Fluorescent Bisphosphonate and Carboxyphosphonate Probes: A Versatile Imaging Toolkit for Applications in Bone Biology and Biomedicine
Sun, Shuting, Błażewska, Katarzyna M, Kadina, Anastasia P, Kashemirov, Boris A, Duan, Xuchen, Triffitt, James T, Dunford, James E, Russell, R. Graham G, Ebetino, Frank H, Roelofs, Anke J, Coxon, Fraser P, Lundy, Mark W, McKenna, Charles E
Published in Bioconjugate chemistry (17.02.2016)
Published in Bioconjugate chemistry (17.02.2016)
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Influence of bone affinity on the skeletal distribution of fluorescently labeled bisphosphonates in vivo
Roelofs, Anke J, Stewart, Charlotte A, Sun, Shuting, Błażewska, Katarzyna M, Kashemirov, Boris A, McKenna, Charles E, Russell, R Graham G, Rogers, Michael J, Lundy, Mark W, Ebetino, Frank H, Coxon, Fraser P
Published in Journal of bone and mineral research (01.04.2012)
Published in Journal of bone and mineral research (01.04.2012)
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Applying the prodrug strategy to alpha-phosphonocarboxylate inhibitors of Rab GGTase - synthesis and stability studies
Joachimiak, Lukasz, Janczewski, Lukasz, Ciekot, Jaroslaw, Boratynski, Janusz, Blazewska, Katarzyna
Published in Organic & biomolecular chemistry (28.06.2015)
Published in Organic & biomolecular chemistry (28.06.2015)
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Fluorescent risedronate analogues reveal bisphosphonate uptake by bone marrow monocytes and localization around osteocytes in vivo
Roelofs, Anke J, Coxon, Fraser P, Ebetino, Frank H, Lundy, Mark W, Henneman, Zachary J, Nancollas, George H, Sun, Shuting, Blazewska, Katarzyna M, Bala, Joy Lynn F, Kashemirov, Boris A, Khalid, Aysha B, McKenna, Charles E, Rogers, Michael J
Published in Journal of bone and mineral research (01.03.2010)
Published in Journal of bone and mineral research (01.03.2010)
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Host modulators of H1N1 cytopathogenicity
Ward, Samuel E, Kim, Hyun Seok, Komurov, Kakajan, Mendiratta, Saurabh, Tsai, Pei-Ling, Schmolke, Mirco, Satterly, Neal, Manicassamy, Balaji, Forst, Christian V, Roth, Michael G, García-Sastre, Adolfo, Blazewska, Katarzyna M, McKenna, Charles E, Fontoura, Beatriz M, White, Michael A
Published in PloS one (02.08.2012)
Published in PloS one (02.08.2012)
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Synthesis, stereochemistry and SAR of a series of minodronate analogues as RGGT inhibitors
Błażewska, Katarzyna M., Ni, Feng, Haiges, Ralf, Kashemirov, Boris A., Coxon, Fraser P., Stewart, Charlotte A., Baron, Rudi, Rogers, Michael J., Seabra, Miguel C., Ebetino, Frank H., McKenna, Charles E.
Published in European journal of medicinal chemistry (01.10.2011)
Published in European journal of medicinal chemistry (01.10.2011)
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Targeting Small GTPases and Their Prenylation in Diabetes Mellitus
Gendaszewska-Darmach, Edyta, Garstka, Malgorzata A, Błażewska, Katarzyna M
Published in Journal of medicinal chemistry (22.07.2021)
Published in Journal of medicinal chemistry (22.07.2021)
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Microwave-assisted synthesis of 3-formyl substituted imidazo[1,2-a]pyridines
Kusy, Damian, Maniukiewicz, Waldemar, Błażewska, Katarzyna M.
Published in Tetrahedron letters (07.11.2019)
Published in Tetrahedron letters (07.11.2019)
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RAB26 and RAB3D Are Direct Transcriptional Targets of MIST1 That Regulate Exocrine Granule Maturation
Tian, Xiaolin, Jin, Ramon U., Bredemeyer, Andrew J., Oates, Edward J., Błażewska, Katarzyna M., McKenna, Charles E., Mills, Jason C.
Published in Molecular and Cellular Biology (01.03.2010)
Published in Molecular and Cellular Biology (01.03.2010)
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Synthesis and Characterization of Novel Fluorescent Nitrogen-Containing Bisphosphonate Imaging Probes for Bone Active Drugs
Sun, Shuting, Błażewska, Katarzyna M., Kashemirov, Boris A., Roelofs, Anke J., Coxon, Fraser P., Rogers, Michael J., Ebetino, Frank H., McKenna, Michael J., McKenna, Charles E.
Published in Phosphorus, sulfur, and silicon and the related elements (01.04.2011)
Published in Phosphorus, sulfur, and silicon and the related elements (01.04.2011)
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Protein Prenyltransferases and Their Inhibitors: Structural and Functional Characterization
Marchwicka, Aleksandra, Kamińska, Daria, Monirialamdari, Mohsen, Błażewska, Katarzyna M, Gendaszewska-Darmach, Edyta
Published in International journal of molecular sciences (12.05.2022)
Published in International journal of molecular sciences (12.05.2022)
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Identification of the Privileged Position in the Imidazo[1,2‑a]pyridine Ring of Phosphonocarboxylates for Development of Rab Geranylgeranyl Transferase (RGGT) Inhibitors
Kaźmierczak, Aleksandra, Kusy, Damian, Niinivehmas, Sanna P, Gmach, Joanna, Joachimiak, Łukasz, Pentikäinen, Olli T, Gendaszewska-Darmach, Edyta, Błażewska, Katarzyna M
Published in Journal of medicinal chemistry (09.11.2017)
Published in Journal of medicinal chemistry (09.11.2017)
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Effect of Metal-Ligand Coordination Complexes on Molecular Dynamics and Structure of Cross-Linked Poly(dimethylosiloxane)
Wrzesińska, Angelika, Bobowska, Izabela, Maczugowska, Paulina, Małolepsza, Joanna, Błażewska, Katarzyna M., Wypych-Puszkarz, Aleksandra
Published in Polymers (28.07.2020)
Published in Polymers (28.07.2020)
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Rational design, optimization, and biological evaluation of novel α-Phosphonopropionic acids as covalent inhibitors of Rab geranylgeranyl transferase
Małolepsza, Joanna, Marchwicka, Aleksandra, Serwa, Remigiusz A., Niinivehmas, Sanna P., Pentikäinen, Olli T., Gendaszewska-Darmach, Edyta, Błażewska, Katarzyna M.
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2022)
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