Crystal Structure of Human Cytochrome P450 2D6
Rowland, Paul, Blaney, Frank E., Smyth, Martin G., Jones, Jo J., Leydon, Vaughan R., Oxbrow, Amanda K., Lewis, Ceri J., Tennant, Mike G., Modi, Sandeep, Eggleston, Drake S., Chenery, Richard J., Bridges, Angela M.
Published in The Journal of biological chemistry (17.03.2006)
Published in The Journal of biological chemistry (17.03.2006)
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Differences in the Central Nervous System Distribution and Pharmacology of the Mouse 5-Hydroxytryptamine-6 Receptor Compared with Rat and Human Receptors Investigated by Radioligand Binding, Site-Directed Mutagenesis, and Molecular Modeling
Hirst, Warren D, Abrahamsen, Bjarke, Blaney, Frank E, Calver, Andrew R, Aloj, Lucia, Price, Gary W, Medhurst, Andrew D
Published in Molecular pharmacology (01.12.2003)
Published in Molecular pharmacology (01.12.2003)
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2-[2-(3,4-Dichloro-phenyl)-2,3-dihydro-1H-isoindol-5-ylamino]-nicotinic Acid (PD-307243) Causes Instantaneous Current through Human Ether-a-go-go-Related Gene Potassium Channels
Gordon, Earl, Lozinskaya, Irina M, Lin, Zuojun, Semus, Simon F, Blaney, Frank E, Willette, Robert N, Xu, Xiaoping
Published in Molecular pharmacology (01.03.2008)
Published in Molecular pharmacology (01.03.2008)
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G-protein-coupled receptor dynamics: dimerization and activation models compared with experiment
Taddese, Bruck, Simpson, Lisa M, Wall, Ian D, Blaney, Frank E, Kidley, Nathan J, Clark, Henry S X, Smith, Richard E, Upton, Graham J G, Gouldson, Paul R, Psaroudakis, George, Bywater, Robert P, Reynolds, Christopher A
Published in Biochemical Society transactions (01.04.2012)
Published in Biochemical Society transactions (01.04.2012)
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CCR2: Characterization of the Antagonist Binding Site from a Combined Receptor Modeling/Mutagenesis Approach
Berkhout, Theo A, Blaney, Frank E, Bridges, Angela M, Cooper, David G, Forbes, Ian T, Gribble, Andrew D, Groot, Pieter H. E, Hardy, Adam, Ife, Robert J, Kaur, Rejbinder, Moores, Kitty E, Shillito, Helen, Willetts, Jennifer, Witherington, Jason
Published in Journal of medicinal chemistry (11.09.2003)
Published in Journal of medicinal chemistry (11.09.2003)
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Structural Determinants of Drugs Acting on the Nav1.8 Channel
Browne, Liam E., Blaney, Frank E., Yusaf, Shahnaz P., Clare, Jeff J., Wray, Dennis
Published in The Journal of biological chemistry (17.04.2009)
Published in The Journal of biological chemistry (17.04.2009)
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Functional analysis of CYP2D6.31 variant: Homology modeling suggests possible disruption of redox partner interaction by Arg440His substitution
Allorge, Delphine, Bréant, Didier, Harlow, Jacky, Chowdry, Joey, Lo-Guidice, Jean-Marc, Chevalier, Dany, Cauffiez, Christelle, Lhermitte, Michel, Blaney, Frank E., Tucker, Geoffrey T., Broly, Franck, Ellis, S. Wynne
Published in Proteins, structure, function, and bioinformatics (01.05.2005)
Published in Proteins, structure, function, and bioinformatics (01.05.2005)
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Modeling GPCR active state conformations: the β(2)-adrenergic receptor
Simpson, Lisa M, Wall, Ian D, Blaney, Frank E, Reynolds, Christopher A
Published in Proteins, structure, function, and bioinformatics (01.05.2011)
Published in Proteins, structure, function, and bioinformatics (01.05.2011)
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1,2,4-Triazolyl Azabicyclo[3.1.0]hexanes: A New Series of Potent and Selective Dopamine D3 Receptor Antagonists
Micheli, Fabrizio, Arista, Luca, Bonanomi, Giorgio, Blaney, Frank E, Braggio, Simone, Capelli, Anna Maria, Checchia, Anna, Damiani, Federica, Di-Fabio, Romano, Fontana, Stefano, Gentile, Gabriella, Griffante, Cristiana, Hamprecht, Dieter, Marchioro, Carla, Mugnaini, Manolo, Piner, Jacqui, Ratti, Emiliangelo, Tedesco, Giovanna, Tarsi, Luca, Terreni, Silvia, Worby, Angela, Ashby, Charles R, Heidbreder, Christian
Published in Journal of medicinal chemistry (14.01.2010)
Published in Journal of medicinal chemistry (14.01.2010)
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Comparison of azabicyclic esters and oxadiazoles as ligands for the muscarinic receptor
Orlek, Barry S, Blaney, Frank E, Brown, Frank, Clark, Michael S. G, Hadley, Michael S, Hatcher, John, Riley, Graham J, Rosenberg, Howard E, Wadsworth, Harry J, Wyman, Paul
Published in Journal of medicinal chemistry (01.09.1991)
Published in Journal of medicinal chemistry (01.09.1991)
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Modeling GPCR active state conformations: The β2-adrenergic receptor
Simpson, Lisa M., Wall, Ian D., Blaney, Frank E., Reynolds, Christopher A.
Published in Proteins, structure, function, and bioinformatics (01.05.2011)
Published in Proteins, structure, function, and bioinformatics (01.05.2011)
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Synthesis and Pharmacological Characterization of Novel Druglike Corticotropin-Releasing Factor 1 Antagonists
Fabio, Romano Di, St-Denis, Yves, Sabbatini, Fabio M, Andreotti, Daniele, Arban, Roberto, Bernasconi, Giovanni, Braggio, Simone, Blaney, Frank E, Capelli, Anna M, Castiglioni, Emiliano, Modugno, Enza Di, Donati, Daniele, Fazzolari, Elettra, Ratti, Emiliangelo, Feriani, Aldo, Contini, Stefania, Gentile, Gabriella, Ghirlanda, Damiano, Provera, Stefano, Marchioro, Carla, Roberts, Karen L, Mingardi, Anna, Mattioli, Mario, Nalin, Arnaldo, Pavone, Francesca, Spada, Simone, Trist, David G, Worby, Angela
Published in Journal of medicinal chemistry (11.12.2008)
Published in Journal of medicinal chemistry (11.12.2008)
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Discovery of Novel 1-Azoniabicyclo[2.2.2]octane Muscarinic Acetylcholine Receptor Antagonists
Lainé, Dramane I, McCleland, Brent, Thomas, Sonia, Neipp, Christopher, Underwood, Brian, Dufour, Jeremy, Widdowson, Katherine L, Palovich, Michael R, Blaney, Frank E, Foley, James J, Webb, Edward F, Luttmann, Mark A, Burman, Miriam, Belmonte, Kristen, Salmon, Michael
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
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Novel 5-HT1A/1B/1D receptors antagonists with potent 5-HT reuptake inhibitory activity
SERAFINOWSKA, Halina T, BLANEY, Frank E, LOVELL, Peter J, MERLO, Giancarlo G, SCOTT, Claire M, SMITH, Paul W, STARR, Kathryn R, WATSON, Jeannette M
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Design, Synthesis, and Structure−Activity Relationship of Tropane Muscarinic Acetylcholine Receptor Antagonists
Lainé, Dramane I, Wan, Zehong, Yan, Hongxing, Zhu, Chongjie, Xie, Haibo, Fu, Wei, Busch-Petersen, Jakob, Neipp, Christopher, Davis, Roderick, Widdowson, Katherine L, Blaney, Frank E, Foley, James, Bacon, Alicia M, Webb, Edward F, Luttmann, Mark A, Burman, Miriam, Sarau, Henry M, Salmon, Michael, Palovich, Michael R, Belmonte, Kristen
Published in Journal of medicinal chemistry (27.08.2009)
Published in Journal of medicinal chemistry (27.08.2009)
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Dihydropyrrole[2,3-d]pyridine Derivatives as Novel Corticotropin-Releasing Factor-1 Antagonists: Mapping of the Receptor Binding Pocket by in Silico Docking Studies
Di Fabio, Romano, Arban, Roberto, Bernasconi, Giovanni, Braggio, Simone, Blaney, Frank E, Capelli, Anna M, Castiglioni, Emiliano, Donati, Daniele, Fazzolari, Elettra, Ratti, Emiliangelo, Feriani, Aldo, Contini, Stefania, Gentile, Gabriella, Ghirlanda, Damiano, Sabbatini, Fabio M, Andreotti, Daniele, Spada, Simone, Marchioro, Carla, Worby, Angela, St-Denis, Yves
Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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6-Chloro-5-methyl-1-[[2-[(2-methyl-3- pyridyl)oxy]-5-pyridyl]carbamoyl]indoline (SB-242084): The First Selective and Brain Penetrant 5-HT2C Receptor Antagonist
Bromidge, Steven M, Duckworth, Malcolm, Forbes, Ian T, Ham, Peter, King, Frank D, Thewlis, Kevin M, Blaney, Frank E, Naylor, Christopher B, Blackburn, Thomas P, Kennett, Guy A, Wood, Martyn D, Clarke, Stephen E
Published in Journal of medicinal chemistry (24.10.1997)
Published in Journal of medicinal chemistry (24.10.1997)
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1,2,4-Triazol-3-yl-thiopropyl-tetrahydrobenzazepines: A Series of Potent and Selective Dopamine D3 Receptor Antagonists
Micheli, Fabrizio, Bonanomi, Giorgio, Blaney, Frank E, Braggio, Simone, Capelli, Anna Maria, Checchia, Anna, Curcuruto, Ornella, Damiani, Federica, Di Fabio, Romano, Donati, Daniele, Gentile, Gabriella, Gribble, Andy, Hamprecht, Dieter, Tedesco, Giovanna, Terreni, Silvia, Tarsi, Luca, Lightfoot, Andrew, Stemp, Geoff, MacDonald, Gregor, Smith, Alex, Pecoraro, Michela, Petrone, Marcella, Perini, Ornella, Piner, Jacqui, Rossi, Tino, Worby, Angela, Pilla, Maria, Valerio, Enzo, Griffante, Cristiana, Mugnaini, Manolo, Wood, Martyn, Scott, Claire, Andreoli, Michela, Lacroix, Laurent, Schwarz, Adam, Gozzi, Alessandro, Bifone, Angelo, Ashby, Charles R, Hagan, Jim J, Heidbreder, Christian
Published in Journal of medicinal chemistry (18.10.2007)
Published in Journal of medicinal chemistry (18.10.2007)
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Modeling the pore structure of voltage-gated sodium channels in closed, open, and fast-inactivated conformation reveals details of site 1 toxin and local anesthetic binding
Scheib, Holger, McLay, Iain, Guex, Nicolas, Clare, Jeff J, Blaney, Frank E, Dale, Tim J, Tate, Simon N, Robertson, Graeme M
Published in Journal of molecular modeling (01.09.2006)
Published in Journal of molecular modeling (01.09.2006)
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