2‑(3-Fluoro-4-methylsulfonylaminophenyl)propanamides as Potent Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists: Structure–Activity Relationships of 2‑Amino Derivatives in the N‑(6-Trifluoromethylpyridin-3-ylmethyl) C‑Region
Kim, Myeong Seop, Ryu, HyungChul, Kang, Dong Wook, Cho, Seong-Hee, Seo, Sejin, Park, Young Soo, Kim, Mi-Yeon, Kwak, Eun Joo, Kim, Yong Soo, Bhondwe, Rahul S, Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, DeAndrea-Lazarus, Ian A, Pearce, Larry V, Blumberg, Peter M, Frank, Robert, Bahrenberg, Gregor, Stockhausen, Hannelore, Kögel, Babette Y, Schiene, Klaus, Christoph, Thomas, Lee, Jeewoo
Published in Journal of medicinal chemistry (11.10.2012)
Published in Journal of medicinal chemistry (11.10.2012)
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Journal Article
Structure–activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-N′-[4-(methylsulfonylamino)benzyl] thiourea template for TRPV1 antagonism
Bhondwe, Rahul S., Kang, Dong Wook, Kim, Myeong Seop, Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, Lang Kuhs, Krystle A., Pavlyukovets, Vladimir A., Pearce, Larry V., Blumberg, Peter M., Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
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Journal Article
N-4-t-Butylbenzyl 2-(4-methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the A-region
Kim, Yong Soo, Kil, Min-Jung, Kang, Sang-Uk, Ryu, HyungChul, Kim, Myeong Seop, Cho, Yongsung, Bhondwe, Rahul S., Thorat, Shivaji A., Sun, Wei, Liu, Keliang, Lee, Jin Hee, Choi, Sun, Pearce, Larry V., Pavlyukovets, Vladimir A., Morgan, Matthew A., Tran, Richard, Lazar, Jozsef, Blumberg, Peter M., Lee, Jeewoo
Published in Bioorganic & medicinal chemistry (01.01.2012)
Published in Bioorganic & medicinal chemistry (01.01.2012)
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Journal Article
2-(4-Methylsulfonylaminophenyl) propanamide TRPV1 antagonists: Structure–activity relationships in the B and C-regions
Sun, Wei, Liu, Keliang, Ryu, HyungChul, Kang, Dong Wook, Kim, Yong Soo, Kim, Myeong Seop, Cho, Yongsung, Bhondwe, Rahul S., Thorat, Shivaji A., Kim, Ho Shin, Pearce, Larry V., Pavlyukovets, Vladimir A., Tran, Richard, Morgan, Matthew A., Lazar, Jozsef, Ryder, Christopher B., Toth, Attila, Blumberg, Peter M., Lee, Jeewoo
Published in Bioorganic & medicinal chemistry (01.02.2012)
Published in Bioorganic & medicinal chemistry (01.02.2012)
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Journal Article
Structure-activity relationships and molecular modeling of the N-(3-pivaloyloxy-2-benzylpropyl)-Na2-[4-(methylsulfonylamino)benzy l] thiourea template for TRPV1 antagonism
Bhondwe, Rahul S, Kang, Dong Wook, Kim, Myeong Seop, Kim, Ho Shin, Park, Seul-gi, Son, Karam, Choi, Sun, Lang Kuhs, Krystle A, Pavlyukovets, Vladimir A, Pearce, Larry V, Blumberg, Peter M, Lee, Jeewoo
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
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Journal Article