Palbociclib Commercial Manufacturing Process Development. Part I: Control of Regioselectivity in a Grignard-Mediated SNAr Coupling
Duan, Shengquan, Place, David, Perfect, Hahdi H, Ide, Nathan D, Maloney, Mark, Sutherland, Karen, Price Wiglesworth, Kristin E, Wang, Ke, Olivier, Mark, Kong, Fangming, Leeman, Kyle, Blunt, Jon, Draper, John, McAuliffe, Marie, O’Sullivan, Maria, Lynch, Denis
Published in Organic process research & development (15.07.2016)
Published in Organic process research & development (15.07.2016)
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Journal Article
Palbociclib Commercial Manufacturing Process Development. Part I: Control of Regioselectivity in a Grignard-Mediated S N Ar Coupling
Duan, Shengquan, Place, David, Perfect, Hahdi H., Ide, Nathan D., Maloney, Mark, Sutherland, Karen, Price Wiglesworth, Kristin E., Wang, Ke, Olivier, Mark, Kong, Fangming, Leeman, Kyle, Blunt, Jon, Draper, John, McAuliffe, Marie, O’Sullivan, Maria, Lynch, Denis
Published in Organic process research & development (15.07.2016)
Published in Organic process research & development (15.07.2016)
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Journal Article
Synthesis of Filibuvir. Part I. Diastereoselective Preparation of a β‑Hydroxy Alkynyl Oxazolidinone and Conversion to a 6,6-Disubstituted 2H‑Pyranone
Singer, Robert A, Ragan, John A, Bowles, Paul, Chisowa, Esmort, Conway, Brian G, Cordi, Eric M, Leeman, Kyle R, Letendre, Leo J, Sieser, Janice E, Sluggett, Gregory W, Stanchina, Corey L, Strohmeyer, Holly, Blunt, Jon, Taylor, Stuart, Byrne, Ciaran, Lynch, Denis, Mullane, Sandra, O’Sullivan, Maria M, Whelan, Marcella
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
Synthesis of Filibuvir. Part II. Second-Generation Synthesis of a 6,6-Disubstituted 2H‑Pyranone via Dieckmann Cyclization of a β‑Acetoxy Ester
Peng, Zhihui, Ragan, John A, Colon-Cruz, Roberto, Conway, Brian G, Cordi, Eric M, Leeman, Kyle, Letendre, Leo J, Ping, Li-Jen, Sieser, Janice E, Singer, Robert A, Sluggett, Gregory W, Strohmeyer, Holly, Vanderplas, Brian C, Blunt, Jon, Mawby, Nicola, Meldrum, Kevin, Taylor, Stuart
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
Synthesis of Filibuvir. Part III. Development of a Process for the Reductive Coupling of an Aldehyde and a β‑Keto-lactone
Ide, Nathan D, Ragan, John. A, Bellavance, Gabriel, Brenek, Steve J, Cordi, Eric M, Jensen, Grace O, Jones, Kris N, LaFrance, Danny, Leeman, Kyle R, Letendre, Leo J, Place, David, Stanchina, Corey L, Sluggett, Gregory W, Strohmeyer, Holly, Blunt, Jon, Meldrum, Kevin, Taylor, Stuart, Byrne, Ciaran, Lynch, Denis, Mullane, Sandra, O’Sullivan, Maria M, Whelan, Marcella
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
Synthesis of Filibuvir. Part II. Second-Generation Synthesis of a 6,6-Disubstituted 2 H -Pyranone via Dieckmann Cyclization of a β-Acetoxy Ester
Peng, Zhihui, Ragan, John A., Colon-Cruz, Roberto, Conway, Brian G., Cordi, Eric M., Leeman, Kyle, Letendre, Leo J., Ping, Li-Jen, Sieser, Janice E., Singer, Robert A., Sluggett, Gregory W., Strohmeyer, Holly, Vanderplas, Brian C., Blunt, Jon, Mawby, Nicola, Meldrum, Kevin, Taylor, Stuart
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
Get full text
Journal Article
Synthesis of Filibuvir. Part I. Diastereoselective Preparation of a β-Hydroxy Alkynyl Oxazolidinone and Conversion to a 6,6-Disubstituted 2 H -Pyranone
Singer, Robert A., Ragan, John A., Bowles, Paul, Chisowa, Esmort, Conway, Brian G., Cordi, Eric M., Leeman, Kyle R., Letendre, Leo J., Sieser, Janice E., Sluggett, Gregory W., Stanchina, Corey L., Strohmeyer, Holly, Blunt, Jon, Taylor, Stuart, Byrne, Ciaran, Lynch, Denis, Mullane, Sandra, O’Sullivan, Maria M., Whelan, Marcella
Published in Organic process research & development (17.01.2014)
Published in Organic process research & development (17.01.2014)
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Journal Article
Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB1 Antagonist for the Treatment of Obesity
Ragan, John A, Bourassa, Dennis E, Blunt, Jon, Breen, Darragh, Busch, Frank R, Cordi, Eric M, Damon, David B, Do, Nga, Engtrakul, Alanya, Lynch, Denis, McDermott, Ruth E, Mongillo, Joseph A, O’Sullivan, Maria M, Rose, Peter R, Vanderplas, Brian C
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Journal Article
Development of a Practical and Efficient Synthesis of CP-945,598-01, a CB 1 Antagonist for the Treatment of Obesity
Ragan, John A., Bourassa, Dennis E., Blunt, Jon, Breen, Darragh, Busch, Frank R., Cordi, Eric M., Damon, David B., Do, Nga, Engtrakul, Alanya, Lynch, Denis, McDermott, Ruth E., Mongillo, Joseph A., O’Sullivan, Maria M., Rose, Peter R., Vanderplas, Brian C.
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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Journal Article