In-vitro biological evaluation of 3,3',5,5'-tetramethoxy-biphenyl-4,4'-diol and molecular docking studies on trypanothione reductase and Gp63 from Leishmania amazonensis demonstrated anti-leishmania potential
Schirmann, Jéseka G, Bortoleti, Bruna T S, Gonçalves, Manoela D, Tomiotto-Pellissier, Fernanda, Camargo, Priscila G, Miranda-Sapla, Milena M, Lima, Camilo H S, Bispo, Marcelle L F, Costa, Idessania N, Conchon-Costa, Ivete, Pavanelli, Wander R, Dekker, Robert F H, Barbosa-Dekker, Aneli M
Published in Scientific reports (28.04.2023)
Published in Scientific reports (28.04.2023)
Get full text
Journal Article
Mycobacterial Targets for Thiourea Derivatives: Opportunities for Virtual Screening in Tuberculosis Drug Discovery
Milani, Vinicius de Melo, Silva, Mariana Luiza, Camargo, Priscila Goes, Bispo, Marcelle de Lima Ferreira
Published in Current medicinal chemistry (01.01.2024)
Published in Current medicinal chemistry (01.01.2024)
Get more information
Journal Article
Exploring Urease Inhibition by Coumarin Derivatives through in silico and in vitro Methods
Fabris, Marciéli, Camargo, Priscila, Silva, Mariana, Silva, Talis, Machado, Sérgio, Rodrigues, Carlos, Lima, Camilo, Albuquerque, Magaly, Bispo, Marcelle
Published in Journal of the Brazilian Chemical Society (2024)
Published in Journal of the Brazilian Chemical Society (2024)
Get full text
Journal Article
Novel Organic Salts Based on Mefloquine: Synthesis, Solubility, Permeability, and In Vitro Activity against Mycobacterium tuberculosis
Silva, Dário, Lopes, Márcio V. C., Petrovski, Željko, Santos, Miguel M., Santos, Jussevania P., Yamada-Ogatta, Sueli F., Bispo, Marcelle L. F., de Souza, Marcus V. N., Duarte, Ana Rita C., Lourenço, Maria C. S., Gonçalves, Raoni Schroeder B., Branco, Luis C.
Published in Molecules (Basel, Switzerland) (13.08.2022)
Published in Molecules (Basel, Switzerland) (13.08.2022)
Get full text
Journal Article
Benzoylthioureas: Design, Synthesis and Antimycobacterial Evaluation
Brito, Tiago O, Abreu, Lethícia O, Gomes, Karen M, Lourenço, Maria C S, Pereira, Patricia M L, Yamada-Ogatta, Sueli F, de Fátima, Ângelo, Tisher, Cesar A, Macedo, Jr, Fernando, Bispo, Marcelle L F
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2020)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2020)
Get more information
Journal Article
Molecular targets for chalcones in antileishmanial drug discovery
de Santiago-Silva, Kaio Maciel, da Silva Gomes, Gabriel Felix, Perez, Carla Cristina, da Silva Lima, Camilo Henrique, de Lima Ferreira Bispo, Marcelle
Published in Mini reviews in medicinal chemistry (01.01.2023)
Published in Mini reviews in medicinal chemistry (01.01.2023)
Get more information
Journal Article
Cyclodextrin-encapsulated new drug with promising anti-Trypanosoma cruzi activity
Zanetti, Igor, do Nascimento Oliveira, Laudicéa, de Azevedo Maia, Fernanda Lima, de Santiago-Silva, Kaio Maciel, Pereira, Patricia M. L., Albuquerque, Magaly Girão, Gonçalves, Raoni Schroeder Borges, de Lima Ferreira Bispo, Marcelle, Yamada-Ogatta, Sueli F., Magalhães, Alviclér, da Silva Lima, Camilo Henrique, Malta, Luiz Fernando Brum
Published in Journal of thermal analysis and calorimetry (01.10.2023)
Published in Journal of thermal analysis and calorimetry (01.10.2023)
Get full text
Journal Article
7-Chloro-4-quinolinyl Hydrazones: A Promising and Potent Class of Antileishmanial Compounds
Coimbra, Elaine S., Antinarelli, Luciana M. R., da Silva, Adilson D., Bispo, Marcelle L. F., Kaiser, Carlos R., de Souza, Marcus V. N.
Published in Chemical biology & drug design (01.05.2013)
Published in Chemical biology & drug design (01.05.2013)
Get full text
Journal Article
Thiohydantoins and hydantoins derived from amino acids as potent urease inhibitors: Inhibitory activity and ligand-target interactions
Camargo, Priscila Goes, Fabris, Marciéli, Nakamae, Matheus Yoshimitsu Tatsuta, de Freitas Oliveira, Breno Germano, da Silva Lima, Camilo Henrique, de Fátima, Ângelo, de Lima Ferreira Bispo, Marcelle, Macedo, Fernando
Published in Chemico-biological interactions (25.09.2022)
Published in Chemico-biological interactions (25.09.2022)
Get full text
Journal Article
In vitro evaluation of antitrypanosomal activity and molecular docking of benzoylthioureas
Pereira, Patricia M.L., Camargo, Priscila G., Fernandes, Bruna T., Flores-Junior, Luiz A.P., Dias, Luiza R.S., Lima, Camilo H.S., Pinge-Filho, Phileno, Lioni, Lucy M.Y., Yamada-Ogatta, Sueli F., Bispo, Marcelle L.F., Macedo Jr, Fernando
Published in Parasitology international (01.02.2021)
Published in Parasitology international (01.02.2021)
Get full text
Journal Article
In silico approaches and in vitro assays identify a coumarin derivative as antiviral potential against SARS-CoV-2
Felix da Silva Gomes, Gabriel, Goes Camargo, Priscila, de Santiago-Silva, Kaio Maciel, Suzukawa, Helena Tiemi, Sotero da Silva Ribeiro, Ana Paula, Orsato, Alexandre, Nakazato, Gerson, Yamada-Ogatta, Sueli Fumie, Faccin-Galhardi, Ligia Carla, da Silva Lima, Camilo Henrique, de Lima Ferreira Bispo, Marcelle, Perez, Carla Cristina
Published in Journal of biomolecular structure & dynamics (12.12.2023)
Published in Journal of biomolecular structure & dynamics (12.12.2023)
Get full text
Journal Article
Investigation of the antileishmanial activity and mechanisms of action of acetyl-thiohydantoins
Bortoleti, Bruna Taciane da Silva, Gonçalves, Manoela Daiele, Tomiotto-Pellissier, Fernanda, Camargo, Priscila Goes, Assolini, João Paulo, Concato, Virginia Marcia, Detoni, Mariana Barbosa, Bidóia, Danielle Larazin, Bispo, Marcelle de Lima Ferreira, Lima, Camilo Henrique da Silva, de Macedo, Fernando Cesar, Conchon-Costa, Ivete, Miranda-Sapla, Milena Menegazzo, Wowk, Pryscilla Fanini, Pavanelli, Wander Rogério
Published in Chemico-biological interactions (05.01.2022)
Published in Chemico-biological interactions (05.01.2022)
Get full text
Journal Article
Carvacrol and its Semi-synthetic Derivatives as Potential Antibacterial Agents
H. Castro, Isabelle, A. A. Oliveira, Fabrício, Perez, Carla C., L. F. Bispo, Marcelle
Published in Revista Virtual de Química (01.09.2023)
Published in Revista Virtual de Química (01.09.2023)
Get full text
Journal Article
Synergistic antifungal interaction of N -(butylcarbamothioyl) benzamide and amphotericin B against Cryptococcus neoformans
Andriani, Gabriella Maria, Spoladori, Lais Fernanda de Almeida, Fabris, Marciéli, Camargo, Priscila Goes, Pereira, Patrícia Morais Lopes, Santos, Jussevania Pereira, Bartolomeu-Gonçalves, Guilherme, Alonso, Lais, Lancheros, Cesar Armando Contreras, Alonso, Antonio, Nakamura, Celso Vataru, Macedo, Jr, Fernando, Pinge-Filho, Phileno, Yamauchi, Lucy Megumi, Bispo, Marcelle de Lima Ferreira, Tavares, Eliandro Reis, Yamada-Ogatta, Sueli Fumie
Published in Frontiers in microbiology (07.03.2023)
Published in Frontiers in microbiology (07.03.2023)
Get full text
Journal Article
A new and potent class of quinoline derivatives against cancer
Bispo, Marcelle de L. F., de Alcantara, Camila C., de Moraes, Manoel O., do Ó Pessoa, Cláudia, Rodrigues, Felipe A. R., Kaiser, Carlos R., Wardell, Solange M. S. V., Wardell, James L., de Souza, Marcus V. N.
Published in Monatshefte für Chemie (01.12.2015)
Published in Monatshefte für Chemie (01.12.2015)
Get full text
Journal Article