A Dual-Site Inhibitor of CBP/p300 KIX is a Selective and Effective Modulator of Myb
Joy, Stephen T., Henley, Madeleine J., De Salle, Samantha N., Beyersdorf, Matthew S., Vock, Isaac W., Huldin, Allison J. L., Mapp, Anna K.
Published in Journal of the American Chemical Society (22.09.2021)
Published in Journal of the American Chemical Society (22.09.2021)
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Assembly States of FliM and FliG within the Flagellar Switch Complex
Sircar, Ria, Borbat, Peter P., Lynch, Michael J., Bhatnagar, Jaya, Beyersdorf, Matthew S., Halkides, Christopher J., Freed, Jack H., Crane, Brian R.
Published in Journal of molecular biology (27.02.2015)
Published in Journal of molecular biology (27.02.2015)
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A Lipopeptidomimetic of Transcriptional Activation Domains Selectively Disrupts the Coactivator Med25 Protein–Protein Interactions
Pattelli, Olivia N., Valdivia, Estefanía Martínez, Beyersdorf, Matthew S., Regan, Clint S., Rivas, Mónica, Hebert, Katherine A., Merajver, Sofia D., Cierpicki, Tomasz, Mapp, Anna K.
Published in Angewandte Chemie International Edition (21.05.2024)
Published in Angewandte Chemie International Edition (21.05.2024)
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Garcinolic Acid Distinguishes Between GACKIX Domains and Modulates Interaction Networks
Breen, Meghan E, Joy, Stephen T, Baruti, Omari J, Beyersdorf, Matthew S, Henley, Madeleine J, De Salle, Samantha N, Ycas, Peter D, Croskey, Ayza, Cierpicki, Tomasz, Pomerantz, William C K, Mapp, Anna K
Published in Chembiochem : a European journal of chemical biology (02.11.2023)
Published in Chembiochem : a European journal of chemical biology (02.11.2023)
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Conservation of coactivator engagement mechanism enables small-molecule allosteric modulators
Henderson, Andrew R., Henley, Matthew J., Foster, Nicholas J., Peiffer, Amanda L., Beyersdorf, Matthew S., Stanford, Kevon D., Sturlis, Steven M., Linhares, Brian M., Hill, Zachary B., Wells, James A., Cierpicki, Tomasz, Brooks, Charles L., Fierke, Carol A., Mapp, Anna K.
Published in Proceedings of the National Academy of Sciences - PNAS (04.09.2018)
Published in Proceedings of the National Academy of Sciences - PNAS (04.09.2018)
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Production, characterization, and assessment of a stable analog of the response regulator CheY‐phosphate from Thermotoga maritima
Beyersdorf, Matthew S., Sircar, Ria, Lookadoo, Daniel B., Bottone, Cory J., Lynch, Michael J., Crane, Brian R., Halkides, Christopher J.
Published in Protein science (01.08.2017)
Published in Protein science (01.08.2017)
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A Lipopeptidomimetic of Transcriptional Activation Domains Selectively Disrupts the Coactivator Med25 Protein–Protein Interactions
Pattelli, Olivia N., Valdivia, Estefanía Martínez, Beyersdorf, Matthew S., Regan, Clint S., Rivas, Mónica, Hebert, Katherine A., Merajver, Sofia D., Cierpicki, Tomasz, Mapp, Anna K.
Published in Angewandte Chemie (21.05.2024)
Published in Angewandte Chemie (21.05.2024)
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A lipopeptidomimetic of transcriptional activation domains selectively disrupts Med25 PPIs
Pattelli, Olivia N, Valdivia, Estefanía Martínez, Beyersdorf, Matthew S, Regan, Clint S, Rivas, Mónica, Merajver, Sofia D, Cierpicki, Tomasz, Mapp, Anna K
Published in bioRxiv (25.03.2023)
Published in bioRxiv (25.03.2023)
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