Review of poly (ADP-ribose) polymerase (PARP) mechanisms of action and rationale for targeting in cancer and other diseases
Morales, Julio, Li, Longshan, Fattah, Farjana J, Dong, Ying, Bey, Erik A, Patel, Malina, Gao, Jinming, Boothman, David A
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Huang, Xiumei, Motea, Edward A., Moore, Zachary R., Yao, Jun, Dong, Ying, Chakrabarti, Gaurab, Kilgore, Jessica A., Silvers, Molly A., Patidar, Praveen L., Cholka, Agnieszka, Fattah, Farjana, Cha, Yoonjeong, Anderson, Glenda G., Kusko, Rebecca, Peyton, Michael, Yan, Jingsheng, Xie, Xian-Jin, Sarode, Venetia, Williams, Noelle S., Minna, John D., Beg, Muhammad, Gerber, David E., Bey, Erik A., Boothman, David A.
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Depleting Tumor-NQO1 Potentiates Anoikis and Inhibits Growth of NSCLC
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Published in Molecular cancer research (01.01.2016)
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NQO1- and PARP-1-mediated cell death pathway induced in non-small-cell lung cancer cells by β-lapachone
Bey, Erik A, Bentle, Melissa S, Reinicke, Kathryn E, Dong, Ying, Yang, Chin-Rang, Girard, Luc, Minna, John D, Bornmann, William G, Gao, Jinming, Boothman, David A
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Published in Proceedings of the National Academy of Sciences - PNAS (10.07.2007)
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NQO1-dependent, Tumor-selective Radiosensitization of Non-small Cell Lung Cancers
Motea, Edward A, Huang, Xiumei, Singh, Naveen, Kilgore, Jessica A, Williams, Noelle S, Xie, Xian-Jin, Gerber, David E, Beg, Muhammad S, Bey, Erik A, Boothman, David A
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Dual Phosphoinositide 3-Kinase/Mammalian Target of Rapamycin Blockade Is an Effective Radiosensitizing Strategy for the Treatment of Non―Small Cell Lung Cancer Harboring K-RAS Mutations
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Published in Cancer research (Chicago, Ill.) (01.10.2009)
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Y Chromosome LncRNA Are Involved in Radiation Response of Male Non-Small Cell Lung Cancer Cells
Brownmiller, Tayvia, Juric, Jamie A, Ivey, Abby D, Harvey, Brandon M, Westemeier, Emily S, Winters, Michael T, Stevens, Alyson M, Stanley, Alana N, Hayes, Karen E, Sprowls, Samuel A, Ammer, Amanda S Gatesman, Walker, Mackenzee, Bey, Erik A, Wu, Xiaoliang, Lim, Zuan-Fu, Zhu, Lin, Wen, Sijin, Hu, Gangqing, Ma, Patrick C, Martinez, Ivan
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An NQO1 Substrate with Potent Antitumor Activity That Selectively Kills by PARP1-Induced Programmed Necrosis
XIUMEI HUANG, YING DONG, JINMING GAO, HERGENROTHER, Paul J, BOOTHMAN, David A, BEY, Erik A, KILGORE, Jessica A, BAIR, Joseph S, LI, Long-Shan, PATES, Malina, PARKINSON, Elizabeth I, YIGUANG WANG, WILLIAMS, Noelle S
Published in Cancer research (Chicago, Ill.) (15.06.2012)
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Prostate Cancer Radiosensitization through Poly(ADP-Ribose) Polymerase-1 Hyperactivation
YING DONG, BEY, Erik A, LI, Long-Shan, KABBANI, Wareef, JINGSHENG YAN, XIE, Xian-Jin, HSIEH, Jer-Tsong, JINMING GAO, BOOTHMAN, David A
Published in Cancer research (Chicago, Ill.) (15.10.2010)
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Catalase abrogates β-lapachone-induced PARP1 hyperactivation-directed programmed necrosis in NQO1-positive breast cancers
Bey, Erik A, Reinicke, Kathryn E, Srougi, Melissa C, Varnes, Marie, Anderson, Vernon E, Pink, John J, Li, Long Shan, Patel, Malina, Cao, Lifen, Moore, Zachary, Rommel, Amy, Boatman, Michael, Lewis, Cheryl, Euhus, David M, Bornmann, William G, Buchsbaum, Donald J, Spitz, Douglas R, Gao, Jinming, Boothman, David A
Published in Molecular cancer therapeutics (01.10.2013)
Published in Molecular cancer therapeutics (01.10.2013)
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β-Lapachone Micellar Nanotherapeutics for Non-Small Cell Lung Cancer Therapy
BLANCO, Elvin, BEY, Erik A, JINMING GAO, KHEMTONG, Chalermchai, YANG, Su-Geun, SETTI-GUTHI, Jagadeesh, HUABING CHEN, KESSINGER, Chase W, CARNEVALE, Kevin A, BORNMANN, William G, BOOTHMAN, David A
Published in Cancer research (Chicago, Ill.) (15.05.2010)
Published in Cancer research (Chicago, Ill.) (15.05.2010)
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β-Lapachone-containing PEG–PLA polymer micelles as novel nanotherapeutics against NQO1-overexpressing tumor cells
Blanco, Elvin, Bey, Erik A., Dong, Ying, Weinberg, Brent D., Sutton, Damon M., Boothman, David A., Gao, Jinming
Published in Journal of controlled release (08.10.2007)
Published in Journal of controlled release (08.10.2007)
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Conference Proceeding
Targeting Base Excision Repair in Cancer: NQO1-Bioactivatable Drugs Improve Tumor Selectivity and Reduce Treatment Toxicity Through Radiosensitization of Human Cancer
Starcher, Colton L., Pay, S. Louise, Singh, Naveen, Yeh, I-Ju, Bhandare, Snehal B., Su, Xiaolin, Huang, Xiumei, Bey, Erik A., Motea, Edward A., Boothman, David A.
Published in Frontiers in oncology (19.08.2020)
Published in Frontiers in oncology (19.08.2020)
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Single-Cell Kinetic Modeling of β-Lapachone Metabolism in Head and Neck Squamous Cell Carcinoma
Raddatz, Andrew D, Furdui, Cristina M, Bey, Erik A, Kemp, Melissa L
Published in Antioxidants (01.03.2023)
Published in Antioxidants (01.03.2023)
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Modulating Endogenous NQO1 Levels Identifies Key Regulatory Mechanisms of Action of β-Lapachone for Pancreatic Cancer Therapy
LONG SHAN LI, BEY, Erik A, JINMING GAO, BOOTHMAN, David A, YING DONG, JIERU MENG, PATRA, Biswanath, JINGSHENG YAN, XIE, Xian-Jin, BREKKEN, Rolf A, BARNETT, Carlton C, BORNMANN, William G
Published in Clinical cancer research (15.01.2011)
Published in Clinical cancer research (15.01.2011)
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Intratumoral Delivery of β-Lapachone via Polymer Implants for Prostate Cancer Therapy
Dong, Ying, Chin, Shook-Fong, Blanco, Elvin, Bey, Erik A, Kabbani, Wareef, Xie, Xian-Jin, Bornmann, William G, Boothman, David A, Gao, Jinming
Published in Clinical cancer research (01.01.2009)
Published in Clinical cancer research (01.01.2009)
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Tumor-selective, futile redox cycle-induced bystander effects elicited by NQO1 bioactivatable radiosensitizing drugs in triple-negative breast cancers
Cao, Lifen, Li, Long Shan, Spruell, Christopher, Xiao, Ling, Chakrabarti, Gaurab, Bey, Erik A, Reinicke, Kathryn E, Srougi, Melissa C, Moore, Zachary, Dong, Ying, Vo, Peggy, Kabbani, Wareef, Yang, Chin-Rang, Wang, Xiaoyu, Fattah, Farjana, Morales, Julio C, Motea, Edward A, Bornmann, William G, Yordy, John S, Boothman, David A
Published in Antioxidants & redox signaling (10.07.2014)
Published in Antioxidants & redox signaling (10.07.2014)
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