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Published in Journal of molecular liquids (01.12.2022)
Published in Journal of molecular liquids (01.12.2022)
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Published in New journal of chemistry (2018)
Published in New journal of chemistry (2018)
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Synthesis of new lophine-carbohydrate hybrids as cholinesterase inhibitors: cytotoxicity evaluation and molecular modeling
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Published in MedChemComm (01.12.2019)
Published in MedChemComm (01.12.2019)
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Design, synthesis, cholinesterase inhibition and molecular modelling study of novel tacrine hybrids with carbohydrate derivatives
Lopes, João Paulo Bizarro, Silva, Luana, da Costa Franarin, Gabriela, Antonio Ceschi, Marco, Seibert Lüdtke, Diogo, Ferreira Dantas, Rafael, de Salles, Cristiane Martins Cardoso, Paes Silva-Jr, Floriano, Roberto Senger, Mario, Alvim Guedes, Isabella, Emmanuel Dardenne, Laurent
Published in Bioorganic & medicinal chemistry (01.11.2018)
Published in Bioorganic & medicinal chemistry (01.11.2018)
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Journal Article
Synthesis of tacrine-lophine hybrids via one-pot four component reaction and biological evaluation as acetyl- and butyrylcholinesterase inhibitors
da Costa, Jesse Sobieski, Bizarro Lopes, Joao Paulo, Russowsky, Dennis, Petzhold, Cesar Liberato, de Amorim Borges, Antonio Cesar, Ceschi, Marco Antonio, Konrath, Eduardo, Batassini, Cristiane, Lunardi, Paula Santana, Saraiva Goncalves, Carlos Alberto
Published in European journal of medicinal chemistry (01.04.2013)
Published in European journal of medicinal chemistry (01.04.2013)
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Journal Article
Tacrine-pyrimidine photoactive molecular hybrids: Synthesis, photophysics, docking and BSA interaction study
Lopes, João Paulo Bizarro, Câmara, Viktor Saraiva, Russowsky, Dennis, Nogara, Pablo Andrei, da Rocha, João Batista Teixeira, da Silveira Santos, Fabiano, Rodembusch, Fabiano Severo, Ceschi, Marco Antonio
Published in Journal of molecular liquids (01.08.2019)
Published in Journal of molecular liquids (01.08.2019)
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Journal Article
Novel series of tacrine-tianeptine hybrids: Synthesis, cholinesterase inhibitory activity, S10013 secretion and a molecular modeling approach
Ceschi, Marco Antonio, da Costa, Jessie Sobieski, Bizarro Lopes, Joao Paulo, Camara, Viktor Saraiva, Campo, Leandra Franciscato, de Amorim Borges, Antonio Cesar, Saraiva Goncalves, Carlos Alberto, de Souza, Daniela Fraga, Konrath, Eduardo Luis, Martins Karl, Ana Luiza, Guedes, Isabella Alvim, Dardenne, Laurent Emmanuel
Published in European journal of medicinal chemistry (04.10.2016)
Published in European journal of medicinal chemistry (04.10.2016)
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Journal Article
Novel series of tacrine-tianeptine hybrids: Synthesis, cholinesterase inhibitory activity, S100B secretion and a molecular modeling approach
Ceschi, Marco Antonio, da Costa, Jessie Sobieski, Lopes, João Paulo Bizarro, Câmara, Viktor Saraiva, Campo, Leandra Franciscato, Borges, Antonio César de Amorim, Gonçalves, Carlos Alberto Saraiva, de Souza, Daniela Fraga, Konrath, Eduardo Luis, Karl, Ana Luiza Martins, Guedes, Isabella Alvim, Dardenne, Laurent Emmanuel
Published in European journal of medicinal chemistry (04.10.2016)
Published in European journal of medicinal chemistry (04.10.2016)
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Journal Article
Lophine and pyrimidine based photoactive molecular hybrids. Synthesis, photophysics, BSA interaction and DFT studyElectronic supplementary information (ESI) available: Original spectroscopic characterisation spectra and additional photophysical study and theoretical calculations. See DOI: 10.1039/c8nj03315c
Lopes, João Paulo Bizarro, Câmara, Viktor Saraiva, Russowsky, Dennis, da Silveira Santos, Fabiano, Beal, Roiney, Nogara, Pablo Andrei, da Rocha, João Batista Teixeira, Gonçalves, Paulo Fernando Bruno, Rodembusch, Fabiano Severo, Ceschi, Marco Antônio
Year of Publication 08.10.2018
Year of Publication 08.10.2018
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Synthesis of new lophine–carbohydrate hybrids as cholinesterase inhibitors: cytotoxicity evaluation and molecular modeling† †Electronic supplementary information (ESI) available: Graphics and extra data of in vitro and in silico experiments and detailed spectroscopic characterization. See DOI: 10.1039/c9md00358d
Lopes, João Paulo Bizarro, Silva, Luana, Ceschi, Marco Antonio, Lüdtke, Diogo Seibert, Zimmer, Aline Rigon, Ruaro, Thais Carine, Dantas, Rafael Ferreira, de Salles, Cristiane Martins Cardoso, Silva-Jr, Floriano Paes, Senger, Mario Roberto, Barbosa, Gisele, Lima, Lídia Moreira, Guedes, Isabella Alvim, Dardenne, Laurent Emmanuel
Published in MedChemComm (08.11.2019)
Published in MedChemComm (08.11.2019)
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Year of Publication 13.08.2019
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molécula híbrida contendo núcleos tacrina e derivados de carboidratos, composição farmacêutica, processo de síntese e seus usos
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Year of Publication 09.07.2019
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molécula híbrida contendo núcleos tacrina e derivados de carboidratos, composição farmacêutica, processo de síntese e seus usos
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Year of Publication 04.07.2017
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processo multicomponente para síntese de compostos híbridos contendo os nùcleos tetraidroacridina e imidazol 1,2,4,5-tetrassubstituídos para fins farmacológicos e produtos
CRISTIANE BATASSINI, JESSÉ SOBIESKI DA COSTA, EDUARDO LUIS KONRATH, PAULA SANTANA LUNARDI, CARLOS ALBERTO SARAIVA GONÇALVES, JOÃO PAULO BIZARRO LOPES, ANTÔNIO CÉSAR DE AMORIM BORGES, DENNIS RUSSOWSKY, CESAR LIBERATO PETZHOLD, MARCO ANTÔNIO CESCHI
Year of Publication 12.04.2016
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Year of Publication 12.04.2016
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