Synthesis and Structure−Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Metabolic Inactivation: An Antedrug Approach
Procopiou, Panayiotis A, Barrett, Victoria J, Bevan, Nicola J, Biggadike, Keith, Box, Philip C, Butchers, Peter R, Coe, Diane M, Conroy, Richard, Emmons, Amanda, Ford, Alison J, Holmes, Duncan S, Horsley, Helen, Kerr, Fern, Li-Kwai-Cheung, Anne-Marie, Looker, Brian E, Mann, Inderjit S, McLay, Iain M, Morrison, Valerie S, Mutch, Peter J, Smith, Claire E, Tomlin, Paula
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Journal Article
Subcellular distribution of GABAB receptor homo- and hetero-dimers
VILLEMURE, Josée-France, ADAM, Lynda, BEVAN, Nicola J., GEARING, Katy, CHÉNIER, Sébastien, BOUVIER, Michel
Published in Biochemical journal (15.05.2005)
Published in Biochemical journal (15.05.2005)
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Journal Article
Synthesis and Structure−Activity Relationships of Long-acting β2 Adrenergic Receptor Agonists Incorporating Arylsulfonamide Groups
Procopiou, Panayiotis A, Barrett, Victoria J, Bevan, Nicola J, Biggadike, Keith, Butchers, Peter R, Coe, Diane M, Conroy, Richard, Edney, Dean D, Field, Rita N, Ford, Alison J, Guntrip, Stephen B, Looker, Brian E, McLay, Iain M, Monteith, Michael J, Morrison, Valerie S, Mutch, Peter J, Richards, Stephen A, Sasse, Rosemary, Smith, Claire E
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
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Journal Article
The discovery of long-acting saligenin β2 adrenergic receptor agonists incorporating hydantoin or uracil rings
Procopiou, Panayiotis A., Barrett, Victoria J., Bevan, Nicola J., Butchers, Peter R., Conroy, Richard, Emmons, Amanda, Ford, Alison J., Jeulin, Séverine, Looker, Brian E., Lunniss, Gillian E., Morrison, Valerie S., Mutch, Peter J., Perciaccante, Rossana, Ruston, Mark, Smith, Claire E., Somers, Graham
Published in Bioorganic & medicinal chemistry (15.07.2011)
Published in Bioorganic & medicinal chemistry (15.07.2011)
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Journal Article
Abstract 749: Antibody internalization assays for cancer drug discovery
Bevan, Nicola J., Dale, Tim J., Trezise, Derek J.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract 1834: Real-time visualization and quantification of flexible, multi-parameter indicators of cancer cell heath and metabolism using live-cell analysis
Schramm, Cicely L., Rauch, John N., Oupicka, Libuse, Skerlos, Laura A., Bevan, Nicola J., Lovell, Gillian F., Perez-Garrido, Sandra, Filonov, Grigory S., Chen, Yong X., Kovalenko, Ilya, Foltin, Susan, Campwala, Hinnah, Dale, Timothy J., Appledorn, Daniel M.
Published in Cancer research (Chicago, Ill.) (15.08.2020)
Published in Cancer research (Chicago, Ill.) (15.08.2020)
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Abstract 5030: Development and optimization of Matrigel-based multi-spheroid 3D tumor assays using real-time live-cell analysis
Patel, Kalpana, Oliver, Miniver, Holtz, Nevine, Jackson, Tim, Dana, Nicholas, Lovell, Gillian, Bevan, Nicola J., Dale, Tim J., Trezise, Derek J.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Synthesis and Structure-Activity Relationships of Long-acting beta(2) Adrenergic Receptor Agonists Incorporating Metabolic Inactivation: An Antedrug Approach
Procopiou, Panayiotis A., Barrett, Victoria J., Bevan, Nicola J., Biggadike, Keith, Box, Philip C., Butchers, Peter R., Coe, Diane M., Conroy, Richard, Emmons, Amanda, Ford, Alison J., Holmes, Duncan S., Horsley, Helen, Kerr, Fern, Li-Kwai-Cheung, Anne-Marie, Looker, Brian E., Mann, Inderjit S., McLay, Iain M., Morrison, Valerie S., Mutch, Peter J., Smith, Claire E., Tomlin, Paula
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Journal Article
Synthesis and Structure-Activity Relationships of Long-acting beta(2) Adrenergic Receptor Agonists Incorporating Arylsulfonamide Groups
Procopiou, Panayiotis A., Barrett, Victoria J., Bevan, Nicola J., Biggadike, Keith, Butchers, Peter R., Coe, Diane M., Conroy, Richard, Edney, Dean D., Field, Rita N., Ford, Alison J., Guntrip, Stephen B., Looker, Brian E., McLay, Iain M., Monteith, Michael J., Morrison, Valerie S., Mutch, Peter J., Richards, Stephen A., Sasse, Rosemary, Smith, Claire E.
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
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Journal Article
Subcellular distribution of GABA(B) receptor homo- and hetero-dimers
Villemure, Josée-France, Adam, Lynda, Bevan, Nicola J, Gearing, Katy, Chénier, Sébastien, Bouvier, Michel
Published in Biochemical journal (15.05.2005)
Published in Biochemical journal (15.05.2005)
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Journal Article
The discovery of long-acting saligenin beta sub(2 adrenergic receptor agonists incorporating hydantoin or uracil rings)
Procopiou, Panayiotis A, Barrett, Victoria J, Bevan, Nicola J, Butchers, Peter R, Conroy, Richard, Emmons, Amanda, d, Alison J, Jeulin, Severine, Looker, Brian E, Lunniss, Gillian E, Morrison, Valerie S, Mutch, Peter J, Perciaccante, Rossana, Ruston, Mark, Smith, Claire E, Somers, Graham, Xepfqmjboitfns-Sanmltnesa-N, InChiKey
Published in Bioorganic & medicinal chemistry (15.07.2011)
Published in Bioorganic & medicinal chemistry (15.07.2011)
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Journal Article
Synthesis and Structure−Activity Relationships of Long-acting β 2 Adrenergic Receptor Agonists Incorporating Metabolic Inactivation: An Antedrug Approach
Procopiou, Panayiotis A., Barrett, Victoria J., Bevan, Nicola J., Biggadike, Keith, Box, Philip C., Butchers, Peter R., Coe, Diane M., Conroy, Richard, Emmons, Amanda, Ford, Alison J., Holmes, Duncan S., Horsley, Helen, Kerr, Fern, Li-Kwai-Cheung, Anne-Marie, Looker, Brian E., Mann, Inderjit S., McLay, Iain M., Morrison, Valerie S., Mutch, Peter J., Smith, Claire E., Tomlin, Paula
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
Get full text
Journal Article
Synthesis and Structure−Activity Relationships of Long-acting β 2 Adrenergic Receptor Agonists Incorporating Arylsulfonamide Groups
Procopiou, Panayiotis A., Barrett, Victoria J., Bevan, Nicola J., Biggadike, Keith, Butchers, Peter R., Coe, Diane M., Conroy, Richard, Edney, Dean D., Field, Rita N., Ford, Alison J., Guntrip, Stephen B., Looker, Brian E., McLay, Iain M., Monteith, Michael J., Morrison, Valerie S., Mutch, Peter J., Richards, Stephen A., Sasse, Rosemary, Smith, Claire E.
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
Get full text
Journal Article
Subcellular distribution of GABA sub(B) receptor homo- and hetero-dimers
Villemure, Josee-France, Adam, Lynda, Bevan, Nicola J, Gearing, Katy, Chenier, Sebastien, Bouvier, Michel
Published in Biochemical journal (15.05.2005)
Published in Biochemical journal (15.05.2005)
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Journal Article
Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating metabolic inactivation: an antedrug approach
Procopiou, Panayiotis A, Barrett, Victoria J, Bevan, Nicola J, Biggadike, Keith, Box, Philip C, Butchers, Peter R, Coe, Diane M, Conroy, Richard, Emmons, Amanda, Ford, Alison J, Holmes, Duncan S, Horsley, Helen, Kerr, Fern, Li-Kwai-Cheung, Anne-Marie, Looker, Brian E, Mann, Inderjit S, McLay, Iain M, Morrison, Valerie S, Mutch, Peter J, Smith, Claire E, Tomlin, Paula
Published in Journal of medicinal chemistry (10.06.2010)
Published in Journal of medicinal chemistry (10.06.2010)
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Journal Article
Synthesis and structure-activity relationships of long-acting beta2 adrenergic receptor agonists incorporating arylsulfonamide groups
Procopiou, Panayiotis A, Barrett, Victoria J, Bevan, Nicola J, Biggadike, Keith, Butchers, Peter R, Coe, Diane M, Conroy, Richard, Edney, Dean D, Field, Rita N, Ford, Alison J, Guntrip, Stephen B, Looker, Brian E, McLay, Iain M, Monteith, Michael J, Morrison, Valerie S, Mutch, Peter J, Richards, Stephen A, Sasse, Rosemary, Smith, Claire E
Published in Journal of medicinal chemistry (23.04.2009)
Published in Journal of medicinal chemistry (23.04.2009)
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Journal Article