemistry letters (17.11.1998)
Published in Bioorganic & medicinal chemistry letters (17.11.1998)
Get full text
Journal Article
Pyrimidinylimidazole inhibitors of p38: cyclic N-1 imidazole substituents enhance p38 kinase inhibition and oral activity
Adams, Jerry L., Boehm, Jeffrey C., Gallagher, Timothy F., Kassis, Shouki, Webb, Edward F., Hall, Ralph, Sorenson, Margaret, Garigipati, Ravi, Griswold, Don E., Lee, John C.
Published in Bioorganic & medicinal chemistry letters (05.11.2001)
Published in Bioorganic & medicinal chemistry letters (05.11.2001)
Get full text
Journal Article
Regulation of stress-induced cytokine production by pyridinylimidazoles; inhibition of CSBP kinase
Gallagher, Timothy F., Seibel, George L., Kassis, Shouki, Laydon, Jeffrey T., Blumenthal, Mary Jane, Lee, John C., Lee, Dennis, Boehm, Jeffrey C., Fier-Thompson, Susan M., Abt, Jeffrey W., Soreson, Margaret E., Smietana, Juanita M., Hall, Ralph F., Garigipati, Ravi S., Bender, Paul E., Erhard, Karl F., Krog, Arnold J., Hofmann, Glenn A., Sheldrake, Peter L., McDonnell, Peter C., Kumar, Sanjay, Young, Peter R., Adams, Jerry L.
Published in Bioorganic & medicinal chemistry (01.01.1997)
Published in Bioorganic & medicinal chemistry (01.01.1997)
Get full text
Journal Article
Multiplicity of peptide permeases in Candida albicans: evidence from novel chromophoric peptides
McCarthy, P.J, Nisbet, L.J, Boehm, J.C, Kingsbury, W.D
Published in Journal of Bacteriology (01.06.1985)
Published in Journal of Bacteriology (01.06.1985)
Get full text
Journal Article
Disease‐modifying activity of SB 242235, a selective inhibitor of p38 mitogen‐activated protein kinase, in rat adjuvant‐induced arthritis
Badger, Alison M., Griswold, Don E., Kapadia, Rasesh, Blake, Simon, Swift, Barbara A., Hoffman, Sandy J., Stroup, George B., Webb, Edward, Rieman, David J., Gowen, Maxine, Boehm, Jeffrey C., Adams, Jerry L., Lee, John C.
Published in Arthritis and rheumatism (01.01.2000)
Published in Arthritis and rheumatism (01.01.2000)
Get full text
Journal Article
A novel peptide delivery system involving peptidase activated prodrugs as antimicrobial agents. Synthesis and biological activity of peptidyl derivatives of 5-fluorouracil
Kingsbury, William D, Boehm, Jeffrey C, Mehta, Rajanikant J, Grappel, Sarah F, Gilvarg, Charles
Published in Journal of medicinal chemistry (01.11.1984)
Published in Journal of medicinal chemistry (01.11.1984)
Get full text
Journal Article
Synthesis and LTB4 receptor antagonist activities of the naturally occurring LTB4 receptor antagonist leucettamine A and related analogs
Boehm, Jeffrey C, Gleason, John G, Pendrak, Israil, Sarau, Henry M, Schmidt, Dulcie B, Foley, James J, Kingsbury, William D
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
Synthesis of structural analogs of leukotriene B4 and their receptor binding activity
Kingsbury, William D, Pendrak, Israil, Leber, Jack D, Boehm, Jeffery C, Mallet, Brenda, Sarau, Henry M, Foley, James J, Schmidt, Dulcie B, Daines, Robert A
Published in Journal of medicinal chemistry (01.10.1993)
Published in Journal of medicinal chemistry (01.10.1993)
Get full text
Journal Article
Semisynthetic cephalosporins. Synthesis and structure-activity relationships of analogues with 7-acyl groups derived from 2-(cyanomethylthio)acetic acid or 2-[(2,2,2-trifluoroethyl)thio]acetic acid and their sulfoxides and sulfones
DeMarinis, R M, Boehm, J C, Dunn, G L, Hoover, J R, Uri, J V, Guarini, J R, Phillips, L, Actor, P, Weisbach, J A
Published in Journal of medicinal chemistry (01.01.1977)
Published in Journal of medicinal chemistry (01.01.1977)
Get full text
Journal Article
Synthesis and biological activity of some broad-spectrum N-acylphenylglycine cephalosporins
DeMarinis, R. M, Boehm, J. C, Uri, J. V, Guarini, J. R, Phillips, L, Dunn, G. L
Published in Journal of medicinal chemistry (01.09.1977)
Published in Journal of medicinal chemistry (01.09.1977)
Get full text
Journal Article