Spermidinyl-CoA-based HAT inhibitors block DNA repair and provide cancer- specific chemo-and radiosensitization
Bandyopadhyay, Keya, Banères, Jean-Louis, Martin, Aimée, Blonski, Casimir, Parello, Joseph, Gjerset, Ruth
Published in Cell cycle (Georgetown, Tex.) (01.09.2009)
Published in Cell cycle (Georgetown, Tex.) (01.09.2009)
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Journal Article
Glycolysis as a target for the design of new anti-trypanosome drugs
Verlinde, Christophe L.M.J., Hannaert, Véronique, Blonski, Casimir, Willson, Michèle, Périé, Jacques J., Fothergill-Gilmore, Linda A., Opperdoes, Fred R., Gelb, Michael H., Hol, Wim G.J., Michels, Paul A.M.
Published in Drug resistance updates (01.02.2001)
Published in Drug resistance updates (01.02.2001)
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Journal Article
Spermidinyl-CoA-based HAT inhibitors block DNA repair and provide cancer-specific chemo- and radiosensitization
Bandyopadhyay, Keya, Banères, Jean-Louis, Martin, Aimée, Blonski, Casimir, Parello, Joseph, Gjerset, Ruth
Published in Cell cycle (Georgetown, Tex.) (01.03.2010)
Published in Cell cycle (Georgetown, Tex.) (01.03.2010)
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Journal Article
Antitrypanosomal alkaloids from Polyalthia suaveolens (Annonaceae): Their effects on three selected glycolytic enzymes of Trypanosoma brucei
Ngantchou, Igor, Nyasse, Barthélemy, Denier, Colette, Blonski, Casimir, Hannaert, Véronique, Schneider, Bernd
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Journal Article
Synthesis and in vitro antikinetoplastid activity of polyamine–hydroxybenzotriazole conjugates
Jagu, Elodie, Pomel, Sébastien, Diez-Martinez, Alba, Ramiandrasoa, Florence, Krauth-Siegel, R. Luise, Pethe, Stéphanie, Blonski, Casimir, Labruère, Raphaël, Loiseau, Philippe M.
Published in Bioorganic & medicinal chemistry (01.01.2017)
Published in Bioorganic & medicinal chemistry (01.01.2017)
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Journal Article
Design, synthesis and in vitro antikinetoplastid evaluation of N-acylated putrescine, spermidine and spermine derivatives
Jagu, Elodie, Djilali, Rachid, Pomel, Sebastien, Ramiandrasoa, Florence, Pethe, Stephanie, Labruere, Raphael, Loiseau, Philippe M., Blonski, Casimir
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
Published in Bioorganic & medicinal chemistry letters (15.01.2015)
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Journal Article
Abstract 5444: Polyamine-based HAT inhibitors as therapy sensitizers
Bandyopadhyay, Keya, Banères, Jean-Louis, Martin, Aimée, Blonski, Casimir, Parello, Joseph, Gjerset, Ruth A.
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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Journal Article
New Potent Bisubstrate Inhibitors of Histone Acetyltransferase p300: Design, Synthesis and Biological Evaluation
Kwie, Franciane Ho A, Briet, Martine, Soupaya, David, Hoffmann, Pascal, Maturano, Marie, Rodriguez, Frédéric, Blonski, Casimir, Lherbet, Christian, Baudoin-Dehoux, Cécile
Published in Chemical biology & drug design (2011)
Published in Chemical biology & drug design (2011)
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Journal Article
Selective Irreversible Inhibition of Fructose 1,6-Bisphosphate Aldolase from Trypanosoma brucei
DAX, Chantal, DUFFIEUX, Francis, CHABOT, Nicolas, COINCON, Mathieu, SYGUSCH, Jurgen, MICHELS, Paul A. M., BLONSKI, Casimir
Published in Journal of medicinal chemistry (09.03.2006)
Published in Journal of medicinal chemistry (09.03.2006)
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Journal Article
Structural flexibility in Trypanosoma brucei enolase revealed by X-ray crystallography and molecular dynamics
Navarro, Marcos V. de A.S, Gomes Dias, Sandra M, Mello, Luciane V, da Silva Giotto, Maria T, Gavalda, Sabine, Blonski, Casimir, Garratt, Richard C, Rigden, Daniel J
Published in The FEBS journal (01.10.2007)
Published in The FEBS journal (01.10.2007)
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Journal Article
In vitro inhibitory effects of palmatine from Enantia chlorantha on Trypanosoma cruzi and Leishmania infantum
Nkwengoua, Ernestine Tchouboun, Ngantchou, Igor, Nyasse, Barthélemy, Denier, Colette, Blonski, Casimir, Schneider, Bernd
Published in Natural product research (01.01.2009)
Published in Natural product research (01.01.2009)
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