Potent and Selective Inhibition of Human Cytomegalovirus Replication by 1263W94, a Benzimidazole l-Riboside with a Unique Mode of Action
BIRON, Karen K, HARVEY, Robert J, STANAT, Sylvia C, DRACH, John C, TOWNSEND, Leroy B, KOSZALKA, George W, CHAMBERLAIN, Stanley C, GOOD, Steven S, SMITH, Albert A, DAVIS, Michelle G, TALARICO, Christine L, MILLER, Wayne H, FERRIS, Robert, DORNSIFE, Ronna E
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Published in Antimicrobial Agents and Chemotherapy (01.08.2002)
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In Vitro Activities of Benzimidazole d- and l-Ribonucleosides against Herpesviruses
WILLIAMS, Stephanie L, HARTLINE, Caroll B, KUSHNER, Nicole L, HARDEN, Emma A, BIDANSET, Deborah J, DRACH, John C, TOWNSEND, Leroy B, UNDERWOOD, Mark R, BIRON, Karen K, KERN, Earl R
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Published in Antimicrobial Agents and Chemotherapy (01.07.2003)
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The Human Cytomegalovirus UL44 Protein Is a Substrate for the UL97 Protein Kinase
Krosky, Paula M, Baek, Moon-Chang, Jahng, Wan Jin, Barrera, Imma, Harvey, Robert J, Biron, Karen K, Coen, Donald M, Sethna, Phiroze B
Published in Journal of Virology (01.07.2003)
Published in Journal of Virology (01.07.2003)
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Mutations in the Human Cytomegalovirus UL27 Gene That Confer Resistance to Maribavir
CHOU, Sunwen, MAROUSEK, Gail I, SENTERS, Anne E, DAVIS, Michelle G, BIRON, Karen K
Published in Journal of Virology (01.07.2004)
Published in Journal of Virology (01.07.2004)
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Preclinical and Toxicology Studies of 1263W94, a Potent and Selective Inhibitor of Human Cytomegalovirus Replication
KOSZALKA, George W, JOHNSON, Nelson W, GOOD, Steven S, BOYD, Leslie, CHAMBERLAIN, Stanley C, TOWNSEND, Leroy B, DRACH, John C, BIRON, Karen K
Published in Antimicrobial Agents and Chemotherapy (01.08.2002)
Published in Antimicrobial Agents and Chemotherapy (01.08.2002)
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Mechanism of Action of the Ribopyranoside Benzimidazole GW275175X against Human Cytomegalovirus
UNDERWOOD, Mark R, FERRIS, Robert G, SELLESETH, Dean W, DAVIS, Michelle G, DRACH, John C, TOWNSEND, Leroy B, BIRON, Karen K, BOYD, F. Leslie
Published in Antimicrobial Agents and Chemotherapy (01.05.2004)
Published in Antimicrobial Agents and Chemotherapy (01.05.2004)
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Activities of Benzimidazole d- and l-Ribonucleosides in Animal Models of Cytomegalovirus Infections
KERN, Earl R, HARTLINE, Caroll B, RYBAK, Rachel J, DRACH, John C, TOWNSEND, Leroy B, BIRON, Karen K, BIDANSET, Deborah J
Published in Antimicrobial Agents and Chemotherapy (01.05.2004)
Published in Antimicrobial Agents and Chemotherapy (01.05.2004)
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Interactions of 1263W94 with Other Antiviral Agents in Inhibition of Human Cytomegalovirus Replication
SELLESETH, Dean W, TALARICO, Christine L, MILLER, Teresa, LUTZ, Michael W, BIRON, Karen K, HARVEY, Robert J
Published in Antimicrobial Agents and Chemotherapy (01.04.2003)
Published in Antimicrobial Agents and Chemotherapy (01.04.2003)
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Mutations Conferring Ganciclovir Resistance in a Cohort of Patients with Acquired Immunodeficiency Syndrome and Cytomegalovirus Retinitis
Jabs, Douglas A., Martin, Barbara K., Forman, Michael S., Dunn, J. P., Davis, Janet L., Weinberg, David V., Biron, Karen K., Baldanti, Fausto
Published in The Journal of infectious diseases (15.01.2001)
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Acyclovir Is Phosphorylated by the Human Cytomegalovirus UL97 Protein
TALARICO, C. L, BURNETTE, T. C, BIRON, K. K, MILLER, W. H, SMITH, S. L, DAVIS, M. G, STANAT, S. C, NG, T. I, ZUWEN HE, COEN, D. M, ROIZMAN, B
Published in Antimicrobial Agents and Chemotherapy (01.08.1999)
Published in Antimicrobial Agents and Chemotherapy (01.08.1999)
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Phosphorylation of β-d-Ribosylbenzimidazoles Is Not Required for Activity against Human Cytomegalovirus
KROSKY, Paula M, BORYSKO, Katherine Z, REZA NASSIRI, M, DEVIVAR, Rodrigo V, PTAK, Roger G, DAVIS, Michelle G, BIRON, Karen K, TOWNSEND, Leroy B, DRACH, John C
Published in Antimicrobial Agents and Chemotherapy (01.02.2002)
Published in Antimicrobial Agents and Chemotherapy (01.02.2002)
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The Cys607→Tyr Change in the UL97 Phosphotransferase Confers Ganciclovir Resistance to Two Human Cytomegalovirus Strains Recovered from Two Immunocompromised Patients
BALDANTI, F, UNDERWOOD, M. R, TALARICO, C. L, SIMONCINI, L, SARASINI, A, BIRON, K. K, GERNA, G
Published in Antimicrobial Agents and Chemotherapy (01.02.1998)
Published in Antimicrobial Agents and Chemotherapy (01.02.1998)
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Inhibition of Human Cytomegalovirus DNA Maturation by a Benzimidazole Ribonucleoside Is Mediated through the UL89 Gene Product
Underwood, M R, Harvey, R J, Stanat, S C, Hemphill, M L, Miller, T, Drach, J C, Townsend, L B, Biron, K K
Published in Journal of Virology (01.01.1998)
Published in Journal of Virology (01.01.1998)
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Resistance of Human Cytomegalovirus to Benzimidazole Ribonucleosides Maps to Two Open Reading Frames: UL89 and UL56
Krosky, P M, Underwood, M R, Turk, S R, Feng, K W, Jain, R K, Ptak, R G, Westerman, A C, Biron, K K, Townsend, L B, Drach, J C
Published in Journal of Virology (01.06.1998)
Published in Journal of Virology (01.06.1998)
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An Enantiospecific Synthesis of the Human Cytomegalovirus Antiviral Agent [(R)-3-((2-Amino-1,6-dihydro-6-oxo-9H-purin-9-yl)methoxy)-4- hydroxybutyl]phosphonic Acid
Chamberlain, Stanley D, Biron, Karen K, Dornsife, Ronna E, Averett, Devron R, Beauchamp, Lilia, Koszalka, George W
Published in Journal of medicinal chemistry (01.04.1994)
Published in Journal of medicinal chemistry (01.04.1994)
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Inhibition of Epstein-Barr Virus Replication by a Benzimidazole l-Riboside: Novel Antiviral Mechanism of 5,6-Dichloro-2-(Isopropylamino)-1-β-l-Ribofuranosyl-1H-Benzimidazole
Zacny, V L, Gershburg, E, Davis, M G, Biron, K K, Pagano, J S
Published in Journal of Virology (01.09.1999)
Published in Journal of Virology (01.09.1999)
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Inhibition of Ganciclovir-Susceptible and -Resistant Human Cytomegalovirus Clinical Isolates by the Benzimidazole l-Riboside 1263W94
McSharry, J J, McDonough, A, Olson, B, Talarico, C, Davis, M, Biron, K K
Published in Clinical and Diagnostic Laboratory Immunology (01.11.2001)
Published in Clinical and Diagnostic Laboratory Immunology (01.11.2001)
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