Antibody-Directed Enzyme Prodrug Therapy with the T268G Mutant of Human Carboxypeptidase A1: In Vitro and in Vivo Studies with Prodrugs of Methotrexate and the Thymidylate Synthase Inhibitors GW1031 and GW1843
Wolfe, L. A, Mullin, R. J, Laethem, R, Blumenkopf, T. A, Cory, M, Miller, J. F, Keith, B. R, Humphreys, J, Smith, G. K
Published in Bioconjugate chemistry (01.01.1999)
Published in Bioconjugate chemistry (01.01.1999)
Get full text
Journal Article
Inactivators of herpes simplex virus ribonucleotide reductase: hematological profiles and in vivo potentiation of the antiviral activity of acyclovir
SPECTOR, T, LOBE, D. C, ELLIS, M. N, BLUMENKOPF, T. A, SZCZECH, G. M
Published in Antimicrobial Agents and Chemotherapy (01.05.1992)
Published in Antimicrobial Agents and Chemotherapy (01.05.1992)
Get full text
Journal Article
2-Acetylpyridine thiocarbonohydrazones. Potent inactivators of herpes simplex virus ribonucleotide reductase
Blumenkopf, Todd A, Harrington, Joan A, Koble, Cecilia S, Bankston, Donald D, Morrison, Robert W, Bigham, Eric C, Styles, Virgil L, Spector, Thomas
Published in Journal of medicinal chemistry (01.06.1992)
Published in Journal of medicinal chemistry (01.06.1992)
Get full text
Journal Article
Toward antibody-directed enzyme prodrug therapy with the T268G mutant of human carboxypeptidase A1 and novel in vivo stable prodrugs of methotrexate
Smith, G K, Banks, S, Blumenkopf, T A, Cory, M, Humphreys, J, Laethem, R M, Miller, J, Moxham, C P, Mullin, R, Ray, P H, Walton, L M, Wolfe, 3rd, L A
Published in The Journal of biological chemistry (20.06.1997)
Published in The Journal of biological chemistry (20.06.1997)
Get full text
Journal Article
Expression and Characterization of Human Pancreatic Preprocarboxypeptidase A1 and Preprocarboxypeptidase A2
Laethem, Ronald M., Blumenkopf, Todd A., Cory, Michael, Elwell, Lynn, Moxham, Cary P., Ray, Paul H., Walton, Leslie M., Smith, Gary K.
Published in Archives of biochemistry and biophysics (01.08.1996)
Published in Archives of biochemistry and biophysics (01.08.1996)
Get full text
Journal Article
Ryanodine Action at Calcium Release Channels. 1. Importance of Hydroxyl Substituents
Jefferies, Phillip R, Blumenkopf, Todd A, Gengo, Peter J, Cole, Loretta C, Casida, John E
Published in Journal of medicinal chemistry (07.06.1996)
Published in Journal of medicinal chemistry (07.06.1996)
Get full text
Journal Article
Total synthesis of (.+-.)-fawcettimine (Burnell's base A)
Heathcock, Clayton H, Smith, Karl M, Blumenkopf, Todd A
Published in Journal of the American Chemical Society (01.08.1986)
Published in Journal of the American Chemical Society (01.08.1986)
Get full text
Journal Article
Preparation of eight-membered cyclic ethers by Lewis acid promoted acetal-alkene cyclizations
Blumenkopf, Todd A, Bratz, Matthias, Castaneda, Armando, Look, Gary C, Overman, Larry E, Rodriguez, Domingo, Thompson, Andrew S
Published in Journal of the American Chemical Society (01.05.1990)
Published in Journal of the American Chemical Society (01.05.1990)
Get full text
Journal Article
Efficient preparations of 8- and 9-membered cyclic ethers
Overman, Larry E, Blumenkopf, Todd A, Castaneda, Armando, Thompson, Andrew S
Published in Journal of the American Chemical Society (01.06.1986)
Published in Journal of the American Chemical Society (01.06.1986)
Get full text
Journal Article
Total synthesis of (.+-.)-fawcettimine
Heathcock, Clayton H, Blumenkopf, Todd A, Smith, Karl M
Published in Journal of organic chemistry (01.03.1989)
Published in Journal of organic chemistry (01.03.1989)
Get full text
Journal Article
EFFICIENT PREPARATIONS OF 8-MEMBERED AND 9-MEMBERED CYCLIC ETHERS
OVERMAN, LE, BLUMENKOPF, TA, CASTANEDA, A, THOMPSON, AS
Published in Journal of the American Chemical Society (11.06.1986)
Published in Journal of the American Chemical Society (11.06.1986)
Get full text
Journal Article