Fragment-Based Discovery of an Apolipoprotein E4 (apoE4) Stabilizer
Petros, Andrew M, Korepanova, Alla, Jakob, Clarissa G, Qiu, Wei, Panchal, Sanjay C, Wang, Jie, Dietrich, Justin D, Brewer, Jason T, Pohlki, Frauke, Kling, Andreas, Wilcox, Kyle, Lakics, Viktor, Bahnassawy, Lamiaa, Reinhardt, Peter, Partha, Sarathy Karunan, Bodelle, Pierre M, Lake, Marc, Charych, Erik I, Stoll, Vincent S, Sun, Chaohong, Mohler, Eric G
Published in Journal of medicinal chemistry (25.04.2019)
Published in Journal of medicinal chemistry (25.04.2019)
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Targeting lysine specific demethylase 4A (KDM4A) tandem TUDOR domain – A fragment based approach
Upadhyay, Anup K., Judge, Russell A., Li, Leiming, Pithawalla, Ron, Simanis, Justin, Bodelle, Pierre M., Marin, Violeta L., Henry, Rodger F., Petros, Andrew M., Sun, Chaohong
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
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Turning a Substrate Peptide into a Potent Inhibitor for the Histone Methyltransferase SETD8
Judge, Russell A, Zhu, Haizhong, Upadhyay, Anup K, Bodelle, Pierre M, Hutchins, Charles W, Torrent, Maricel, Marin, Violeta L, Yu, Wenyu, Vedadi, Masoud, Li, Fengling, Brown, Peter J, Pappano, William N, Sun, Chaohong, Petros, Andrew M
Published in ACS medicinal chemistry letters (08.12.2016)
Published in ACS medicinal chemistry letters (08.12.2016)
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