Discovery of imidazo[1,2-a]pyridine-thiophene derivatives as FLT3 and FLT3 mutants inhibitors for acute myeloid leukemia through structure-based optimization of an NEK2 inhibitor
Zhang, Lingtian, Lakkaniga, Naga Rajiv, Bharate, Jaideep B., Mcconnell, Nicholas, Wang, Xiuqi, Kharbanda, Anupreet, Leung, Yuet-Kin, Frett, Brendan, Shah, Neil P., Li, Hong-yu
Published in European journal of medicinal chemistry (05.12.2021)
Published in European journal of medicinal chemistry (05.12.2021)
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Journal Article
Tandem Ring Opening/Intramolecular [2 + 2] Cycloaddition Reaction for the Synthesis of Cyclobutane Fused Thiazolino-2-Pyridones
Tyagi, Mohit, Adolfsson, Dan E, Singh, Pardeep, Ådén, Jörgen, Jayaweera, Sanduni Wasana, Gharibyan, Anna, Bharate, Jaideep B, Kiss, Anita, Sarkar, Souvik, Olofsson, Anders, Almqvist, Fredrik
Published in Journal of organic chemistry (03.12.2021)
Published in Journal of organic chemistry (03.12.2021)
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Journal Article
Discovery of N‑Trisubstituted Pyrimidine Derivatives as Type I RET and RET Gatekeeper Mutant Inhibitors with a Novel Kinase Binding Pose
Zhang, Lingtian, Moccia, Marialuisa, Briggs, David C, Bharate, Jaideep B, Lakkaniga, Naga Rajiv, Knowles, Phillip, Yan, Wei, Tran, Phuc, Kharbanda, Anupreet, Wang, Xiuqi, Leung, Yuet-Kin, Frett, Brendan, Santoro, Massimo, McDonald, Neil Q, Carlomagno, Francesca, Li, Hong-yu
Published in Journal of medicinal chemistry (27.01.2022)
Published in Journal of medicinal chemistry (27.01.2022)
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Journal Article
K2S2O8-mediated coupling of 6-amino-7-aminomethyl-thiazolino-pyridones with aldehydes to construct amyloid affecting pyrimidine-fused thiazolino-2-pyridones
Bharate, Jaideep B., Aden, Jorgen, Gharibyan, Anna, Adolfsson, Dan E., Jayaweera, Sanduni Wasana, Singh, Pardeep, Vielfort, Katarina, Tyagi, Mohit, Bonde, Mari, Bergstrom, Sven, Olofsson, Anders, Almqvist, Fredrik
Published in Organic & biomolecular chemistry (18.11.2021)
Published in Organic & biomolecular chemistry (18.11.2021)
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Journal Article
K 2 S 2 O 8 -mediated coupling of 6-amino-7-aminomethyl-thiazolino-pyridones with aldehydes to construct amyloid affecting pyrimidine-fused thiazolino-2-pyridones
Bharate, Jaideep B, Ådén, Jörgen, Gharibyan, Anna, Adolfsson, Dan E, Jayaweera, Sanduni Wasana, Singh, Pardeep, Vielfort, Katarina, Tyagi, Mohit, Bonde, Mari, Bergström, Sven, Olofsson, Anders, Almqvist, Fredrik
Published in Organic & biomolecular chemistry (18.11.2021)
Published in Organic & biomolecular chemistry (18.11.2021)
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Journal Article
Discovery of 3,3′-diindolylmethanes as potent antileishmanial agents
Bharate, Sandip B., Bharate, Jaideep B., Khan, Shabana I., Tekwani, Babu L., Jacob, Melissa R., Mudududdla, Ramesh, Yadav, Rammohan R., Singh, Baljinder, Sharma, P.R., Maity, Sudip, Singh, Baldev, Khan, Ikhlas A., Vishwakarma, Ram A.
Published in European journal of medicinal chemistry (01.05.2013)
Published in European journal of medicinal chemistry (01.05.2013)
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Journal Article
Metal-Free, Ionic Liquid-Mediated Synthesis of Functionalized Quinolines
Bharate, Jaideep B, Bharate, Sandip B, Vishwakarma, Ram A
Published in ACS combinatorial science (10.11.2014)
Published in ACS combinatorial science (10.11.2014)
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Journal Article
Cobalt(II) catalyzed C(sp)-H bond functionalization of alkynes with phenyl hydrazines: facile access to diaryl 1,2-diketones
Bharate, Jaideep B., Abbat, Sheenu, Sharma, Rohit, Bharatam, Prasad V., Vishwakarma, Ram A., Bharate, Sandip B.
Published in Organic & biomolecular chemistry (14.05.2015)
Published in Organic & biomolecular chemistry (14.05.2015)
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Journal Article
Rational Design, Synthesis and Biological Evaluation of Pyrimidine-4,6-diamine derivatives as Type-II inhibitors of FLT3 Selective Against c-KIT
Bharate, Jaideep B., McConnell, Nicholas, Naresh, Gunaganti, Zhang, Lingtian, Lakkaniga, Naga Rajiv, Ding, Lucky, Shah, Neil P., Frett, Brendan, Li, Hong-yu
Published in Scientific reports (27.02.2018)
Published in Scientific reports (27.02.2018)
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Journal Article
CuBr catalyzed aerobic oxidative coupling of 2-aminopyridines with cinnamaldehydes: direct access to 3-formyl-2-phenyl-imidazo[1,2-a]pyridines
Bharate, Jaideep B., Abbat, Sheenu, Bharatam, Prasad V., Vishwakarma, Ram A., Bharate, Sandip B.
Published in Organic & biomolecular chemistry (28.07.2015)
Published in Organic & biomolecular chemistry (28.07.2015)
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Journal Article
Discovery of 4-acetyl-3-(4-fluorophenyl)-1-(p-tolyl)-5-methylpyrrole as a dual inhibitor of human P-glycoprotein and Staphylococcus aureus Nor A efflux pump
Bharate, Jaideep B, Singh, Samsher, Wani, Abubakar, Sharma, Sadhana, Joshi, Prashant, Khan, Inshad A, Kumar, Ajay, Vishwakarma, Ram A, Bharate, Sandip B
Published in Organic & biomolecular chemistry (21.05.2015)
Published in Organic & biomolecular chemistry (21.05.2015)
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Journal Article
Synthesis, and the antioxidant, neuroprotective and P-glycoprotein induction activity of 4-arylquinoline-2-carboxylates
Bharate, Jaideep B., Wani, Abubakar, Sharma, Sadhana, Reja, Shahi Imam, Kumar, Manoj, Vishwakarma, Ram A., Kumar, Ajay, Bharate, Sandip B.
Published in Organic & biomolecular chemistry (28.08.2014)
Published in Organic & biomolecular chemistry (28.08.2014)
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Journal Article
Synthesis and P-glycoprotein induction activity of colupulone analogs
Bharate, Jaideep B., Batarseh, Yazan S., Wani, Abubakar, Sharma, Sadhana, Vishwakarma, Ram A., Kaddoumi, Amal, Kumar, Ajay, Bharate, Sandip B.
Published in Organic & biomolecular chemistry (21.05.2015)
Published in Organic & biomolecular chemistry (21.05.2015)
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Journal Article
Tandem one-pot synthesis of flavans by recyclable silica-HClO4 catalyzed Knoevenagel condensation and [4+2]-Diels-Alder cycloaddition
Bharate, Sandip B., Mudududdla, Ramesh, Bharate, Jaideep B., Battini, Narsaiah, Battula, Satyanarayana, Yadav, Rammohan R., Singh, Baldev, Vishwakarma, Ram A.
Published in Organic & biomolecular chemistry (01.01.2012)
Published in Organic & biomolecular chemistry (01.01.2012)
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Journal Article
ortho-Amidoalkylation of Phenols via Tandem One-Pot Approach Involving Oxazine Intermediate
Mudududdla, Ramesh, Jain, Shreyans K, Bharate, Jaideep B, Gupta, Ajai P, Singh, Baldev, Vishwakarma, Ram A, Bharate, Sandip B
Published in Journal of organic chemistry (05.10.2012)
Published in Journal of organic chemistry (05.10.2012)
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Journal Article
Montmorillonite clay catalyzed synthesis of functionalized pyrroles through domino four-component coupling of amines, aldehydes, 1,3-dicarbonyl compounds and nitroalkanes
Bharate, Jaideep B., Sharma, Rajni, Aravinda, Subrayashastry, Gupta, Vivek K., Singh, Baldev, Bharate, Sandip B., Vishwakarma, Ram A.
Published in RSC advances (01.01.2013)
Published in RSC advances (01.01.2013)
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Journal Article
Deformylation of indole and azaindole-3-carboxaldehydes using anthranilamide and solid acid heterogeneous catalyst via quinazolinone intermediate
Yadav, Rammohan R., Battini, Narsaiah, Mudududdla, Ramesh, Bharate, Jaideep B., Muparappu, Nagaraju, Bharate, Sandip B., Vishwakarma, Ram A.
Published in Tetrahedron letters (25.04.2012)
Published in Tetrahedron letters (25.04.2012)
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Journal Article
KF/alumina catalyzed regioselective benzylation and benzoylation using solvent-free grind-stone chemistry
Jain, Shreyans K., Meena, Samdarshi, Singh, Baljinder, Bharate, Jaideep B., Joshi, Prashant, Singh, Varun P., Vishwakarma, Ram A., Bharate, Sandip B.
Published in RSC advances (01.01.2012)
Published in RSC advances (01.01.2012)
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Journal Article
Cu–Mn spinel oxide catalyzed synthesis of imidazo[1,2-a]pyridines through domino three-component coupling and 5-exo-dig cyclization in water
Bharate, Jaideep B., Guru, Santosh K., Jain, Shreyans K., Meena, Samdarshi, Singh, Parvinder Pal, Bhushan, Shashi, Singh, Baldev, Bharate, Sandip B., Vishwakarma, Ram A.
Published in RSC advances (01.01.2013)
Published in RSC advances (01.01.2013)
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Journal Article