The Wnt Antagonist Secreted Frizzled-Related Protein-1 Is a Negative Regulator of Trabecular Bone Formation in Adult Mice
Bodine, Peter V. N, Zhao, Weiguang, Kharode, Yogendra P, Bex, Frederick J, Lambert, Andre-Jean, Goad, Mary Beth, Gaur, Tripti, Stein, Gary S, Lian, Jane B, Komm, Barry S
Published in Molecular endocrinology (Baltimore, Md.) (01.05.2004)
Published in Molecular endocrinology (Baltimore, Md.) (01.05.2004)
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High Bone Mass in Mice Expressing a Mutant LRP5 Gene
Babij, Philip, Zhao, Weiguang, Small, Clayton, Kharode, Yogendra, Yaworsky, Paul J, Bouxsein, Mary L, Reddy, Padmalatha S, Bodine, Peter Vn, Robinson, John A, Bhat, Bheem, Marzolf, James, Moran, Robert A, Bex, Frederick
Published in Journal of bone and mineral research (01.06.2003)
Published in Journal of bone and mineral research (01.06.2003)
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Bone anabolic effects of parathyroid hormone are blunted by deletion of the Wnt antagonist secreted frizzled-related protein-1
Bodine, Peter V.N., Seestaller-Wehr, Laura, Kharode, Yogendra P., Bex, Frederick J., Komm, Barry S.
Published in Journal of cellular physiology (01.02.2007)
Published in Journal of cellular physiology (01.02.2007)
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(1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-yl)methanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate
Pelletier, Jeffrey C, Lundquist, Joseph T, Gilbert, Adam M, Alon, Nipa, Bex, Frederick J, Bhat, Bheem M, Bursavich, Mattew G, Coleburn, Valerie E, Felix, Luciana A, Green, Daniel M, Green, Paula, Hauze, Diane B, Kharode, Yogendra P, Lam, Ho-Sun, Lockhead, Susan R, Magolda, Ronald L, Matteo, Jeanne J, Mehlmann, John F, Milligan, Colleen, Murrills, Richard J, Pirrello, Jennifer, Selim, Sally, Sharp, Michael C, Unwalla, Ray J, Vera, Matthew D, Wrobel, Jay E, Yaworsky, Paul, Bodine, Peter V. N
Published in Journal of medicinal chemistry (26.11.2009)
Published in Journal of medicinal chemistry (26.11.2009)
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Systemically administered rhBMP-2 promotes MSC activity and reverses bone and cartilage loss in osteopenic mice
Turgeman, Gadi, Zilberman, Yoram, Zhou, Shuanhu, Kelly, Pam, Moutsatsos, Ioannis K., Kharode, Yogendra P., Borella, Luis E., Bex, Frederick J., Komm, Barry S., Bodine, Peter V.N., Gazit, Dan
Published in Journal of cellular biochemistry (2002)
Published in Journal of cellular biochemistry (2002)
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Structure-based mutation analysis shows the importance of LRP5 β-propeller 1 in modulating Dkk1-mediated inhibition of Wnt signaling
Bhat, Bheem M., Allen, Kristina M., Liu, Wei, Graham, James, Morales, Art, Anisowicz, Anthony, Lam, Ho-Sun, McCauley, Catherine, Coleburn, Valerie, Cain, Michael, Fortier, Eric, Bhat, Ramesh A., Bex, Frederick J., Yaworsky, Paul J.
Published in Gene (15.04.2007)
Published in Gene (15.04.2007)
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Osteogenic effects of a potent Src-over-Abl-selective kinase inhibitor in the mouse
Murrills, Richard J, Fukayama, Shoichi, Boschelli, Frank, Matteo, Jeanne J, Owens, Jane, Golas, Jennifer M, Patel, Dharmesh, Lane, Giovan, Liu, Yao-Bin, Carter, Laura, Jussif, Jason, Spaulding, Vikki, Wang, Yanong D, Boschelli, Diane H, McKew, John C, Li, X Jian, Lockhead, Susan, Milligan, Colleen, Kharode, Yogendra P, Diesl, Veronica, Bai, Yuchen, Follettie, Max, Bex, Frederick J, Komm, Barry, Bodine, Peter V N
Published in The Journal of pharmacology and experimental therapeutics (01.03.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2012)
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A cell-based Dkk1 binding assay reveals roles for extracellular domains of LRP5 in Dkk1 interaction and highlights differences between wild-type and the high bone mass mutant LRP5(G171V)
Murrills, Richard J., Matteo, Jeanne J., Bhat, Bheem M., Coleburn, Valerie E., Allen, Kristina M., Chen, Wei, Damagnez, Veronique, Bhat, Ramesh A., Bex, Frederick J., Bodine, Peter V.N.
Published in Journal of cellular biochemistry (01.12.2009)
Published in Journal of cellular biochemistry (01.12.2009)
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Journal Article
Hit to lead studies on (hetero)arylpyrimidines—Agonists of the canonical Wnt-β-catenin cellular messaging system
Gilbert, Adam M., Bursavich, Matthew G., Alon, Nippa, Bhat, Bheem M., Bex, Frederick J., Cain, Michael, Coleburn, Valerie, Gironda, Virginia, Green, Paula, Hauze, Diane B., Kharode, Yogendra, Krishnamurthy, Girija, Kirisits, Matthew, Lam, Ho-Sun, Liu, Yao-Bin, Lombardi, Sabrina, Matteo, Jeanne, Murrills, Richard, Robinson, John A., Selim, Sally, Sharp, Michael, Unwalla, Raymond, Varadarajan, Usha, Zhao, Weiguang, Yaworsky, Paul J.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
Parathyroid hormone synergizes with non-cyclic AMP pathways to activate the cyclic AMP response element
Murrills, Richard J., Andrews, Jennifer L., Samuel, Rachelle L., Coleburn, Valerie E., Bhat, Bheem M., Bhat, Ramesh A., Bex, Frederick J., Bodine, Peter V.N.
Published in Journal of cellular biochemistry (01.04.2009)
Published in Journal of cellular biochemistry (01.04.2009)
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Journal Article
Wnt/β-Catenin Signaling Is a Normal Physiological Response to Mechanical Loading in Bone
Robinson, John A., Chatterjee-Kishore, Moitreyee, Yaworsky, Paul J., Cullen, Diane M., Zhao, Weiguang, Li, Christine, Kharode, Yogendra, Sauter, Linda, Babij, Philip, Brown, Eugene L., Hill, Andrew A., Akhter, Mohammed P., Johnson, Mark L., Recker, Robert R., Komm, Barry S., Bex, Frederick J.
Published in The Journal of biological chemistry (20.10.2006)
Published in The Journal of biological chemistry (20.10.2006)
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Journal Article
In vitro and in vivo activities of C-terminally truncated PTH peptides reveal a disconnect between cAMP signaling and functional activity
Murrills, Richard J., Matteo, Jeanne J., Samuel, Rachelle L., Andrews, Jennifer L., Bhat, Bheem M., Coleburn, Valerie E., Kharode, Yogendra P., Bex, Frederick J.
Published in Bone (New York, N.Y.) (01.12.2004)
Published in Bone (New York, N.Y.) (01.12.2004)
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Journal Article
Isogenic Human Cell Lines for Drug Discovery: Regulation of Target Gene Expression by Engineered Zinc-Finger Protein Transcription Factors
Liu, Pei-Qi, Tan, Siyuan, Mendel, Matthew C., Murrills, Richard J., Bhat, Bheem M., Schlag, Brian, Samuel, Rachelle, Matteo, Jeanne J., de la Rosa, Ragan, Howes, Katherine, Reik, Andreas, Case, Casey C., Bex, Frederick J., Young, Kathleen, Gregory, Philip D.
Published in Journal of biomolecular screening (01.06.2005)
Published in Journal of biomolecular screening (01.06.2005)
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Journal Article
Wnt/β-Catenin Signaling Is a Normal Physiological Response to Mechanical Loading in Bone
Robinson, John A., Chatterjee-Kishore, Moitreyee, Yaworsky, Paul J., Cullen, Diane M., Zhao, Weiguang, Li, Christine, Kharode, Yogendra, Sauter, Linda, Babij, Philip, Brown, Eugene L., Hill, Andrew A., Akhter, Mohammed P., Johnson, Mark L., Recker, Robert R., Komm, Barry S., Bex, Frederick J.
Published in The Journal of biological chemistry (20.10.2006)
Published in The Journal of biological chemistry (20.10.2006)
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Journal Article
The integrin specificity of human recombinant osteopontin
Caltabiano, Stephen, Hum, Wah-Tung, Attwell, Gwilym J., Gralnick, David N., Budman, Lori J., Cannistraci, AnnaMarie, Bex, Frederick J.
Published in Biochemical pharmacology (15.11.1999)
Published in Biochemical pharmacology (15.11.1999)
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Journal Article
Hit to lead studies on (hetero)arylpyrimidines - Agonists of the canonical Wnt-b-catenin cellular messaging system
Gilbert, Adam M, Bursavich, Matthew G, Alon, Nippa, Bhat, Bheem M, Bex, Frederick J, Cain, Michael, Coleburn, Valerie, Gironda, Virginia, Green, Paula, Hauze, Diane B, Kharode, Yogendra, Krishnamurthy, Girija, Kirisits, Matthew, Lam, Ho-Sun, Liu, Yao-Bin, Lombardi, Sabrina, Matteo, Jeanne, Murrills, Richard, Robinson, John A, Selim, Sally, Sharp, Michael, Unwalla, Raymond, Varadarajan, Usha, Zhao, Weiguang, Yaworsky, Paul J
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Journal Article
1-(4-(Naphthalen-2-yl)pyrimidin-2-yl)piperidin-4-ylmethanamine: A Wingless β-Catenin Agonist That Increases Bone Formation Rate
PELLETIER, Jeffrey C, LUNDQUIST, Joseph T, GREEN, Paula, HAUZE, Diane B, KHARODE, Yogendra P, LAM, Ho-Sun, LOCKHEAD, Susan R, MAGOLDA, Ronald L, MATTEO, Jeanne J, MEHLMANN, John F, MILLIGAN, Colleen, MURRILLS, Richard J, GILBERT, Adam M, PIRRELLO, Jennifer, SELIM, Sally, SHARP, Michael C, UNWALLA, Ray J, VERA, Matthew D, WROBEL, Jay E, YAWORSKY, Paul, BODINE, Peter V. N, ALON, Nipa, BEX, Frederick J, BHAT, Bheem M, BURSAVICH, Mattew G, COLEBURN, Valerie E, FELIX, Luciana A, GREEN, Daniel M
Published in Journal of medicinal chemistry (2009)
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Published in Journal of medicinal chemistry (2009)
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