Structure of hepcidin-bound ferroportin reveals iron homeostatic mechanisms
Billesbølle, Christian B, Azumaya, Caleigh M, Kretsch, Rachael C, Powers, Alexander S, Gonen, Shane, Schneider, Simon, Arvedson, Tara, Dror, Ron O, Cheng, Yifan, Manglik, Aashish
Published in Nature (London) (29.10.2020)
Published in Nature (London) (29.10.2020)
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Structural basis of odorant recognition by a human odorant receptor
Billesbølle, Christian B, de March, Claire A, van der Velden, Wijnand J C, Ma, Ning, Tewari, Jeevan, Del Torrent, Claudia Llinas, Li, Linus, Faust, Bryan, Vaidehi, Nagarajan, Matsunami, Hiroaki, Manglik, Aashish
Published in Nature (London) (23.03.2023)
Published in Nature (London) (23.03.2023)
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Autoantibody mimicry of hormone action at the thyrotropin receptor
Faust, Bryan, Billesbølle, Christian B, Suomivuori, Carl-Mikael, Singh, Isha, Zhang, Kaihua, Hoppe, Nicholas, Pinto, Antonio F M, Diedrich, Jolene K, Muftuoglu, Yagmur, Szkudlinski, Mariusz W, Saghatelian, Alan, Dror, Ron O, Cheng, Yifan, Manglik, Aashish
Published in Nature (London) (22.09.2022)
Published in Nature (London) (22.09.2022)
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Docking for EP4R antagonists active against inflammatory pain
Gahbauer, Stefan, DeLeon, Chelsea, Braz, Joao M, Craik, Veronica, Kang, Hye Jin, Wan, Xiaobo, Huang, Xi-Ping, Billesbølle, Christian B, Liu, Yongfeng, Che, Tao, Deshpande, Ishan, Jewell, Madison, Fink, Elissa A, Kondratov, Ivan S, Moroz, Yurii S, Irwin, John J, Basbaum, Allan I, Roth, Bryan L, Shoichet, Brian K
Published in Nature communications (06.12.2023)
Published in Nature communications (06.12.2023)
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Journal Article
Transition metal ion FRET uncovers K + regulation of a neurotransmitter/sodium symporter
Billesbølle, Christian B, Mortensen, Jonas S, Sohail, Azmat, Schmidt, Solveig G, Shi, Lei, Sitte, Harald H, Gether, Ulrik, Loland, Claus J
Published in Nature communications (28.09.2016)
Published in Nature communications (28.09.2016)
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Substrate-induced Unlocking of the Inner Gate Determines the Catalytic Efficiency of a Neurotransmitter:Sodium Symporter
Billesbølle, Christian B., Krüger, Mie B., Shi, Lei, Quick, Matthias, Li, Zheng, Stolzenberg, Sebastian, Kniazeff, Julie, Gotfryd, Kamil, Mortensen, Jonas S., Javitch, Jonathan A., Weinstein, Harel, Loland, Claus J., Gether, Ulrik
Published in The Journal of biological chemistry (30.10.2015)
Published in The Journal of biological chemistry (30.10.2015)
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Novel and High Affinity Fluorescent Ligands for the Serotonin Transporter Based on (S)‑Citalopram
Kumar, Vivek, Rahbek-Clemmensen, Troels, Billesbølle, Christian B, Jorgensen, Trine Nygaard, Gether, Ulrik, Newman, Amy Hauck
Published in ACS medicinal chemistry letters (12.06.2014)
Published in ACS medicinal chemistry letters (12.06.2014)
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A virtual high-throughput screening approach to the discovery of novel inhibitors of the bacterial leucine transporter, LeuT
Simmons, Katie J., Gotfryd, Kamil, Billesbølle, Christian B., Loland, Claus J., Gether, Ulrik, Fishwick, Colin W. G., Johnson, A. Peter
Published in Molecular membrane biology (01.03.2013)
Published in Molecular membrane biology (01.03.2013)
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An ultrapotent synthetic nanobody neutralizes SARS-CoV-2 by stabilizing inactive Spike
Schoof, Michael, Faust, Bryan, Saunders, Reuben A, Sangwan, Smriti, Rezelj, Veronica, Hoppe, Nick, Boone, Morgane, Billesbølle, Christian B, Puchades, Cristina, Azumaya, Caleigh M, Kratochvil, Huong T, Zimanyi, Marcell, Deshpande, Ishan, Liang, Jiahao, Dickinson, Sasha, Nguyen, Henry C, Chio, Cynthia M, Merz, Gregory E, Thompson, Michael C, Diwanji, Devan, Schaefer, Kaitlin, Anand, Aditya A, Dobzinski, Niv, Zha, Beth Shoshana, Simoneau, Camille R, Leon, Kristoffer, White, Kris M, Chio, Un Seng, Gupta, Meghna, Jin, Mingliang, Li, Fei, Liu, Yanxin, Zhang, Kaihua, Bulkley, David, Sun, Ming, Smith, Amber M, Rizo, Alexandrea N, Moss, Frank, Brilot, Axel F, Pourmal, Sergei, Trenker, Raphael, Pospiech, Thomas, Gupta, Sayan, Barsi-Rhyne, Benjamin, Belyy, Vladislav, Barile-Hill, Andrew W, Nock, Silke, Liu, Yuwei, Krogan, Nevan J, Ralston, Corie Y, Swaney, Danielle L, García-Sastre, Adolfo, Ott, Melanie, Vignuzzi, Marco, Walter, Peter, Manglik, Aashish
Published in Science (18.12.2020)
Published in Science (18.12.2020)
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An ultra-potent synthetic nanobody neutralizes SARS-CoV-2 by locking Spike into an inactive conformation
Schoof, Michael, Faust, Bryan, Saunders, Reuben A, Sangwan, Smriti, Rezelj, Veronica, Hoppe, Nick, Boone, Morgane, Billesbølle, Christian B, Puchades, Cristina, Azumaya, Caleigh M, Kratochvil, Huong T, Zimanyi, Marcell, Deshpande, Ishan, Liang, Jiahao, Dickinson, Sasha, Nguyen, Henry C, Chio, Cynthia M, Merz, Gregory E, Thompson, Michael C, Diwanji, Devan, Schaefer, Kaitlin, Anand, Aditya A, Dobzinski, Niv, Zha, Beth Shoshana, Simoneau, Camille R, Leon, Kristoffer, White, Kris M, Chio, Un Seng, Gupta, Meghna, Jin, Mingliang, Li, Fei, Liu, Yanxin, Zhang, Kaihua, Bulkley, David, Sun, Ming, Smith, Amber M, Rizo, Alexandrea N, Moss, Frank, Brilot, Axel F, Pourmal, Sergei, Trenker, Raphael, Pospiech, Thomas, Gupta, Sayan, Barsi-Rhyne, Benjamin, Belyy, Vladislav, Barile-Hill, Andrew W, Nock, Silke, Liu, Yuwei, Krogan, Nevan J, Ralston, Corie Y, Swaney, Danielle L, García-Sastre, Adolfo, Ott, Melanie, Vignuzzi, Marco, Walter, Peter, Manglik, Aashish
Published in bioRxiv : the preprint server for biology (17.08.2020)
Published in bioRxiv : the preprint server for biology (17.08.2020)
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Engineered odorant receptors illuminate structural principles of odor discrimination
De March, Claire A, Ma, Ning, Billesboelle, Christian B, Tewari, Jeevan, Claudia Llinas Del Torrent, Winjand Jc Van Der Velden, Ojiro, Ichie, Takayama, Ikumi, Faust, Bryan, Li, Linus, Nagarajan Vaidehi, Manglik, Aashish, Matsunami, Hiroaki
Published in bioRxiv (17.11.2023)
Published in bioRxiv (17.11.2023)
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CryoEM and AI reveal a structure of SARS-CoV-2 Nsp2, a multifunctional protein involved in key host processes
Gupta, Meghna, Azumaya, Caleigh M, Moritz, Michelle, Pourmal, Sergei, Diallo, Amy, Merz, Gregory E, Jang, Gwendolyn, Bouhaddou, Mehdi, Fossati, Andrea, Brilot, Axel F, Diwanji, Devan, Hernandez, Evelyn, Herrera, Nadia, Kratochvil, Huong T, Lam, Victor L, Li, Fei, Li, Yang, Nguyen, Henry C, Nowotny, Carlos, Owens, Tristan W, Peters, Jessica K, Rizo, Alexandrea N, Schulze-Gahmen, Ursula, Smith, Amber M, Young, Iris D, Yu, Zanlin, Asarnow, Daniel, Billesbølle, Christian, Campbell, Melody G, Chen, Jen, Chen, Kuei-Ho, Chio, Un Seng, Dickinson, Miles Sasha, Doan, Loan, Jin, Mingliang, Kim, Kate, Li, Junrui, Li, Yen-Li, Linossi, Edmond, Liu, Yanxin, Lo, Megan, Lopez, Jocelyne, Lopez, Kyle E, Mancino, Adamo, Moss, 3rd, Frank R, Paul, Michael D, Pawar, Komal Ishwar, Pelin, Adrian, Pospiech, Jr, Thomas H, Puchades, Cristina, Remesh, Soumya Govinda, Safari, Maliheh, Schaefer, Kaitlin, Sun, Ming, Tabios, Mariano C, Thwin, Aye C, Titus, Erron W, Trenker, Raphael, Tse, Eric, Tsui, Tsz Kin Martin, Wang, Feng, Zhang, Kaihua, Zhang, Yang, Zhao, Jianhua, Zhou, Fengbo, Zhou, Yuan, Zuliani-Alvarez, Lorena, Agard, David A, Cheng, Yifan, Fraser, James S, Jura, Natalia, Kortemme, Tanja, Manglik, Aashish, Southworth, Daniel R, Stroud, Robert M, Swaney, Danielle L, Krogan, Nevan J, Frost, Adam, Rosenberg, Oren S, Verba, Kliment A
Published in Research square (19.05.2021)
Published in Research square (19.05.2021)
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CryoEM and AI reveal a structure of SARS-CoV-2 Nsp2, a multifunctional protein involved in key host processes
Gupta, Meghna, Azumaya, Caleigh M, Moritz, Michelle, Pourmal, Sergei, Diallo, Amy, Merz, Gregory E, Jang, Gwendolyn, Bouhaddou, Mehdi, Fossati, Andrea, Brilot, Axel F, Diwanji, Devan, Hernandez, Evelyn, Herrera, Nadia, Kratochvil, Huong T, Lam, Victor L, Li, Fei, Li, Yang, Nguyen, Henry C, Nowotny, Carlos, Owens, Tristan W, Peters, Jessica K, Rizo, Alexandrea N, Schulze-Gahmen, Ursula, Smith, Amber M, Young, Iris D, Yu, Zanlin, Asarnow, Daniel, Billesbølle, Christian, Campbell, Melody G, Chen, Jen, Chen, Kuei-Ho, Chio, Un Seng, Dickinson, Miles Sasha, Doan, Loan, Jin, Mingliang, Kim, Kate, Li, Junrui, Li, Yen-Li, Linossi, Edmond, Liu, Yanxin, Lo, Megan, Lopez, Jocelyne, Lopez, Kyle E, Mancino, Adamo, Moss, 3rd, Frank R, Paul, Michael D, Pawar, Komal Ishwar, Pelin, Adrian, Pospiech, Jr, Thomas H, Puchades, Cristina, Remesh, Soumya Govinda, Safari, Maliheh, Schaefer, Kaitlin, Sun, Ming, Tabios, Mariano C, Thwin, Aye C, Titus, Erron W, Trenker, Raphael, Tse, Eric, Tsui, Tsz Kin Martin, Wang, Feng, Zhang, Kaihua, Zhang, Yang, Zhao, Jianhua, Zhou, Fengbo, Zhou, Yuan, Zuliani-Alvarez, Lorena, Agard, David A, Cheng, Yifan, Fraser, James S, Jura, Natalia, Kortemme, Tanja, Manglik, Aashish, Southworth, Daniel R, Stroud, Robert M, Swaney, Danielle L, Krogan, Nevan J, Frost, Adam, Rosenberg, Oren S, Verba, Kliment A
Published in bioRxiv : the preprint server for biology (11.05.2021)
Published in bioRxiv : the preprint server for biology (11.05.2021)
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Journal Article
Structural basis of odorant recognition by a human odorant receptor
Billesboelle, Christian B, De March, Claire A, Wijnand Jc Van Der Velden, Ma, Ning, Tewari, Jeevan, Claudia Linas Del Torrent, Li, Linus, Faust, Bryan, Nagarajan Vaidehi, Matsunami, Hiroaki, Manglik, Aashish
Published in bioRxiv (20.12.2022)
Published in bioRxiv (20.12.2022)
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