Functional Consequences of Cysteine Modification in the Ligand Binding Sites of Peroxisome Proliferator Activated Receptors by GW9662
Leesnitzer, Lisa M, Parks, Derek J, Bledsoe, Randy K, Cobb, Jeff E, Collins, Jon L, Consler, Thomas G, Davis, Roderick G, Hull-Ryde, Emily A, Lenhard, James M, Patel, Lisa, Plunket, Kelli D, Shenk, Jennifer L, Stimmel, Julie B, Therapontos, Christina, Willson, Timothy M, Blanchard, Steven G
Published in Biochemistry (Easton) (28.05.2002)
Published in Biochemistry (Easton) (28.05.2002)
Get full text
Journal Article
Bile Acids: Natural Ligands for an Orphan Nuclear Receptor
Parks, Derek J., Blanchard, Steven G., Bledsoe, Randy K., Chandra, Gyan, Consler, Thomas G., Kliewer, Steven A., Stimmel, Julie B., Willson, Timothy M., Zavacki, Ann Marie, Moore, David D., Lehmann, Jürgen M.
Published in Science (American Association for the Advancement of Science) (21.05.1999)
Published in Science (American Association for the Advancement of Science) (21.05.1999)
Get full text
Journal Article
Design and x-ray crystal structures of high-potency nonsteroidal glucocorticoid agonists exploiting a novel binding site on the receptor
Biggadike, Keith, Bledsoe, Randy K, Coe, Diane M, Cooper, Tony W.J, House, David, Iannone, Marie A, Macdonald, Simon J.F, Madauss, Kevin P, McLay, Iain M, Shipley, Tracy J, Taylor, Simon J, Tran, Thuy B, Uings, Iain J, Weller, Victoria, Williams, Shawn P
Published in Proceedings of the National Academy of Sciences - PNAS (27.10.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (27.10.2009)
Get full text
Journal Article
A Ligand-mediated Hydrogen Bond Network Required for the Activation of the Mineralocorticoid Receptor[boxs]
Bledsoe, Randy K., Madauss, Kevin P., Holt, Jason A., Apolito, Christopher J., Lambert, Millard H., Pearce, Kenneth H., Stanley, Thomas B., Stewart, Eugene L., Trump, Ryan P., Willson, Timothy M., Williams, Shawn P.
Published in The Journal of biological chemistry (02.09.2005)
Published in The Journal of biological chemistry (02.09.2005)
Get full text
Journal Article
Crystallization of protein-ligand complexes
Hassell, Anne M., An, Gang, Bledsoe, Randy K., Bynum, Jane M., Carter III, H. Luke, Deng, Su-Jun J., Gampe, Robert T., Grisard, Tamara E., Madauss, Kevin P., Nolte, Robert T., Rocque, Warren J., Wang, Liping, Weaver, Kurt L., Williams, Shawn P., Wisely, G. Bruce, Xu, Robert, Shewchuk, Lisa M.
Published in Acta crystallographica. Section D, Biological crystallography. (01.01.2007)
Published in Acta crystallographica. Section D, Biological crystallography. (01.01.2007)
Get full text
Journal Article
Structure and Function of the Glucocorticoid Receptor Ligand Binding Domain
Get full text
Book Chapter
Journal Article
X-ray Crystal Structure of the Novel Enhanced-Affinity Glucocorticoid Agonist Fluticasone Furoate in the Glucocorticoid Receptor−Ligand Binding Domain
Biggadike, Keith, Bledsoe, Randy K, Hassell, Anne M, Kirk, Barrie E, McLay, Iain M, Shewchuk, Lisa M, Stewart, Eugene L
Published in Journal of medicinal chemistry (26.06.2008)
Published in Journal of medicinal chemistry (26.06.2008)
Get full text
Journal Article
Orphan Nuclear Receptors Constitutive Androstane Receptor and Pregnane X Receptor Share Xenobiotic and Steroid Ligands
Moore, Linda B., Parks, Derek J., Jones, Stacey A., Bledsoe, Randy K., Consler, Thomas G., Stimmel, Julie B., Goodwin, Bryan, Liddle, Christopher, Blanchard, Steven G., Willson, Timothy M., Collins, Jon L., Kliewer, Steven A.
Published in The Journal of biological chemistry (19.05.2000)
Published in The Journal of biological chemistry (19.05.2000)
Get full text
Journal Article
The first X-ray crystal structure of the glucocorticoid receptor bound to a non-steroidal agonist
MADAUSS, Kevin P, BLEDSOE, Randy K, MCLAY, Iain, STEWART, Eugene L, UINGS, Iain J, WEINGARTEN, Gordon, WILLIAMS, Shawn P
Published in Bioorganic & medicinal chemistry (01.12.2008)
Published in Bioorganic & medicinal chemistry (01.12.2008)
Get full text
Journal Article
X-ray crystal structure of the liver X receptor beta ligand binding domain: regulation by a histidine-tryptophan switch
Williams, Shawn, Bledsoe, Randy K, Collins, Jon L, Boggs, Sharon, Lambert, Millard H, Miller, Ann B, Moore, John, McKee, David D, Moore, Linda, Nichols, Jason, Parks, Derek, Watson, Mike, Wisely, Bruce, Willson, Timothy M
Published in The Journal of biological chemistry (18.07.2003)
Published in The Journal of biological chemistry (18.07.2003)
Get full text
Journal Article
Production of monoclonal antibodies using recombinant baculovirus displaying gp64–fusion proteins
Lindley, Kathryn M, Su, Jui-Lan, Hodges, Paula K, Wisely, G.Bruce, Bledsoe, Randy K, Condreay, J.Patrick, Winegar, Deborah A, Hutchins, Jeff T, Kost, Thomas A
Published in Journal of immunological methods (03.02.2000)
Published in Journal of immunological methods (03.02.2000)
Get full text
Journal Article
Pharmacophore Analysis of the Nuclear Oxysterol Receptor LXRα
Spencer, Thomas A, Li, Dansu, Russel, Jonathon S, Collins, Jon L, Bledsoe, Randy K, Consler, Thomas G, Moore, Linda B, Galardi, Cristin M, McKee, David D, Moore, John T, Watson, Michael A, Parks, Derek J, Lambert, Millard H, Willson, Timothy M
Published in Journal of medicinal chemistry (15.03.2001)
Published in Journal of medicinal chemistry (15.03.2001)
Get full text
Journal Article
Structure-Based Design of Potent Retinoid X Receptor α Agonists
Haffner, Curt D., Lenhard, James M., Miller, Aaron B., McDougald, Darryl L., Dwornik, Kate, Ittoop, Olivia R., Gampe, Robert T., Xu, H. Eric, Blanchard, Steve, Montana, Valerie G., Consler, Tom G., Bledsoe, Randy K., Ayscue, Andrea, Croom, Dallas
Published in Journal of medicinal chemistry (08.04.2004)
Published in Journal of medicinal chemistry (08.04.2004)
Get full text
Journal Article
Cloning of the rat and human mitochondrial branched chain aminotransferases (BCAT m)
Bledsoe, Randy K, Dawson, Paul A, Hutson, Susan M
Published in Biochimica et biophysica acta (25.04.1997)
Published in Biochimica et biophysica acta (25.04.1997)
Get full text
Journal Article
Asymmetry in the PPARγ/RXRα Crystal Structure Reveals the Molecular Basis of Heterodimerization among Nuclear Receptors
Gampe, Robert T., Montana, Valerie G., Lambert, Millard H., Miller, Aaron B., Bledsoe, Randy K., Milburn, Michael V., Kliewer, Steven A., Willson, Timothy M., Xu, H.Eric
Published in Molecular cell (01.03.2000)
Published in Molecular cell (01.03.2000)
Get full text
Journal Article
X-ray Crystal Structure of the Liver X Receptor β Ligand Binding Domain
Williams, Shawn, Bledsoe, Randy K., Collins, Jon L., Boggs, Sharon, Lambert, Millard H., Miller, Ann B., Moore, John, McKee, David D., Moore, Linda, Nichols, Jason, Parks, Derek, Watson, Mike, Wisely, Bruce, Willson, Timothy M.
Published in The Journal of biological chemistry (18.07.2003)
Published in The Journal of biological chemistry (18.07.2003)
Get full text
Journal Article
X-ray Crystal Structure of the Liver X Receptor β Ligand Binding Domain
Shawn Williams, Randy K. Bledsoe, Jon L. Collins, Sharon Boggs, Millard H. Lambert, Ann B. Miller, John Moore, David D. McKee, Linda Moore, Jason Nichols, Derek Parks, Mike Watson, Bruce Wisely, Timothy M. Willson
Published in The Journal of biological chemistry (18.07.2003)
Published in The Journal of biological chemistry (18.07.2003)
Get full text
Journal Article